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DRUG CLASS:
Bcl-xL inhibitor
DRUG CLASS:
Bcl-xL inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
ABT 263 (19)
APG-1252 (8)
A-1331852 (6)
APG1244 (2)
AT 101 (1)
ABBV-637 (0)
AZD0466 (0)
AZD4320 (0)
LP-118 (0)
ABBV-155 (0)
ONT-701 (0)
ABT 263 (19)
APG-1252 (8)
A-1331852 (6)
APG1244 (2)
AT 101 (1)
ABBV-637 (0)
AZD0466 (0)
AZD4320 (0)
LP-118 (0)
ABBV-155 (0)
ONT-701 (0)
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Associations
(36)
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Trials
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EGFR L858R
Non Small Cell Lung Cancer
EGFR L858R
Non Small Cell Lung Cancer
osimertinib + ABT 263
Sensitive: C2 – Inclusion Criteria
osimertinib + ABT 263
Sensitive
:
C2
osimertinib + ABT 263
Sensitive: C2 – Inclusion Criteria
osimertinib + ABT 263
Sensitive
:
C2
EGFR T790M
Non Small Cell Lung Cancer
EGFR T790M
Non Small Cell Lung Cancer
osimertinib + ABT 263
Sensitive: C2 – Inclusion Criteria
osimertinib + ABT 263
Sensitive
:
C2
osimertinib + ABT 263
Sensitive: C2 – Inclusion Criteria
osimertinib + ABT 263
Sensitive
:
C2
BRAF mutation
Melanoma
BRAF mutation
Melanoma
trametinib + dabrafenib + ABT 263
Sensitive: C2 – Inclusion Criteria
trametinib + dabrafenib + ABT 263
Sensitive
:
C2
trametinib + dabrafenib + ABT 263
Sensitive: C2 – Inclusion Criteria
trametinib + dabrafenib + ABT 263
Sensitive
:
C2
EGFR T790M
Non Small Cell Lung Cancer
EGFR T790M
Non Small Cell Lung Cancer
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
EGFR mutation
Non Small Cell Lung Cancer
EGFR mutation
Non Small Cell Lung Cancer
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
TP53 mutation
Acute Myelogenous Leukemia
TP53 mutation
Acute Myelogenous Leukemia
A-1331852
Sensitive: C3 – Early Trials
A-1331852
Sensitive
:
C3
A-1331852
Sensitive: C3 – Early Trials
A-1331852
Sensitive
:
C3
TP53 mutation
Acute Myelogenous Leukemia
TP53 mutation
Acute Myelogenous Leukemia
ABT 263
Sensitive: C3 – Early Trials
ABT 263
Sensitive
:
C3
ABT 263
Sensitive: C3 – Early Trials
ABT 263
Sensitive
:
C3
BCL2L1 overexpression
Non Small Cell Lung Cancer
BCL2L1 overexpression
Non Small Cell Lung Cancer
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
TP53 mutation
Non Small Cell Lung Cancer
TP53 mutation
Non Small Cell Lung Cancer
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
osimertinib + APG-1252
Sensitive: C3 – Early Trials
osimertinib + APG-1252
Sensitive
:
C3
STRN-ALK rearrangement
Mesothelioma
STRN-ALK rearrangement
Mesothelioma
ABT 263
Sensitive: D – Preclinical
ABT 263
Sensitive
:
D
ABT 263
Sensitive: D – Preclinical
ABT 263
Sensitive
:
D
KRAS mutation
Non Small Cell Lung Cancer
KRAS mutation
Non Small Cell Lung Cancer
trametinib + ABT 263
Sensitive: D – Preclinical
trametinib + ABT 263
Sensitive
:
D
trametinib + ABT 263
Sensitive: D – Preclinical
trametinib + ABT 263
Sensitive
:
D
EGFR T790M
Non Small Cell Lung Cancer
EGFR T790M
Non Small Cell Lung Cancer
APG-1252
Sensitive: D – Preclinical
APG-1252
Sensitive
:
D
APG-1252
Sensitive: D – Preclinical
APG-1252
Sensitive
:
D
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