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Association details:
Evidence:
Evidence Level:
Sensitive: C4 – Case Studies
Title:

MRTX1719 is an MTA-cooperative PRMT5 inhibitor that exhibits synthetic lethality in preclinical models and patients with MTAP deleted cancer

Published date:
11/01/2023
Excerpt:
A 61-year-old female with NSCLC harboring EGFR mutation and both EGFR and MET gene amplification with progressive disease after treatment with osimertinib was enrolled in the 1719-001 clinical trial. NGS demonstrated homozygous MTAP deletion….The patient was administered MRTX1719 at 400 mg q.d. p.o. on a 21-day cycle and tolerated the treatment well. The first on-study disease assessment at cycle 2 day 20 demonstrated a RECIST-defined partial response with a 41% reduction of the target lesion and was confirmed at cycle 5 day 1 (Fig. 6). The patient remains on study treatment through cycle 6.
DOI:
https://doi.org/10.1158/2159-8290.CD-23-0669