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DRUG CLASS:
Androgen receptor inhibitor
DRUG CLASS:
Androgen receptor inhibitor
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News alerts, weekly reports and conference planners
Related drugs:
‹
enzalutamide capsule (63)
bicalutamide (13)
darolutamide (6)
flutamide (4)
EPI-7170 (1)
SID 3712502 (1)
enzalutamide capsule (63)
bicalutamide (13)
darolutamide (6)
flutamide (4)
EPI-7170 (1)
SID 3712502 (1)
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Associations
(88)
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No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
enzalutamide capsule
Sensitive: A1 - Approval
enzalutamide capsule
Sensitive
:
A1
enzalutamide capsule
Sensitive: A1 - Approval
enzalutamide capsule
Sensitive
:
A1
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
darolutamide
Sensitive: A1 - Approval
darolutamide
Sensitive
:
A1
darolutamide
Sensitive: A1 - Approval
darolutamide
Sensitive
:
A1
AR splice variant 7
Prostate Cancer
AR splice variant 7
Prostate Cancer
enzalutamide capsule
Resistant: A2 - Guideline
enzalutamide capsule
Resistant
:
A2
enzalutamide capsule
Resistant: A2 - Guideline
enzalutamide capsule
Resistant
:
A2
AR positive
Salivary Gland Cancer
AR positive
Salivary Gland Cancer
bicalutamide
Sensitive: A2 - Guideline
bicalutamide
Sensitive
:
A2
bicalutamide
Sensitive: A2 - Guideline
bicalutamide
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
bicalutamide + goserelin acetate
Sensitive: A2 - Guideline
bicalutamide + goserelin acetate
Sensitive
:
A2
bicalutamide + goserelin acetate
Sensitive: A2 - Guideline
bicalutamide + goserelin acetate
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
goserelin acetate + flutamide
Sensitive: A2 - Guideline
goserelin acetate + flutamide
Sensitive
:
A2
goserelin acetate + flutamide
Sensitive: A2 - Guideline
goserelin acetate + flutamide
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
bicalutamide + triptorelin
Sensitive: A2 - Guideline
bicalutamide + triptorelin
Sensitive
:
A2
bicalutamide + triptorelin
Sensitive: A2 - Guideline
bicalutamide + triptorelin
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
triptorelin + flutamide
Sensitive: A2 - Guideline
triptorelin + flutamide
Sensitive
:
A2
triptorelin + flutamide
Sensitive: A2 - Guideline
triptorelin + flutamide
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
leuprolide acetate + bicalutamide
Sensitive: A2 - Guideline
leuprolide acetate + bicalutamide
Sensitive
:
A2
leuprolide acetate + bicalutamide
Sensitive: A2 - Guideline
leuprolide acetate + bicalutamide
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
leuprolide acetate + flutamide
Sensitive: A2 - Guideline
leuprolide acetate + flutamide
Sensitive
:
A2
leuprolide acetate + flutamide
Sensitive: A2 - Guideline
leuprolide acetate + flutamide
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
bicalutamide + histrelin acetate
Sensitive: A2 - Guideline
bicalutamide + histrelin acetate
Sensitive
:
A2
bicalutamide + histrelin acetate
Sensitive: A2 - Guideline
bicalutamide + histrelin acetate
Sensitive
:
A2
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
histrelin acetate + flutamide
Sensitive: A2 - Guideline
histrelin acetate + flutamide
Sensitive
:
A2
histrelin acetate + flutamide
Sensitive: A2 - Guideline
histrelin acetate + flutamide
Sensitive
:
A2
AR amplification
Prostate Cancer
AR amplification
Prostate Cancer
enzalutamide capsule
Resistant: B - Late Trials
enzalutamide capsule
Resistant
:
B
enzalutamide capsule
Resistant: B - Late Trials
enzalutamide capsule
Resistant
:
B
PTEN mutation
Prostate Cancer
PTEN mutation
Prostate Cancer
bicalutamide
Sensitive: B - Late Trials
bicalutamide
Sensitive
:
B
bicalutamide
Sensitive: B - Late Trials
bicalutamide
Sensitive
:
B
TP53 deletion
Prostate Cancer
TP53 deletion
Prostate Cancer
enzalutamide capsule
Resistant: B - Late Trials
enzalutamide capsule
Resistant
:
B
enzalutamide capsule
Resistant: B - Late Trials
enzalutamide capsule
Resistant
:
B
RB1 deletion
Prostate Cancer
RB1 deletion
Prostate Cancer
enzalutamide capsule
Resistant: B - Late Trials
enzalutamide capsule
Resistant
:
B
enzalutamide capsule
Resistant: B - Late Trials
enzalutamide capsule
Resistant
:
B
BRCA2 deletion
Prostate Cancer
BRCA2 deletion
Prostate Cancer
enzalutamide capsule
Sensitive: B - Late Trials
enzalutamide capsule
Sensitive
:
B
enzalutamide capsule
Sensitive: B - Late Trials
enzalutamide capsule
Sensitive
:
B
CD8 expression
Prostate Cancer
CD8 expression
Prostate Cancer
atezolizumab + enzalutamide capsule
Sensitive: B - Late Trials
atezolizumab + enzalutamide capsule
Sensitive
:
B
atezolizumab + enzalutamide capsule
Sensitive: B - Late Trials
atezolizumab + enzalutamide capsule
Sensitive
:
B
PD-L1 overexpression
Prostate Cancer
PD-L1 overexpression
Prostate Cancer
atezolizumab + enzalutamide capsule
Sensitive: B - Late Trials
atezolizumab + enzalutamide capsule
Sensitive
:
B
atezolizumab + enzalutamide capsule
Sensitive: B - Late Trials
atezolizumab + enzalutamide capsule
Sensitive
:
B
No biomarker
Prostate Cancer
No biomarker
Prostate Cancer
talazoparib + enzalutamide capsule
Sensitive: B - Late Trials
talazoparib + enzalutamide capsule
Sensitive
:
B
talazoparib + enzalutamide capsule
Sensitive: B - Late Trials
talazoparib + enzalutamide capsule
Sensitive
:
B
HR positive
Hormone Receptor Positive Breast Cancer
HR positive
Hormone Receptor Positive Breast Cancer
enzalutamide capsule
Sensitive: C2 – Inclusion Criteria
enzalutamide capsule
Sensitive
:
C2
enzalutamide capsule
Sensitive: C2 – Inclusion Criteria
enzalutamide capsule
Sensitive
:
C2
AR positive
Triple Negative Breast Cancer
AR positive
Triple Negative Breast Cancer
enzalutamide capsule
Sensitive: C2 – Inclusion Criteria
enzalutamide capsule
Sensitive
:
C2
enzalutamide capsule
Sensitive: C2 – Inclusion Criteria
enzalutamide capsule
Sensitive
:
C2
AR positive
Triple Negative Breast Cancer
AR positive
Triple Negative Breast Cancer
darolutamide
Sensitive: C2 – Inclusion Criteria
darolutamide
Sensitive
:
C2
darolutamide
Sensitive: C2 – Inclusion Criteria
darolutamide
Sensitive
:
C2
AR-V7 positive
Prostate Cancer
AR-V7 positive
Prostate Cancer
enzalutamide capsule
Resistant: C2 – Inclusion Criteria
enzalutamide capsule
Resistant
:
C2
enzalutamide capsule
Resistant: C2 – Inclusion Criteria
enzalutamide capsule
Resistant
:
C2
AR F877L
Prostate Cancer
AR F877L
Prostate Cancer
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
AR positive
Salivary Gland Cancer
AR positive
Salivary Gland Cancer
leuprolide acetate + bicalutamide
Sensitive: C3 – Early Trials
leuprolide acetate + bicalutamide
Sensitive
:
C3
leuprolide acetate + bicalutamide
Sensitive: C3 – Early Trials
leuprolide acetate + bicalutamide
Sensitive
:
C3
PLIN2 expression
Salivary Gland Cancer
PLIN2 expression
Salivary Gland Cancer
leuprolide acetate + bicalutamide
Sensitive: C3 – Early Trials
leuprolide acetate + bicalutamide
Sensitive
:
C3
leuprolide acetate + bicalutamide
Sensitive: C3 – Early Trials
leuprolide acetate + bicalutamide
Sensitive
:
C3
AR F876L
Prostate Cancer
AR F876L
Prostate Cancer
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
PTEN expression
Salivary Gland Cancer
PTEN expression
Salivary Gland Cancer
bicalutamide
Sensitive: C3 – Early Trials
bicalutamide
Sensitive
:
C3
bicalutamide
Sensitive: C3 – Early Trials
bicalutamide
Sensitive
:
C3
MSI-H/dMMR
Prostate Cancer
MSI-H/dMMR
Prostate Cancer
pembrolizumab + enzalutamide capsule
Sensitive: C3 – Early Trials
pembrolizumab + enzalutamide capsule
Sensitive
:
C3
pembrolizumab + enzalutamide capsule
Sensitive: C3 – Early Trials
pembrolizumab + enzalutamide capsule
Sensitive
:
C3
AR mutation
Prostate Cancer
AR mutation
Prostate Cancer
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
AR expression
Prostate Cancer
AR expression
Prostate Cancer
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
enzalutamide capsule
Resistant: C3 – Early Trials
enzalutamide capsule
Resistant
:
C3
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