Group by Gene: Include preclinical: Tyrosine Kinase Inhibitors Serine-Threonine Kinase Inhibitors FGF Immunotherapy CD Protein Inhibitors Immune Checkpoint Inhibitors Threonine-Tyrosine Kinase Inhibitors Other EGFR Interleukins Epigenetics | Multi-tyrosine kinase inhibitor cabozantinib tablet | cabozantinib capsule | TrkB receptor inhibitor, TrkC kinase inhibitor, TrkA receptor inhibitor larotrectinib | RANK ligand inhibitor denosumab | BRAF inhibitor, BRAF V600E inhibitor vemurafenib | FORE-8394 | MEK inhibitor, BRAF inhibitor trametinib + dabrafenib | BRAF inhibitor + MEK inhibitor | RET inhibitor selpercatinib | pralsetinib | PD1 inhibitor pembrolizumab | BRAF inhibitor dabrafenib | IL-6 inhibitor siltuximab | TrkB receptor inhibitor, TrkC kinase inhibitor, ROS1 inhibitor, TrkA receptor antagonist AB-106 | FGFR inhibitor, VEGFR inhibitor, RET inhibitor, c-KIT inhibitor, PDGFR α antagonist lenvatinib | pan-RAF inhibitor, Multi-tyrosine kinase inhibitor sorafenib | TrkB receptor inhibitor, TrkC kinase inhibitor, ROS1 inhibitor, TrkA receptor inhibitor, ALK inhibitor, JAK2 inhibitor, TNK2 inhibitor entrectinib | BRAF inhibitor, MEK1 inhibitor, BRAF V600E inhibitor vemurafenib + cobimetinib | pan-RAF inhibitor, EGFR inhibitor BGB-283 | BRAF inhibitor, BRAF V600E inhibitor, Cytochrome P450 inhibitor FORE-8394 + cobicistat | MEK inhibitor, BRAF inhibitor, MEK2 inhibitor, MEK1 inhibitor, BRAF V600E inhibitor vemurafenib + HL-085 | AKT inhibitor MK-2206 | Bcr-abl tyrosine kinase inhibitor, MEK inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist dasatinib + CI-1040 | Bcr-abl tyrosine kinase inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist dasatinib | Aurora kinase inhibitor, MEK inhibitor, SRC-family kinase (SFK) inhibitor CI-1040 + SU6656 | MEK inhibitor, Src kinase inhibitor CI-1040 + PP2 | MEK inhibitor CI-1040 | JAK1 inhibitor, JAK2 inhibitor AZD1480 | MEK inhibitor, BRAF inhibitor, WEE1 inhibitor trametinib + dabrafenib + AZD1775 | Src kinase inhibitor PP2 |
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No biomarker | ||||||||||||||||||||||||||||||
BRAF V600 | ||||||||||||||||||||||||||||||
BRAF V600E | ||||||||||||||||||||||||||||||
BRAF mutation | ||||||||||||||||||||||||||||||
RET fusion | ||||||||||||||||||||||||||||||
NTRK1 fusion | ||||||||||||||||||||||||||||||
NTRK1 overexpression | ||||||||||||||||||||||||||||||
RET rearrangement | ||||||||||||||||||||||||||||||
RET C634W | ||||||||||||||||||||||||||||||
RET M918T | ||||||||||||||||||||||||||||||
TMB-H | ||||||||||||||||||||||||||||||
NCOA4-RET fusion | ||||||||||||||||||||||||||||||
NTRK3 fusion | ||||||||||||||||||||||||||||||
GLI3 overexpression | ||||||||||||||||||||||||||||||
GLI2 overexpression | ||||||||||||||||||||||||||||||
GLI1 overexpression | ||||||||||||||||||||||||||||||
TPM3-NTRK1 fusion | ||||||||||||||||||||||||||||||
EGFR overexpression | ||||||||||||||||||||||||||||||
NTRK2 fusion | ||||||||||||||||||||||||||||||
NRAS Q61K + BRAF V600E | ||||||||||||||||||||||||||||||
PDGFRB overexpression | ||||||||||||||||||||||||||||||
MSI-H/dMMR | ||||||||||||||||||||||||||||||
RET-PTC1 rearrangement | ||||||||||||||||||||||||||||||
BRAF V600E + TERT mutation | ||||||||||||||||||||||||||||||
PTEN R130del | ||||||||||||||||||||||||||||||
PIK3CA E545K |