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DRUG CLASS:
IDH2 inhibitor
DRUG CLASS:
IDH2 inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
enasidenib (16)
vorasidenib (6)
TQB3455 (2)
LY3410738 (1)
NMS-173 (1)
AGI-6780 (0)
SH1573 (0)
HMPL-306 (0)
enasidenib (16)
vorasidenib (6)
TQB3455 (2)
LY3410738 (1)
NMS-173 (1)
AGI-6780 (0)
SH1573 (0)
HMPL-306 (0)
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Associations
(27)
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VERI cancer hierarchy
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IDH2 mutation
Acute Myelogenous Leukemia
IDH2 mutation
Acute Myelogenous Leukemia
enasidenib
Sensitive: A1 - Approval
enasidenib
Sensitive
:
A1
enasidenib
Sensitive: A1 - Approval
enasidenib
Sensitive
:
A1
IDH2 mutation
Oligodendroglioma
IDH2 mutation
Oligodendroglioma
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
IDH2 mutation
Astrocytoma
IDH2 mutation
Astrocytoma
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
IDH1 mutation
Astrocytoma
IDH1 mutation
Astrocytoma
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
IDH1 mutation
Oligodendroglioma
IDH1 mutation
Oligodendroglioma
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
vorasidenib
Sensitive: A1 - Approval
vorasidenib
Sensitive
:
A1
IDH2 R172
Acute Myelogenous Leukemia
IDH2 R172
Acute Myelogenous Leukemia
enasidenib
Sensitive: B - Late Trials
enasidenib
Sensitive
:
B
enasidenib
Sensitive: B - Late Trials
enasidenib
Sensitive
:
B
IDH2 mutation
Glioma
IDH2 mutation
Glioma
vorasidenib
Sensitive: B - Late Trials
vorasidenib
Sensitive
:
B
vorasidenib
Sensitive: B - Late Trials
vorasidenib
Sensitive
:
B
IDH1 mutation
Glioma
IDH1 mutation
Glioma
vorasidenib
Sensitive: B - Late Trials
vorasidenib
Sensitive
:
B
vorasidenib
Sensitive: B - Late Trials
vorasidenib
Sensitive
:
B
IDH2 mutation
Acute Lymphocytic Leukemia
IDH2 mutation
Acute Lymphocytic Leukemia
enasidenib
Sensitive: B - Late Trials
enasidenib
Sensitive
:
B
enasidenib
Sensitive: B - Late Trials
enasidenib
Sensitive
:
B
IDH2 mutation
Myelodysplastic Syndrome
IDH2 mutation
Myelodysplastic Syndrome
enasidenib
Sensitive: C2 – Inclusion Criteria
enasidenib
Sensitive
:
C2
enasidenib
Sensitive: C2 – Inclusion Criteria
enasidenib
Sensitive
:
C2
IDH2 mutation
Acute Myelogenous Leukemia
IDH2 mutation
Acute Myelogenous Leukemia
venetoclax + enasidenib
Sensitive: C3 – Early Trials
venetoclax + enasidenib
Sensitive
:
C3
venetoclax + enasidenib
Sensitive: C3 – Early Trials
venetoclax + enasidenib
Sensitive
:
C3
IDH2 R140
Acute Myelogenous Leukemia
IDH2 R140
Acute Myelogenous Leukemia
enasidenib
Sensitive: C3 – Early Trials
enasidenib
Sensitive
:
C3
enasidenib
Sensitive: C3 – Early Trials
enasidenib
Sensitive
:
C3
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