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DRUG:
patritumab deruxtecan (U3-1402)
i
Other names:
U3-1402, U3 1402, U3-1402a, U31402, Patritumab-DX-8951 conjugate, HER3-DXd, MK-1022
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News alerts, weekly reports and conference planners
Associations
(28)
News
Trials
Company:
Daiichi Sankyo, Merck (MSD)
Drug class:
Topoisomerase I inhibitor, HER3-targeted antibody-drug conjugate
Related drugs:
‹
fam-trastuzumab deruxtecan-nxki (90)
irinotecan (48)
sacituzumab govitecan-hziy (17)
topotecan (16)
SHR-A1811 (15)
DS-1062a (11)
AZD8205 (5)
DS-7300 (5)
AMB302 (4)
BNT323 (4)
DB-1310 (4)
DM002 (4)
BL-M07D1 (3)
DS-6157 (3)
HRA00129-C004 (3)
nanoliposomal irinotecan (3)
PLX038 (3)
MK-2870 (3)
ABBV-400 (3)
CUSP06 (2)
DAN-222 (2)
DM005 (2)
PRO1102 (2)
SSH20 (2)
IMMU-130 (2)
AZD9592 (2)
AMT-562 (1)
AZD5335 (1)
BAT8008 (1)
BL-M02D1 (1)
camptothecin nanosomal (1)
DAN-311 (1)
ELU001 (1)
ESG401 (1)
HMBD-501 (1)
IMMU-140 (1)
IT-141 (1)
OBI-992 (1)
SGN-35C (1)
SGN-CD30C (1)
STRO-003 (1)
ZW191 (1)
ZW220 (1)
ZW251 (1)
BL-B01D1 (1)
PRO1184 (1)
ABBV-706 (0)
BAT8007 (0)
BAT8010 (0)
BL-M11D1 (0)
BNT324 (0)
BNT326 (0)
CEB-01 (0)
belotecan (0)
DS-3939 (0)
FZ-AD004 (0)
GSK5733584 (0)
HA-irinotecan (0)
HLX43 (0)
HS-20093 (0)
IBI-354 (0)
ICAM‑1 ADC (0)
JSKN003 (0)
LMP744 (0)
lentinan (0)
TLC388 (0)
M9140 (0)
MBK-103 (0)
MHB036C (0)
MHB088C (0)
MK-1200 (0)
NK012 (0)
etirinotecan pegol (0)
PRO1160 (0)
SHR-A1921 (0)
SHR-A2009 (0)
TQB2102 (0)
YL201 (0)
CBX-12 (0)
EP0057 (0)
LMP400 (0)
HR070803 (0)
irinotecan liposomal (0)
LY01616 (0)
FF-10850 (0)
PEN-866 (0)
DS-6000 (0)
simmitecan (0)
topotecan episcleral (0)
ORM-5029 (2)
fam-trastuzumab deruxtecan-nxki (90)
irinotecan (48)
sacituzumab govitecan-hziy (17)
topotecan (16)
SHR-A1811 (15)
DS-1062a (11)
AZD8205 (5)
DS-7300 (5)
AMB302 (4)
BNT323 (4)
DB-1310 (4)
DM002 (4)
BL-M07D1 (3)
DS-6157 (3)
HRA00129-C004 (3)
nanoliposomal irinotecan (3)
PLX038 (3)
MK-2870 (3)
ABBV-400 (3)
CUSP06 (2)
DAN-222 (2)
DM005 (2)
PRO1102 (2)
SSH20 (2)
IMMU-130 (2)
AZD9592 (2)
AMT-562 (1)
AZD5335 (1)
BAT8008 (1)
BL-M02D1 (1)
camptothecin nanosomal (1)
DAN-311 (1)
ELU001 (1)
ESG401 (1)
HMBD-501 (1)
IMMU-140 (1)
IT-141 (1)
OBI-992 (1)
SGN-35C (1)
SGN-CD30C (1)
STRO-003 (1)
ZW191 (1)
ZW220 (1)
ZW251 (1)
BL-B01D1 (1)
PRO1184 (1)
ABBV-706 (0)
BAT8007 (0)
BAT8010 (0)
BL-M11D1 (0)
BNT324 (0)
BNT326 (0)
CEB-01 (0)
belotecan (0)
DS-3939 (0)
FZ-AD004 (0)
GSK5733584 (0)
HA-irinotecan (0)
HLX43 (0)
HS-20093 (0)
IBI-354 (0)
ICAM‑1 ADC (0)
JSKN003 (0)
LMP744 (0)
lentinan (0)
TLC388 (0)
M9140 (0)
MBK-103 (0)
MHB036C (0)
MHB088C (0)
MK-1200 (0)
NK012 (0)
etirinotecan pegol (0)
PRO1160 (0)
SHR-A1921 (0)
SHR-A2009 (0)
TQB2102 (0)
YL201 (0)
CBX-12 (0)
EP0057 (0)
LMP400 (0)
HR070803 (0)
irinotecan liposomal (0)
LY01616 (0)
FF-10850 (0)
PEN-866 (0)
DS-6000 (0)
simmitecan (0)
topotecan episcleral (0)
ORM-5029 (2)
›
Associations
(28)
News
Trials
VERI cancer hierarchy
Reset Filters
EGFR mutation
Non Small Cell Lung Cancer
EGFR mutation
Non Small Cell Lung Cancer
U3-1402
Sensitive: B - Late Trials
U3-1402
Sensitive
:
B
U3-1402
Sensitive: B - Late Trials
U3-1402
Sensitive
:
B
ERBB3 expression
Colorectal Cancer
ERBB3 expression
Colorectal Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
ERBB3 expression
Breast Cancer
ERBB3 expression
Breast Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
EGFR L858R
Non Small Cell Lung Cancer
EGFR L858R
Non Small Cell Lung Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
EGFR exon 19 deletion
Non Small Cell Lung Cancer
EGFR exon 19 deletion
Non Small Cell Lung Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
HR positive
HER2 Negative Breast Cancer
HR positive
HER2 Negative Breast Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
ALK fusion
Non Small Cell Lung Cancer
ALK fusion
Non Small Cell Lung Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
ROS1 fusion
Non Small Cell Lung Cancer
ROS1 fusion
Non Small Cell Lung Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
HER-2 negative
Triple Negative Breast Cancer
HER-2 negative
Triple Negative Breast Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
HER-2 positive
HER2 Positive Breast Cancer
HER-2 positive
HER2 Positive Breast Cancer
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
U3-1402
Sensitive: C2 – Inclusion Criteria
U3-1402
Sensitive
:
C2
EGFR C797S
Non Small Cell Lung Cancer
EGFR C797S
Non Small Cell Lung Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
MET amplification
Non Small Cell Lung Cancer
MET amplification
Non Small Cell Lung Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
HER-2 mutation
Non Small Cell Lung Cancer
HER-2 mutation
Non Small Cell Lung Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
BRAF fusion
Non Small Cell Lung Cancer
BRAF fusion
Non Small Cell Lung Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
PIK3CA mutation
Non Small Cell Lung Cancer
PIK3CA mutation
Non Small Cell Lung Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
HR positive + ERBB3 underexpression
HER2 Negative Breast Cancer
HR positive + ERBB3 underexpression
HER2 Negative Breast Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
HR positive + ERBB3 overexpression
HER2 Negative Breast Cancer
HR positive + ERBB3 overexpression
HER2 Negative Breast Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
ERBB3 overexpression
Breast Cancer
ERBB3 overexpression
Breast Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
KRAS mutation
Non Small Cell Lung Cancer
KRAS mutation
Non Small Cell Lung Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
EGFR exon 20 insertion
Non Small Cell Lung Cancer
EGFR exon 20 insertion
Non Small Cell Lung Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
HR positive + HER-2 underexpression
Breast Cancer
HR positive + HER-2 underexpression
Breast Cancer
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
U3-1402
Sensitive: C3 – Early Trials
U3-1402
Sensitive
:
C3
NRAS mutation
Non Small Cell Lung Cancer
NRAS mutation
Non Small Cell Lung Cancer
U3-1402
Sensitive: C4 – Case Studies
U3-1402
Sensitive
:
C4
U3-1402
Sensitive: C4 – Case Studies
U3-1402
Sensitive
:
C4
EGFR mutation
Non Small Cell Lung Cancer
EGFR mutation
Non Small Cell Lung Cancer
osimertinib + U3-1402
Sensitive: D – Preclinical
osimertinib + U3-1402
Sensitive
:
D
osimertinib + U3-1402
Sensitive: D – Preclinical
osimertinib + U3-1402
Sensitive
:
D
ERBB3 overexpression
Colorectal Cancer
ERBB3 overexpression
Colorectal Cancer
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
ERBB3 expression
Melanoma
ERBB3 expression
Melanoma
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
ERBB3 expression
Estrogen Receptor Positive Breast Cancer
ERBB3 expression
Estrogen Receptor Positive Breast Cancer
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
ERBB3 mutation
Breast Cancer
ERBB3 mutation
Breast Cancer
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
U3-1402
Sensitive: D – Preclinical
U3-1402
Sensitive
:
D
ERBB3 expression
Estrogen Receptor Positive Breast Cancer
ERBB3 expression
Estrogen Receptor Positive Breast Cancer
U3-1402 + BAY 1895344
Sensitive: D – Preclinical
U3-1402 + BAY 1895344
Sensitive
:
D
U3-1402 + BAY 1895344
Sensitive: D – Preclinical
U3-1402 + BAY 1895344
Sensitive
:
D
^
^
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