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DRUG:
dasatinib
i
Other names:
BMS 354825, BMS-354825, BMS354825
Contact us
to learn more about our Premium Content:
News alerts, weekly reports and conference planners
Associations
(214)
News
Twitter
Trials
Company:
Generic mfg.
Drug class:
c-KIT inhibitor, Bcr-abl tyrosine kinase inhibitor, Src kinase inhibitor, EphA2 receptor antagonist, PDGFR β antagonist
Related drugs:
‹
imatinib (165)
sunitinib (128)
lenvatinib (82)
midostaurin (41)
YD312 (21)
ripretinib (10)
MLN518 (8)
SU5614 (6)
pexidartinib (6)
AG-1296 (1)
flumatinib (1)
M4205 (1)
MP470 (1)
PLX9486 (1)
CS 2164 (1)
E7050 (1)
nilotinib (65)
bosutinib (44)
olverembatinib (7)
asciminib (7)
INNO-406 (3)
PF-114 (1)
SCO - 088 (1)
TPX-0022 (8)
AZD0530 (7)
BAL3833 (4)
NXP900 (2)
PP2 (2)
TPX-0046 (2)
ALW-II-41-27 (2)
BCY6033 (1)
imatinib (165)
sunitinib (128)
lenvatinib (82)
midostaurin (41)
YD312 (21)
ripretinib (10)
MLN518 (8)
SU5614 (6)
pexidartinib (6)
AG-1296 (1)
flumatinib (1)
M4205 (1)
MP470 (1)
PLX9486 (1)
CS 2164 (1)
E7050 (1)
nilotinib (65)
bosutinib (44)
olverembatinib (7)
asciminib (7)
INNO-406 (3)
PF-114 (1)
SCO - 088 (1)
TPX-0022 (8)
AZD0530 (7)
BAL3833 (4)
NXP900 (2)
PP2 (2)
TPX-0046 (2)
ALW-II-41-27 (2)
BCY6033 (1)
›
Associations
(214)
News
Twitter
Trials
Reset Filters
VERI cancer hierarchy
x
x
x
x
HER-2 positive
HER2 Positive Breast Cancer
HER-2 positive
HER2 Positive Breast Cancer
dasatinib + lapatinib
Sensitive: D – Preclinical
PLoS One - 1 week (New D)
dasatinib + lapatinib
Sensitive
:
D
PLoS One - 1wk
dasatinib + lapatinib
Sensitive: D – Preclinical
PLoS One - 1 week
dasatinib + lapatinib
Sensitive
:
D
PLoS One - 1 week - (New D)
BCR-ABL1 fusion
Chronic Myeloid Leukemia
BCR-ABL1 fusion
Chronic Myeloid Leukemia
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
BCR-ABL1 fusion
Acute Lymphocytic Leukemia
BCR-ABL1 fusion
Acute Lymphocytic Leukemia
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
dasatinib
Sensitive: A1 - Approval
dasatinib
Sensitive
:
A1
BCR-ABL1 V299L
Acute Lymphocytic Leukemia
BCR-ABL1 V299L
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317I
Acute Lymphocytic Leukemia
BCR-ABL1 F317I
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 T315I
Acute Lymphocytic Leukemia
BCR-ABL1 T315I
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 T315I
Chronic Myeloid Leukemia
BCR-ABL1 T315I
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
No biomarker
Chronic Myeloid Leukemia
No biomarker
Chronic Myeloid Leukemia
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
PDGFRA fusion
Childhood B Acute Lymphoblastic Leukemia
PDGFRA fusion
Childhood B Acute Lymphoblastic Leukemia
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
ABL2 fusion
Childhood B Acute Lymphoblastic Leukemia
ABL2 fusion
Childhood B Acute Lymphoblastic Leukemia
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
FGFR fusion
Childhood B Acute Lymphoblastic Leukemia
FGFR fusion
Childhood B Acute Lymphoblastic Leukemia
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
No biomarker
Chordoma
No biomarker
Chordoma
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
BCR-ABL1 F317L
Chronic Myeloid Leukemia
BCR-ABL1 F317L
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
PDGFRA D842V
Gastrointestinal Stromal Tumor
PDGFRA D842V
Gastrointestinal Stromal Tumor
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
ABL1 fusion
Childhood B Acute Lymphoblastic Leukemia
ABL1 fusion
Childhood B Acute Lymphoblastic Leukemia
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
PDGFRB fusion
Childhood B Acute Lymphoblastic Leukemia
PDGFRB fusion
Childhood B Acute Lymphoblastic Leukemia
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
BCR-ABL1 fusion
B Acute Lymphoblastic Leukemia
BCR-ABL1 fusion
B Acute Lymphoblastic Leukemia
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
BCR-ABL1 V299L
Chronic Myeloid Leukemia
BCR-ABL1 V299L
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 T315A
Chronic Myeloid Leukemia
BCR-ABL1 T315A
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317I
Chronic Myeloid Leukemia
BCR-ABL1 F317I
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317V
Chronic Myeloid Leukemia
BCR-ABL1 F317V
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317C
Chronic Myeloid Leukemia
BCR-ABL1 F317C
Chronic Myeloid Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317L
Acute Lymphocytic Leukemia
BCR-ABL1 F317L
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317C
Acute Lymphocytic Leukemia
BCR-ABL1 F317C
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 F317V
Acute Lymphocytic Leukemia
BCR-ABL1 F317V
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
BCR-ABL1 T315A
Acute Lymphocytic Leukemia
BCR-ABL1 T315A
Acute Lymphocytic Leukemia
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
dasatinib
Resistant: A2 - Guideline
dasatinib
Resistant
:
A2
No biomarker
Sarcoma
No biomarker
Sarcoma
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
dasatinib
Sensitive: A2 - Guideline
dasatinib
Sensitive
:
A2
BCR-ABL1 L248V
Chronic Myeloid Leukemia
BCR-ABL1 L248V
Chronic Myeloid Leukemia
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
BCR-ABL1 G250E
Chronic Myeloid Leukemia
BCR-ABL1 G250E
Chronic Myeloid Leukemia
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
BCR-ABL1 Q252H
Chronic Myeloid Leukemia
BCR-ABL1 Q252H
Chronic Myeloid Leukemia
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
BCR-ABL1 E255K
Chronic Myeloid Leukemia
BCR-ABL1 E255K
Chronic Myeloid Leukemia
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
BCR-ABL1 F359C
Chronic Myeloid Leukemia
BCR-ABL1 F359C
Chronic Myeloid Leukemia
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
BCR-ABL1 Y253H
Chronic Myeloid Leukemia
BCR-ABL1 Y253H
Chronic Myeloid Leukemia
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
dasatinib
Sensitive: B - Late Trials
dasatinib
Sensitive
:
B
^
^
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