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CANCER:

Thyroid Gland Papillary Carcinoma





Show legend
Group by Gene:
Include preclinical:

0
Multi-tyrosine kinase inhibitor
cabozantinib tablet
cabozantinib capsule
1
TrkB receptor inhibitor, TrkC kinase inhibitor, TrkA receptor inhibitor
larotrectinib
2
RANK ligand inhibitor
denosumab
3
BRAF inhibitor, BRAF V600E inhibitor
vemurafenib
FORE-8394
4
MEK inhibitor, BRAF inhibitor
trametinib + dabrafenib
BRAF inhibitor + MEK inhibitor
5
RET inhibitor
selpercatinib
pralsetinib
6
PD1 inhibitor
pembrolizumab
7
BRAF inhibitor
dabrafenib
8
IL-6 inhibitor
siltuximab
9
TrkB receptor inhibitor, TrkC kinase inhibitor, ROS1 inhibitor, TrkA receptor antagonist
AB-106
10
FGFR inhibitor, VEGFR inhibitor, RET inhibitor, c-KIT inhibitor, PDGFR α antagonist
lenvatinib
11
pan-RAF inhibitor, Multi-tyrosine kinase inhibitor
sorafenib
12
TrkB receptor inhibitor, TrkC kinase inhibitor, ROS1 inhibitor, TrkA receptor inhibitor, ALK inhibitor, JAK2 inhibitor, TNK2 inhibitor
entrectinib
13
BRAF inhibitor, MEK1 inhibitor, BRAF V600E inhibitor
vemurafenib + cobimetinib
14
pan-RAF inhibitor, EGFR inhibitor
BGB-283
15
BRAF inhibitor, BRAF V600E inhibitor, Cytochrome P450 inhibitor
FORE-8394 + cobicistat
16
MEK inhibitor, BRAF inhibitor, MEK2 inhibitor, MEK1 inhibitor, BRAF V600E inhibitor
vemurafenib + HL-085
17
AKT inhibitor
MK-2206
18
Bcr-abl tyrosine kinase inhibitor, MEK inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib + CI-1040
19
Bcr-abl tyrosine kinase inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib
20
Aurora kinase inhibitor, MEK inhibitor, SRC-family kinase (SFK) inhibitor
CI-1040 + SU6656
21
MEK inhibitor, Src kinase inhibitor
CI-1040 + PP2
22
MEK inhibitor
CI-1040
23
JAK1 inhibitor, JAK2 inhibitor
AZD1480
24
MEK inhibitor, BRAF inhibitor, WEE1 inhibitor
trametinib + dabrafenib + AZD1775
25
Src kinase inhibitor
PP2
No biomarker
BRAF V600
BRAF V600E
BRAF mutation
RET fusion
NTRK1 fusion
NTRK1 overexpression
RET rearrangement
RET C634W
RET M918T
TMB-H
NCOA4-RET fusion
NTRK3 fusion
GLI3 overexpression
GLI2 overexpression
GLI1 overexpression
TPM3-NTRK1 fusion
EGFR overexpression
NTRK2 fusion
NRAS Q61K + BRAF V600E
PDGFRB overexpression
MSI-H/dMMR
RET-PTC1 rearrangement
BRAF V600E + TERT mutation
PTEN R130del
PIK3CA E545K