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DRUG CLASS:
FGFR2 inhibitor
DRUG CLASS:
FGFR2 inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
RLY-4008 (3)
Max-40279 (2)
TT-00434 (1)
HMPL-453 (1)
ABSK061 (0)
ASP5878 (0)
CGT4859 (0)
DS-1123 (0)
LY2874455 (0)
S-49076 (0)
RPT835 (0)
PBI-05204 (0)
3D185 (0)
RLY-4008 (3)
Max-40279 (2)
TT-00434 (1)
HMPL-453 (1)
ABSK061 (0)
ASP5878 (0)
CGT4859 (0)
DS-1123 (0)
LY2874455 (0)
S-49076 (0)
RPT835 (0)
PBI-05204 (0)
3D185 (0)
›
Associations
(10)
News
Trials
VERI cancer hierarchy
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FGFR2 fusion
Cholangiocarcinoma
FGFR2 fusion
Cholangiocarcinoma
RLY-4008
Sensitive: C2 – Inclusion Criteria
RLY-4008
Sensitive
:
C2
RLY-4008
Sensitive: C2 – Inclusion Criteria
RLY-4008
Sensitive
:
C2
FGFR2 fusion
Cholangiocarcinoma
FGFR2 fusion
Cholangiocarcinoma
HMPL-453
Sensitive: C2 – Inclusion Criteria
HMPL-453
Sensitive
:
C2
HMPL-453
Sensitive: C2 – Inclusion Criteria
HMPL-453
Sensitive
:
C2
FGFR3 S249C
Urothelial Cancer
FGFR3 S249C
Urothelial Cancer
FGFR2 inhibitor
Resistant: C3 – Early Trials
FGFR2 inhibitor
Resistant
:
C3
FGFR2 inhibitor
Resistant: C3 – Early Trials
FGFR2 inhibitor
Resistant
:
C3
FGFR3 Y373C
Urothelial Cancer
FGFR3 Y373C
Urothelial Cancer
FGFR2 inhibitor
Resistant: C3 – Early Trials
FGFR2 inhibitor
Resistant
:
C3
FGFR2 inhibitor
Resistant: C3 – Early Trials
FGFR2 inhibitor
Resistant
:
C3
FGFR2 mutation
Cholangiocarcinoma
FGFR2 mutation
Cholangiocarcinoma
FGFR2 inhibitor
Resistant: C3 – Early Trials
FGFR2 inhibitor
Resistant
:
C3
FGFR2 inhibitor
Resistant: C3 – Early Trials
FGFR2 inhibitor
Resistant
:
C3
FGFR2 rearrangement
Cholangiocarcinoma
FGFR2 rearrangement
Cholangiocarcinoma
RLY-4008
Sensitive: C3 – Early Trials
RLY-4008
Sensitive
:
C3
RLY-4008
Sensitive: C3 – Early Trials
RLY-4008
Sensitive
:
C3
FGFR2-ARHGAP24 fusion
Cholangiocarcinoma
FGFR2-ARHGAP24 fusion
Cholangiocarcinoma
TT-00434
Sensitive: C3 – Early Trials
TT-00434
Sensitive
:
C3
TT-00434
Sensitive: C3 – Early Trials
TT-00434
Sensitive
:
C3
FLT3-ITD mutation
Acute Myelogenous Leukemia
FLT3-ITD mutation
Acute Myelogenous Leukemia
Max-40279
Sensitive: D – Preclinical
Max-40279
Sensitive
:
D
Max-40279
Sensitive: D – Preclinical
Max-40279
Sensitive
:
D
FLT3 D835Y
Acute Myelogenous Leukemia
FLT3 D835Y
Acute Myelogenous Leukemia
Max-40279
Sensitive: D – Preclinical
Max-40279
Sensitive
:
D
Max-40279
Sensitive: D – Preclinical
Max-40279
Sensitive
:
D
FGFR2 N549K
Endometrial Cancer
FGFR2 N549K
Endometrial Cancer
RLY-4008
Sensitive: D – Preclinical
RLY-4008
Sensitive
:
D
RLY-4008
Sensitive: D – Preclinical
RLY-4008
Sensitive
:
D
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