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DRUG CLASS:
CSF-1R inhibitor
DRUG CLASS:
CSF-1R inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
avapritinib (13)
TPX-0022 (8)
surufatinib (7)
pexidartinib (6)
HX301 (2)
chiauranib (1)
vorolanib (1)
OPN-7486 (1)
BMS-986227 (1)
ABSK021 (1)
AMB-05X (0)
C019199 (0)
LY3022855 (0)
NMS-088 (0)
axatilimab-csfr (0)
vimseltinib (0)
SU 14813 (0)
SYHA1813 (0)
Q702 (0)
3D185 (0)
SYHA1817 (0)
BLZ-945 (0)
avapritinib (13)
TPX-0022 (8)
surufatinib (7)
pexidartinib (6)
HX301 (2)
chiauranib (1)
vorolanib (1)
OPN-7486 (1)
BMS-986227 (1)
ABSK021 (1)
AMB-05X (0)
C019199 (0)
LY3022855 (0)
NMS-088 (0)
axatilimab-csfr (0)
vimseltinib (0)
SU 14813 (0)
SYHA1813 (0)
Q702 (0)
3D185 (0)
SYHA1817 (0)
BLZ-945 (0)
›
Associations
(41)
News
Trials
VERI cancer hierarchy
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PDGFRA D842V
Gastrointestinal Stromal Tumor
PDGFRA D842V
Gastrointestinal Stromal Tumor
avapritinib
Sensitive: A1 - Approval
avapritinib
Sensitive
:
A1
avapritinib
Sensitive: A1 - Approval
avapritinib
Sensitive
:
A1
No biomarker
Neuroendocrine Tumor
No biomarker
Neuroendocrine Tumor
surufatinib
Sensitive: A1 - Approval
surufatinib
Sensitive
:
A1
surufatinib
Sensitive: A1 - Approval
surufatinib
Sensitive
:
A1
PDGFRA exon 18 mutation
Gastrointestinal Stromal Tumor
PDGFRA exon 18 mutation
Gastrointestinal Stromal Tumor
avapritinib
Sensitive: A1 - Approval
avapritinib
Sensitive
:
A1
avapritinib
Sensitive: A1 - Approval
avapritinib
Sensitive
:
A1
No biomarker
Tenosynovial Giant Cell Tumor
No biomarker
Tenosynovial Giant Cell Tumor
pexidartinib
Sensitive: A1 - Approval
pexidartinib
Sensitive
:
A1
pexidartinib
Sensitive: A1 - Approval
pexidartinib
Sensitive
:
A1
No biomarker
Mantle Cell Lymphoma
No biomarker
Mantle Cell Lymphoma
avapritinib
Sensitive: A1 - Approval
avapritinib
Sensitive
:
A1
avapritinib
Sensitive: A1 - Approval
avapritinib
Sensitive
:
A1
No biomarker
Small Cell Lung Cancer
No biomarker
Small Cell Lung Cancer
chiauranib
Sensitive: B - Late Trials
chiauranib
Sensitive
:
B
chiauranib
Sensitive: B - Late Trials
chiauranib
Sensitive
:
B
PDGFRA mutation
Gastrointestinal Stromal Tumor
PDGFRA mutation
Gastrointestinal Stromal Tumor
avapritinib
Sensitive: C2 – Inclusion Criteria
avapritinib
Sensitive
:
C2
avapritinib
Sensitive: C2 – Inclusion Criteria
avapritinib
Sensitive
:
C2
KIT mutation
Gastrointestinal Stromal Tumor
KIT mutation
Gastrointestinal Stromal Tumor
avapritinib
Sensitive: C2 – Inclusion Criteria
avapritinib
Sensitive
:
C2
avapritinib
Sensitive: C2 – Inclusion Criteria
avapritinib
Sensitive
:
C2
MET amplification
Gastric Cancer
MET amplification
Gastric Cancer
TPX-0022
Sensitive: C2 – Inclusion Criteria
TPX-0022
Sensitive
:
C2
TPX-0022
Sensitive: C2 – Inclusion Criteria
TPX-0022
Sensitive
:
C2
MET mutation
Gastric Cancer
MET mutation
Gastric Cancer
TPX-0022
Sensitive: C2 – Inclusion Criteria
TPX-0022
Sensitive
:
C2
TPX-0022
Sensitive: C2 – Inclusion Criteria
TPX-0022
Sensitive
:
C2
FLT3-ITD mutation
Acute Myelogenous Leukemia
FLT3-ITD mutation
Acute Myelogenous Leukemia
pexidartinib
Sensitive: C2 – Inclusion Criteria
pexidartinib
Sensitive
:
C2
pexidartinib
Sensitive: C2 – Inclusion Criteria
pexidartinib
Sensitive
:
C2
KIT mutation
Acute Myelogenous Leukemia
KIT mutation
Acute Myelogenous Leukemia
avapritinib
Sensitive: C2 – Inclusion Criteria
avapritinib
Sensitive
:
C2
avapritinib
Sensitive: C2 – Inclusion Criteria
avapritinib
Sensitive
:
C2
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