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DRUG:
Tafinlar (dabrafenib)
i
Other names:
GSK2118436, GSK436, 2118436, DRB 436, GSK-2118436A, GSK2118436A, GSK-2118436, GSK 2118436
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News alerts, weekly reports and conference planners
Associations
(201)
News
Twitter
Trials
Company:
Novartis
Drug class:
BRAF inhibitor
Related drugs:
‹
vemurafenib (200)
PLX4720 (64)
encorafenib (61)
VS-6766 (27)
FORE-8394 (20)
RAF265 (7)
GDC 0879 (6)
RXDX-105 (5)
ERAS-254 (5)
ABM-1310 (3)
HI-511 (1)
SB-590885 (1)
BGB-3245 (1)
PF-07284890 (1)
AFX-1251 (0)
ASN003 (0)
AZ304 (0)
BDTX-4933 (0)
BMS-908662 (0)
DP-2514 (0)
DP-3346 (0)
EBI-907 (0)
EBI-945 (0)
PF-07799933 (0)
RG6344 (0)
RO5212054 (0)
RX208 (0)
NSC311152 (0)
vemurafenib (200)
PLX4720 (64)
encorafenib (61)
VS-6766 (27)
FORE-8394 (20)
RAF265 (7)
GDC 0879 (6)
RXDX-105 (5)
ERAS-254 (5)
ABM-1310 (3)
HI-511 (1)
SB-590885 (1)
BGB-3245 (1)
PF-07284890 (1)
AFX-1251 (0)
ASN003 (0)
AZ304 (0)
BDTX-4933 (0)
BMS-908662 (0)
DP-2514 (0)
DP-3346 (0)
EBI-907 (0)
EBI-945 (0)
PF-07799933 (0)
RG6344 (0)
RO5212054 (0)
RX208 (0)
NSC311152 (0)
›
Associations
(201)
News
Twitter
Trials
VERI cancer hierarchy
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BRAF V600E
Melanoma
BRAF V600E
Melanoma
trametinib + dabrafenib
Sensitive: A1 - Approval
ASCO 2023 - 1 week (New C3)
trametinib + dabrafenib
Sensitive
:
A1
ASCO 2023 - 1wk
trametinib + dabrafenib
Sensitive: A1 - Approval
ASCO 2023 - 1 week
trametinib + dabrafenib
Sensitive
:
A1
ASCO 2023 - 1 week - (New C3)
BRAF V600K
Melanoma
BRAF V600K
Melanoma
trametinib + dabrafenib
Sensitive: A1 - Approval
ASCO 2023 - 1 week (New C3)
trametinib + dabrafenib
Sensitive
:
A1
ASCO 2023 - 1wk
trametinib + dabrafenib
Sensitive: A1 - Approval
ASCO 2023 - 1 week
trametinib + dabrafenib
Sensitive
:
A1
ASCO 2023 - 1 week - (New C3)
BRAF V600
Melanoma
BRAF V600
Melanoma
trametinib + dabrafenib
Sensitive: A1 - Approval
ASCO 2023 - 1 week (New C3)
trametinib + dabrafenib
Sensitive
:
A1
ASCO 2023 - 1wk
trametinib + dabrafenib
Sensitive: A1 - Approval
ASCO 2023 - 1 week
trametinib + dabrafenib
Sensitive
:
A1
ASCO 2023 - 1 week - (New C3)
BRAF mutation
Melanoma
BRAF mutation
Melanoma
trametinib + dabrafenib + ABT 263
Sensitive: C3 – Early Trials
ASCO 2023 - 1 week (New C3)
trametinib + dabrafenib + ABT 263
Sensitive
:
C3
ASCO 2023 - 1wk
trametinib + dabrafenib + ABT 263
Sensitive: C3 – Early Trials
ASCO 2023 - 1 week
trametinib + dabrafenib + ABT 263
Sensitive
:
C3
ASCO 2023 - 1 week - (New C3)
BRAF mutation
Melanoma
BRAF mutation
Melanoma
dabrafenib + ivosidenib
Sensitive: D – Preclinical
ASCO 2023 - 1 week (New D)
dabrafenib + ivosidenib
Sensitive
:
D
ASCO 2023 - 1wk
dabrafenib + ivosidenib
Sensitive: D – Preclinical
ASCO 2023 - 1 week
dabrafenib + ivosidenib
Sensitive
:
D
ASCO 2023 - 1 week - (New D)
BRAF V600
Non Small Cell Lung Cancer
BRAF V600
Non Small Cell Lung Cancer
trametinib + dabrafenib
Sensitive: A1 - Approval
Precision Oncology News - 3 weeks (New A2)
trametinib + dabrafenib
Sensitive
:
A1
Precision Oncology News - 3wk
trametinib + dabrafenib
Sensitive: A1 - Approval
Precision Oncology News - 3 weeks
trametinib + dabrafenib
Sensitive
:
A1
Precision Oncology News - 3 weeks - (New A2)
BRAF V600E
Melanoma
BRAF V600E
Melanoma
dabrafenib
Sensitive: A1 - Approval
dabrafenib
Sensitive
:
A1
dabrafenib
Sensitive: A1 - Approval
dabrafenib
Sensitive
:
A1
BRAF V600E
Non Small Cell Lung Cancer
BRAF V600E
Non Small Cell Lung Cancer
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
BRAF V600E
Thyroid Gland Anaplastic Carcinoma
BRAF V600E
Thyroid Gland Anaplastic Carcinoma
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
BRAF V600E
Thyroid Gland Anaplastic Carcinoma
BRAF V600E
Thyroid Gland Anaplastic Carcinoma
dabrafenib
Sensitive: A1 - Approval
dabrafenib
Sensitive
:
A1
dabrafenib
Sensitive: A1 - Approval
dabrafenib
Sensitive
:
A1
BRAF V600
Melanoma
BRAF V600
Melanoma
dabrafenib
Sensitive: A1 - Approval
dabrafenib
Sensitive
:
A1
dabrafenib
Sensitive: A1 - Approval
dabrafenib
Sensitive
:
A1
BRAF V600E
Solid Tumor
BRAF V600E
Solid Tumor
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
BRAF V600E
Glioma
BRAF V600E
Glioma
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
trametinib + dabrafenib
Sensitive: A1 - Approval
trametinib + dabrafenib
Sensitive
:
A1
BRAF V600E
Non Small Cell Lung Cancer
BRAF V600E
Non Small Cell Lung Cancer
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
BRAF V600E
Glioblastoma
BRAF V600E
Glioblastoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Ganglioglioma
BRAF V600E
Ganglioglioma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Neuroendocrine Tumor
BRAF V600E
Neuroendocrine Tumor
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Cutaneous Melanoma
BRAF V600E
Cutaneous Melanoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Biliary Tract Cancer
BRAF V600E
Biliary Tract Cancer
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Astrocytoma
BRAF V600E
Astrocytoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF mutation
Melanoma
BRAF mutation
Melanoma
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
BRAF V600E
Astrocytoma
BRAF V600E
Astrocytoma
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
BRAF V600E
Ganglioglioma
BRAF V600E
Ganglioglioma
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
BRAF V600
Cutaneous Melanoma
BRAF V600
Cutaneous Melanoma
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
BRAF V600K
Cutaneous Melanoma
BRAF V600K
Cutaneous Melanoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Colorectal Cancer
BRAF V600E
Colorectal Cancer
trametinib + dabrafenib + panitumumab
Sensitive: A2 - Guideline
trametinib + dabrafenib + panitumumab
Sensitive
:
A2
trametinib + dabrafenib + panitumumab
Sensitive: A2 - Guideline
trametinib + dabrafenib + panitumumab
Sensitive
:
A2
BRAF V600K
Melanoma
BRAF V600K
Melanoma
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
BRAF V600E
Colorectal Cancer
BRAF V600E
Colorectal Cancer
cetuximab + trametinib + dabrafenib
Sensitive: A2 - Guideline
cetuximab + trametinib + dabrafenib
Sensitive
:
A2
cetuximab + trametinib + dabrafenib
Sensitive: A2 - Guideline
cetuximab + trametinib + dabrafenib
Sensitive
:
A2
BRAF V600
Cutaneous Melanoma
BRAF V600
Cutaneous Melanoma
pembrolizumab + dabrafenib
Sensitive: A2 - Guideline
pembrolizumab + dabrafenib
Sensitive
:
A2
pembrolizumab + dabrafenib
Sensitive: A2 - Guideline
pembrolizumab + dabrafenib
Sensitive
:
A2
BRAF V600E
Cutaneous Melanoma
BRAF V600E
Cutaneous Melanoma
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
dabrafenib
Sensitive: A2 - Guideline
dabrafenib
Sensitive
:
A2
BRAF V600E
Ovarian Serous Adenocarcinoma
BRAF V600E
Ovarian Serous Adenocarcinoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
IDH2 mutation + BRAF V600E
Astrocytoma
IDH2 mutation + BRAF V600E
Astrocytoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
IDH1 mutation + BRAF V600E
Astrocytoma
IDH1 mutation + BRAF V600E
Astrocytoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
IDH2 mutation + Chr del(1p) + Chr del(19q) + BRAF V600E
Oligodendroglioma
IDH2 mutation + Chr del(1p) + Chr del(19q) + BRAF V600E
Oligodendroglioma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
IDH1 mutation + Chr del(1p) + Chr del(19q) + BRAF V600E
Oligodendroglioma
IDH1 mutation + Chr del(1p) + Chr del(19q) + BRAF V600E
Oligodendroglioma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Pancreatic Adenocarcinoma
BRAF V600E
Pancreatic Adenocarcinoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Ampulla of Vater Carcinoma
BRAF V600E
Ampulla of Vater Carcinoma
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
BRAF V600E
Salivary Gland Cancer
BRAF V600E
Salivary Gland Cancer
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
trametinib + dabrafenib
Sensitive: A2 - Guideline
trametinib + dabrafenib
Sensitive
:
A2
^
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