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BIOMARKER:
FLT3-TKD mutation
i
Other names:
FLT3, Fms Related Tyrosine Kinase 3, Receptor-Type Tyrosine-Protein Kinase FLT3, Stem Cell Tyrosine Kinase 1, Fms-Like Tyrosine Kinase 3, CD135, FLK-2, STK1, Growth Factor Receptor Tyrosine Kinase Type III, Fetal Liver Kinase 2
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Entrez ID:
2322
Related biomarkers:
Expression
Mutation
CNA
Fusion
Others
‹
FLT3-ITD mutation (90)
FLT3 mutation (67)
FLT3 D835Y (12)
FLT3 F691L (11)
FLT3 D835 (8)
FLT3 D835V (6)
FLT3-ITD mutation + FLT3-TKD mutation (5)
DNMT3A mutation + FLT3-ITD mutation (4)
FLT3 D698N (4)
FLT3 D835H (4)
FLT3 G697R (4)
FLT3 N676K (4)
FLT3 Y842C (4)
FLT3 mutation + NPM1 mutation (4)
FLT3 N676D (3)
FLT3 N676D + FLT3 Y842C (3)
FLT3 N676T (3)
FLT3 mutation + DNMT3A mutation (3)
FLT3 mutation + NRAS mutation (3)
FLT3 wild-type (3)
FLT3-ITD mutation + FLT3 D835 (3)
FLT3-ITD mutation + MLL rearrangement (3)
FLT3-ITD mutation + NPM1 mutation (3)
FLT3‐ITD + NPM1 mutation (3)
FLT3‐ITD mutation + DNMT3A mutation + NPM1 mutation (3)
FLT3 D835A (2)
FLT3 D835F (2)
FLT3 D835N (2)
FLT3 I836 (2)
FLT3 Y842H (2)
FLT3 mutation + MLL mutation (2)
FLT3-ITD mutation + FLT3 D835Y (2)
FLT3-ITD mutation + FLT3 F691L (2)
FLT3-ITD mutation + IDH1 mutation (2)
FLT3-ITD mutation + IDH2 mutation (2)
FLT3-ITD mutation + WT1 mutation (2)
FLT3‐ITD (2)
CEBPZ rearrangement + FLT3-TKD mutation (1)
FLT3 840GS (1)
FLT3 A627T (1)
FLT3 D651G (1)
FLT3 D835E (1)
FLT3 D835G (1)
FLT3 D839G (1)
FLT3 E588_Y589INSKYFYVDFRE (1)
FLT3 F691L + FLT3 D835F (1)
FLT3 F691L + FLT3 D835H (1)
FLT3 F691L + FLT3 D835V (1)
FLT3 F691L + FLT3 D835Y (1)
FLT3 F691L + FLT3 D839G (1)
FLT3 F691L + FLT3 Y842C (1)
FLT3 G619C (1)
FLT3 G846S (1)
FLT3 I687F (1)
FLT3 NPOS + FLT3 D835N (1)
FLT3 V592A + FLT3 D835N (1)
FLT3 V592_D593INSDFREY (1)
FLT3 Y591_V592INSVDFREYE (1)
FLT3 mutation + IDH1 mutation (1)
FLT3 mutation + NRAS mutation + PTPN11 mutation (1)
FLT3 mutation + PTPN11 mutation (1)
FLT3 positive (1)
FLT3-ITD F692L + NPM1 mutation (1)
FLT3-ITD mutation + ASXL1 mutation (1)
FLT3-ITD mutation + ASXL1 mutation + NRAS mutation (1)
FLT3-ITD mutation + DNMT3A mutation + ASXL1 mutation (1)
FLT3-ITD mutation + DNMT3A mutation + NRAS mutation (1)
FLT3-ITD mutation + FLT3 D835Y + FLT3 F691L (1)
FLT3-ITD mutation + NRAS mutation + GATA2 mutation (1)
FLT3-ITD mutation+ DNMT3A mutation + ASXL1 mutation + NRAS mutation (1)
FLT3‐ITD + DNMT3A mutation (1)
FLT3‐ITD + WT1 mutation (1)
MLL rearrangement + FLT3 mutation (1)
NPM1 mutation + FLT3-ITD mutation + TET2 mutation + CUX1 mutation (1)
NPM1 mutation + FLT3-TKD mutation (1)
NPM1 mutation + SRSF2 mutation + FLT3-ITD mutation+ DNMT3A mutation + ASXL1 mutation + NRAS mutation (1)
FLT3 A848P (0)
FLT3 F691I (0)
FLT3 F691L + FLT3 Y842H (0)
FLT3 V592A (0)
FLT3-ITD F692L (0)
FLT3-ITD mutation (90)
FLT3 mutation (67)
FLT3 D835Y (12)
FLT3 F691L (11)
FLT3 D835 (8)
FLT3 D835V (6)
FLT3-ITD mutation + FLT3-TKD mutation (5)
DNMT3A mutation + FLT3-ITD mutation (4)
FLT3 D698N (4)
FLT3 D835H (4)
FLT3 G697R (4)
FLT3 N676K (4)
FLT3 Y842C (4)
FLT3 mutation + NPM1 mutation (4)
FLT3 N676D (3)
FLT3 N676D + FLT3 Y842C (3)
FLT3 N676T (3)
FLT3 mutation + DNMT3A mutation (3)
FLT3 mutation + NRAS mutation (3)
FLT3 wild-type (3)
FLT3-ITD mutation + FLT3 D835 (3)
FLT3-ITD mutation + MLL rearrangement (3)
FLT3-ITD mutation + NPM1 mutation (3)
FLT3‐ITD + NPM1 mutation (3)
FLT3‐ITD mutation + DNMT3A mutation + NPM1 mutation (3)
FLT3 D835A (2)
FLT3 D835F (2)
FLT3 D835N (2)
FLT3 I836 (2)
FLT3 Y842H (2)
FLT3 mutation + MLL mutation (2)
FLT3-ITD mutation + FLT3 D835Y (2)
FLT3-ITD mutation + FLT3 F691L (2)
FLT3-ITD mutation + IDH1 mutation (2)
FLT3-ITD mutation + IDH2 mutation (2)
FLT3-ITD mutation + WT1 mutation (2)
FLT3‐ITD (2)
CEBPZ rearrangement + FLT3-TKD mutation (1)
FLT3 840GS (1)
FLT3 A627T (1)
FLT3 D651G (1)
FLT3 D835E (1)
FLT3 D835G (1)
FLT3 D839G (1)
FLT3 E588_Y589INSKYFYVDFRE (1)
FLT3 F691L + FLT3 D835F (1)
FLT3 F691L + FLT3 D835H (1)
FLT3 F691L + FLT3 D835V (1)
FLT3 F691L + FLT3 D835Y (1)
FLT3 F691L + FLT3 D839G (1)
FLT3 F691L + FLT3 Y842C (1)
FLT3 G619C (1)
FLT3 G846S (1)
FLT3 I687F (1)
FLT3 NPOS + FLT3 D835N (1)
FLT3 V592A + FLT3 D835N (1)
FLT3 V592_D593INSDFREY (1)
FLT3 Y591_V592INSVDFREYE (1)
FLT3 mutation + IDH1 mutation (1)
FLT3 mutation + NRAS mutation + PTPN11 mutation (1)
FLT3 mutation + PTPN11 mutation (1)
FLT3 positive (1)
FLT3-ITD F692L + NPM1 mutation (1)
FLT3-ITD mutation + ASXL1 mutation (1)
FLT3-ITD mutation + ASXL1 mutation + NRAS mutation (1)
FLT3-ITD mutation + DNMT3A mutation + ASXL1 mutation (1)
FLT3-ITD mutation + DNMT3A mutation + NRAS mutation (1)
FLT3-ITD mutation + FLT3 D835Y + FLT3 F691L (1)
FLT3-ITD mutation + NRAS mutation + GATA2 mutation (1)
FLT3-ITD mutation+ DNMT3A mutation + ASXL1 mutation + NRAS mutation (1)
FLT3‐ITD + DNMT3A mutation (1)
FLT3‐ITD + WT1 mutation (1)
MLL rearrangement + FLT3 mutation (1)
NPM1 mutation + FLT3-ITD mutation + TET2 mutation + CUX1 mutation (1)
NPM1 mutation + FLT3-TKD mutation (1)
NPM1 mutation + SRSF2 mutation + FLT3-ITD mutation+ DNMT3A mutation + ASXL1 mutation + NRAS mutation (1)
FLT3 A848P (0)
FLT3 F691I (0)
FLT3 F691L + FLT3 Y842H (0)
FLT3 V592A (0)
FLT3-ITD F692L (0)
›
Related tests:
LeukoStrat® CDx FLT3 Mutation Assay (6)
LeukoStrat® CDx FLT3 Mutation Assay (6)
Associations
(13)
News
Trials
Search handles
@AaronGoodman33
@hemedoc
Search handles
@AaronGoodman33
@hemedoc
Filter by
Latest
1year
NPM1 or CBF in FLT3-TKD-mutated AML identifies a favourable subtype where midostaurin improves only EFS and not OS. Here is an interesting analysis from RATIFY. https://t.co/RKRqB0ucfs (@RanjitKSMD)
1 year ago
FLT3 (Fms-related tyrosine kinase 3) • NPM1 (Nucleophosmin 1)
|
FLT3-TKD mutation
|
Rydapt (midostaurin)
over2years
Great question. Issue of prognostic significance of FLT3-TKD mutations in AML often comes up. Cant resist posting the (old) paper from my PhD studing UK AML trial data. If anything TKD associated with a more favourable prognosis (quite distinct to ITD): https://t.co/UvMLWA91qn (@AdamMead_Oxford)
over 2 years ago
FLT3 (Fms-related tyrosine kinase 3)
|
FLT3-TKD mutation
over2years
AML Question!!! 40 year old with inv(16) AML treated with 7+3->CR. HiDAC x 3. Unfortunately 2 years later presents with relapsed disease. NGS with FLT3 TKD mutation (VAF 30%). Cytogenetics inv(16). Patient is fit. WBC 50,000, ANC 100, Plt 15. You recommend (off trial) (@AaronGoodman33)
over 2 years ago
Clinical • Next-generation sequencing
|
FLT3 (Fms-related tyrosine kinase 3)
|
FLT3-TKD mutation
over3years
#ASH20 #leusm Perl: Important to remember Sorafenib and Quizartinib are not effective for FLT3-TKD mutations. (@hemedoc)
over 3 years ago
FLT3 (Fms-related tyrosine kinase 3)
|
FLT3-TKD mutation
|
sorafenib • Vanflyta (quizartinib)
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