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DRUG:
Gilotrif (afatinib)
i
Other names:
BIBW 2992, BIBW 2992 MA2, BIBW-2992
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Associations
(216)
News
Twitter
Trials
Company:
Boehringer Ingelheim
Drug class:
EGFR inhibitor, HER2 inhibitor, HER4 inhibitor
Related drugs:
‹
cetuximab (316)
osimertinib (234)
erlotinib (228)
gefitinib (183)
panitumumab (113)
lapatinib (105)
neratinib (99)
pyrotinib (63)
brigatinib (45)
icotinib (36)
aumolertinib (18)
amivantamab-vmjw (15)
BGB-283 (12)
lazertinib (9)
mobocertinib (7)
furmonertinib (7)
tarloxotinib bromide (7)
WZ4002 (7)
CH7233163 (6)
H002 (6)
ASLAN001 (6)
CL-387785 (5)
nimotuzumab (5)
rociletinib (5)
BDTX-189 (5)
AEE788 (4)
BI-4020 (4)
BLU-945 (4)
tomuzotuximab (4)
GB263T (4)
JIN-A02 (4)
TAS2940 (4)
EGF816 (4)
BBT-176 (3)
BLU-701 (3)
GC-1118A (3)
ASP8273 (3)
DZD9008 (3)
Bay846 (2)
MCLA-129 (2)
OBX02-011 (2)
olmutinib (2)
necitumumab (2)
QL1203 (2)
S95026 (2)
CLN-081 (2)
14aj (1)
ABP 494 (cetuximab biosimilar) (1)
AFM24 (1)
APL-103 (1)
BDTX-1535 (1)
BLU-451 (1)
BPI-15086 (1)
BPI-361175 (1)
Compound 6a (1)
abivertinib (1)
ORIC-114 (1)
befotertinib (1)
TAS3351 (1)
S-222611 (1)
HMPL-813 (1)
ASK120067 (1)
MET306 (1)
SH-1028 (1)
HLX07 (1)
KD019 (1)
trastuzumab (362)
tucatinib (32)
trastuzumab-pkrb (23)
margetuximab (17)
poziotinib (15)
MCLA-128 (15)
KN026 (12)
trastuzumab-dttb (11)
ZW25 (10)
trastuzumab-anns (9)
trastuzumab-dkst (9)
trastuzumab-qyyp (9)
LZM-005 (8)
PRS-343 (8)
Zercepac (trastuzumab biosimilar) (7)
inetetamab (2)
Her-VAXX (2)
trastuzumab/hyaluronidase-oysk (2)
JBJ-08–178–01 (2)
pertuzumab/trastuzumab/hyaluronidase-zzxf (2)
AB-201 (1)
ABL105 (1)
ACE1702 (1)
AST-301 (1)
Hercease (trastuzumab biosimilar) (1)
CT-0508 (1)
EG12014 (trastuzumab biosimilar) (1)
HERtiCAD (trastuzumab biosimilar) (1)
Hervelous (trastuzumab biosimilar) (1)
MP0274 (1)
SAR443216 (1)
TX05 (trastuzumab biosimilar) (1)
VRN101099 (1)
trastuzumab-IFN-β mutein (1)
cetuximab (316)
osimertinib (234)
erlotinib (228)
gefitinib (183)
panitumumab (113)
lapatinib (105)
neratinib (99)
pyrotinib (63)
brigatinib (45)
icotinib (36)
aumolertinib (18)
amivantamab-vmjw (15)
BGB-283 (12)
lazertinib (9)
mobocertinib (7)
furmonertinib (7)
tarloxotinib bromide (7)
WZ4002 (7)
CH7233163 (6)
H002 (6)
ASLAN001 (6)
CL-387785 (5)
nimotuzumab (5)
rociletinib (5)
BDTX-189 (5)
AEE788 (4)
BI-4020 (4)
BLU-945 (4)
tomuzotuximab (4)
GB263T (4)
JIN-A02 (4)
TAS2940 (4)
EGF816 (4)
BBT-176 (3)
BLU-701 (3)
GC-1118A (3)
ASP8273 (3)
DZD9008 (3)
Bay846 (2)
MCLA-129 (2)
OBX02-011 (2)
olmutinib (2)
necitumumab (2)
QL1203 (2)
S95026 (2)
CLN-081 (2)
14aj (1)
ABP 494 (cetuximab biosimilar) (1)
AFM24 (1)
APL-103 (1)
BDTX-1535 (1)
BLU-451 (1)
BPI-15086 (1)
BPI-361175 (1)
Compound 6a (1)
abivertinib (1)
ORIC-114 (1)
befotertinib (1)
TAS3351 (1)
S-222611 (1)
HMPL-813 (1)
ASK120067 (1)
MET306 (1)
SH-1028 (1)
HLX07 (1)
KD019 (1)
trastuzumab (362)
tucatinib (32)
trastuzumab-pkrb (23)
margetuximab (17)
poziotinib (15)
MCLA-128 (15)
KN026 (12)
trastuzumab-dttb (11)
ZW25 (10)
trastuzumab-anns (9)
trastuzumab-dkst (9)
trastuzumab-qyyp (9)
LZM-005 (8)
PRS-343 (8)
Zercepac (trastuzumab biosimilar) (7)
inetetamab (2)
Her-VAXX (2)
trastuzumab/hyaluronidase-oysk (2)
JBJ-08–178–01 (2)
pertuzumab/trastuzumab/hyaluronidase-zzxf (2)
AB-201 (1)
ABL105 (1)
ACE1702 (1)
AST-301 (1)
Hercease (trastuzumab biosimilar) (1)
CT-0508 (1)
EG12014 (trastuzumab biosimilar) (1)
HERtiCAD (trastuzumab biosimilar) (1)
Hervelous (trastuzumab biosimilar) (1)
MP0274 (1)
SAR443216 (1)
TX05 (trastuzumab biosimilar) (1)
VRN101099 (1)
trastuzumab-IFN-β mutein (1)
›
Associations
(216)
News
Twitter
Trials
Reset Filters
VERI cancer hierarchy
x
x
x
x
EGFR exon 19 deletion
Non Small Cell Lung Cancer
EGFR exon 19 deletion
Non Small Cell Lung Cancer
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
EGFR L858R
Non Small Cell Lung Cancer
EGFR L858R
Non Small Cell Lung Cancer
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
EGFR mutation
Non Small Cell Lung Cancer
EGFR mutation
Non Small Cell Lung Cancer
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
No biomarker
Non Small Cell Lung Cancer
No biomarker
Non Small Cell Lung Cancer
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
No biomarker
Lung Non-Small Cell Squamous Cancer
No biomarker
Lung Non-Small Cell Squamous Cancer
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
afatinib
Sensitive: A1 - Approval
afatinib
Sensitive
:
A1
No biomarker
Oral Cancer
No biomarker
Oral Cancer
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
No biomarker
Oropharyngeal Cancer
No biomarker
Oropharyngeal Cancer
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
EGFR S768I
Non Small Cell Lung Cancer
EGFR S768I
Non Small Cell Lung Cancer
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
EGFR G719X
Non Small Cell Lung Cancer
EGFR G719X
Non Small Cell Lung Cancer
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
EGFR L861Q
Non Small Cell Lung Cancer
EGFR L861Q
Non Small Cell Lung Cancer
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
HER-2 mutation
Non Small Cell Lung Cancer
HER-2 mutation
Non Small Cell Lung Cancer
afatinib
Resistant: A2 - Guideline
afatinib
Resistant
:
A2
afatinib
Resistant: A2 - Guideline
afatinib
Resistant
:
A2
EGFR mutation
Lung Non-Squamous Non-Small Cell Cancer
EGFR mutation
Lung Non-Squamous Non-Small Cell Cancer
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
afatinib
Sensitive: A2 - Guideline
afatinib
Sensitive
:
A2
EGFR exon 20 insertion
Non Small Cell Lung Cancer
EGFR exon 20 insertion
Non Small Cell Lung Cancer
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
EGFR T790M
Non Small Cell Lung Cancer
EGFR T790M
Non Small Cell Lung Cancer
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
EGFR mutation
Lung Adenocarcinoma
EGFR mutation
Lung Adenocarcinoma
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
EGFR L858R + EGFR T790M
Non Small Cell Lung Cancer
EGFR L858R + EGFR T790M
Non Small Cell Lung Cancer
osimertinib + afatinib
Sensitive: B - Late Trials
osimertinib + afatinib
Sensitive
:
B
osimertinib + afatinib
Sensitive: B - Late Trials
osimertinib + afatinib
Sensitive
:
B
EGFR exon 19 deletion
Lung Adenocarcinoma
EGFR exon 19 deletion
Lung Adenocarcinoma
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
EGFR amplification
Squamous Cell Carcinoma of Head and Neck
EGFR amplification
Squamous Cell Carcinoma of Head and Neck
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
ERBB3-L
Squamous Cell Carcinoma of Head and Neck
ERBB3-L
Squamous Cell Carcinoma of Head and Neck
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
CDKN2A negative
Squamous Cell Carcinoma of Head and Neck
CDKN2A negative
Squamous Cell Carcinoma of Head and Neck
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
PTEN-H
Squamous Cell Carcinoma of Head and Neck
PTEN-H
Squamous Cell Carcinoma of Head and Neck
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
ERBB4 G668V
Lung Non-Small Cell Squamous Cancer
ERBB4 G668V
Lung Non-Small Cell Squamous Cancer
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
EGFR R1052K
Lung Non-Small Cell Squamous Cancer
EGFR R1052K
Lung Non-Small Cell Squamous Cancer
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
HER-2 E395K
Lung Non-Small Cell Squamous Cancer
HER-2 E395K
Lung Non-Small Cell Squamous Cancer
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
HER-2 Q57R
Lung Non-Small Cell Squamous Cancer
HER-2 Q57R
Lung Non-Small Cell Squamous Cancer
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
EGFR L858R
Lung Adenocarcinoma
EGFR L858R
Lung Adenocarcinoma
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
afatinib
Sensitive: B - Late Trials
afatinib
Sensitive
:
B
EGFR mutation
Esophageal Squamous Cell Carcinoma
EGFR mutation
Esophageal Squamous Cell Carcinoma
afatinib
Sensitive: C1 - Off-label
afatinib
Sensitive
:
C1
afatinib
Sensitive: C1 - Off-label
afatinib
Sensitive
:
C1
EGFR mutation
Gastric Cancer
EGFR mutation
Gastric Cancer
afatinib
Sensitive: C1 - Off-label
afatinib
Sensitive
:
C1
afatinib
Sensitive: C1 - Off-label
afatinib
Sensitive
:
C1
EGFR exon 20 insertion
Non Small Cell Lung Cancer
EGFR exon 20 insertion
Non Small Cell Lung Cancer
cetuximab + afatinib
Sensitive: C2 – Inclusion Criteria
cetuximab + afatinib
Sensitive
:
C2
cetuximab + afatinib
Sensitive: C2 – Inclusion Criteria
cetuximab + afatinib
Sensitive
:
C2
KRAS mutation
Non Small Cell Lung Cancer
KRAS mutation
Non Small Cell Lung Cancer
afatinib + selumetinib
Sensitive: C2 – Inclusion Criteria
afatinib + selumetinib
Sensitive
:
C2
afatinib + selumetinib
Sensitive: C2 – Inclusion Criteria
afatinib + selumetinib
Sensitive
:
C2
HER-2 amplification
Non Small Cell Lung Cancer
HER-2 amplification
Non Small Cell Lung Cancer
afatinib
Sensitive: C2 – Inclusion Criteria
afatinib
Sensitive
:
C2
afatinib
Sensitive: C2 – Inclusion Criteria
afatinib
Sensitive
:
C2
HER-2 amplification
Urothelial Cancer
HER-2 amplification
Urothelial Cancer
afatinib
Sensitive: C2 – Inclusion Criteria
afatinib
Sensitive
:
C2
afatinib
Sensitive: C2 – Inclusion Criteria
afatinib
Sensitive
:
C2
^
^
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