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DRUG CLASS:

CDK2/9 inhibitor

Related drugs:
8d
Anti-Tumor Activity of Cdk2/9 Inhibitor Fadraciclib in an In Vivo Model of Temozolomide Refractory Neuroblastoma. (PubMed, Mol Cancer Ther)
Treatment with the CDK2/9 inhibitor fadraciclib led to significant response and an overall survival benefit in temozolomide-resistant Th-MYCN tumors and allografts generated from these resistant tumours. These findings demonstrate the utility of genetically-engineered mouse models as platforms to dissect the evolution of chemoresistance in neuroblastoma and they provide a mechanistic rationale to support the evaluation of fadraciclib in ongoing paediatric phase I studies of chemotherapy combined with temozolomide in relapsed, treatment refractory neuroblastoma patients.
Preclinical • Journal
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MYCN (MYCN Proto-Oncogene BHLH Transcription Factor)
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temozolomide • fadraciclib (CYC065)