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CANCER:

Genito-urinary Cancer





Show legend
Group by Gene:
Include preclinical:

PD1 inhibitor
nivolumab
pembrolizumab
toripalimab-tpzi
cemiplimab-rwlc
0
PD1 inhibitor
camrelizumab
tislelizumab
PF-06801591
sintilimab
retifanlimab-dlwr
zimberelimab
dostarlimab-gxly
PARP inhibitor
olaparib
1
PARP inhibitor
rucaparib
niraparib
talazoparib
IMP4297
Krabeva (bevacizumab biosimilar)
bevacizumab-tnjn
bevacizumab-adcd
2
VEGF-A inhibitor
bevacizumab
bevacizumab-awwb
bevacizumab-bvzr
bevacizumab-maly
Aybintio (bevacizumab biosimilar)
PD-L1 inhibitor
3
PD-L1 inhibitor
atezolizumab
durvalumab
avelumab
cisplatin
cisplatin + gemcitabine
4
DNA synthesis inhibitor
gemcitabine
mitomycin urothelial gel
gemcitabine-releasing intravesical system
leuprolide 6-month depot
leuprolide acetate
5
GnRH agonist
triptorelin
histrelin acetate
goserelin acetate
leuprorelin depot
mTOR inhibitor
6
mTOR inhibitor
everolimus
temsirolimus
Androgen receptor inhibitor
enzalutamide capsule
7
Androgen receptor inhibitor
darolutamide
bicalutamide
enzalutamide capsule + EPI-7170
SID 3712502
pazopanib
cabozantinib tablet
8
Multi-tyrosine kinase inhibitor
cabozantinib capsule
midostaurin
anlotinib
ponatinib
FGFR inhibitor
BAY 1163877
infigratinib
ABSK091
9
FGFR inhibitor
pemigatinib
futibatinib
ARQ 087
Debio 1347
AZ8010
abiraterone acetate + histrelin acetate
10
CYP17A1 inhibitor, GnRH agonist
abiraterone acetate + goserelin acetate
abiraterone acetate + triptorelin
abiraterone acetate + leuprolide acetate
triptorelin + nilutamide
leuprolide acetate + nilutamide
11
Androgen receptor antagonist, GnRH agonist
histrelin acetate + nilutamide
goserelin acetate + nilutamide
leuprolide acetate + apalutamide
12
PD1 inhibitor, CTLA4 inhibitor
nivolumab + ipilimumab
CYP17A1 inhibitor
13
CYP17A1 inhibitor
abiraterone acetate
abiraterone acetate
abiraterone acetate
cetuximab
14
EGFR inhibitor
erlotinib
icotinib
15
IFNα stimulant, VEGF-A inhibitor
bevacizumab + pegylated interferon α -2a
Aybintio (bevacizumab biosimilar) + pegylated interferon α -2a
5-fluorouracil
16
Thymidylate synthase inhibitor
capecitabine
5-fluorouracil
17
GnRH antagonist
degarelix
relugolix
etoposide IV
18
Topoisomerase II inhibitor
mitoxantrone
doxorubicin hydrochloride
pembrolizumab + axitinib
19
VEGFR inhibitor, PD1 inhibitor
toripalimab-tpzi + axitinib
sintilimab + axitinib
20
PD1 inhibitor, Multi-tyrosine kinase inhibitor
nivolumab + cabozantinib tablet
21
VEGFR inhibitor, PD-L1 inhibitor
avelumab + axitinib
apalutamide
22
Androgen receptor antagonist
EPI-7386
BMS-641988
23
c-MET inhibitor
c-MET inhibitor
savolitinib
24
Microtubule inhibitor
cabazitaxel
25
Tubulin polymerization promoter
carboplatin
26
VEGF-A inhibitor, EGFR inhibitor
bevacizumab + erlotinib
27
HIF-2α inhibitor
belzutifan
28
Tubulin polymerization promoter, DNA synthesis inhibitor
carboplatin + gemcitabine
29
VEGFR inhibitor
VEGFR inhibitor
axitinib
30
IFNα stimulant
nadofaragene firadenovec-vncg
31
Bifunctional alkylating agent
ifosfamide
32
Topoisomerase II inhibitor, RNA synthesis inhibitor
dactinomycin
33
VEGF-A inhibitor, mTOR inhibitor
bevacizumab + everolimus
34
Tubulin polymerization promoter, Microtubule inhibitor
carboplatin + cabazitaxel
35
Topoisomerase II inhibitor, DNA inhibitor, DNA synthesis inhibitor
cisplatin + etoposide oral
36
Topoisomerase II inhibitor, DNA inhibitor
etoposide oral
37
Immunostimulant, Prostatic acid phosphatase inhibitor
sipuleucel-T
38
Bone resorption factor inhibitor, Osteoclast inhibitor
zoledronic acid
39
Tubulin polymerization promoter, Bcl2 inhibitor
carboplatin + paclitaxel
paclitaxel
40
DNA synthesis inhibitor, Topoisomerase I inhibitor
cisplatin + irinotecan
41
Ionizing radiation emitter, PSMA inhibitor
PNT2002
lutetium Lu 177 vipivotide tetraxetan
42
Androgen receptor degrader
ARV-110
AC0176
43
CXCL12 inhibitor, Farnesyl transferase inhibitor
tipifarnib
44
PI3K inhibitor, AKT inhibitor
RG7440
45
FGFR inhibitor, PD-L1 inhibitor
atezolizumab + BAY 1163877
durvalumab + ABSK091
46
PD1 inhibitor, PI3Kγ inhibitor
nivolumab + IPI-549
47
CTLA4 inhibitor
CTLA4 inhibitor
ipilimumab
48
Androgen receptor inhibitor, PARP inhibitor
talazoparib + enzalutamide capsule
49
ALK inhibitor
crizotinib
alectinib
50
AXL inhibitor, GAS6 inhibitor
AVB-500
51
PLK1 inhibitor
PCM-075
52
HLA G-targeted CAR-T immunotherapy
IVS-3001
53
Apoptosis stimulant
Alpha1H
54
IL-15 superagonist
nogapendekin alfa inbakicept-pmln
55
Immunostimulant
RV001
56
CD70-targeted CAR-T immunotherapy
ALLO-316
57
CLDN6-targeted CAR-T immunotherapy
BNT211
58
Reactive oxygen species stimulant
AU-011
59
PD1 inhibitor, Multi-tyrosine kinase inhibitor, CTLA4 inhibitor
nivolumab + ipilimumab + cabozantinib tablet
60
PD1 inhibitor, PARP inhibitor
nivolumab + rucaparib
pembrolizumab + olaparib
FGFR3 inhibitor
61
FGFR3 inhibitor
B-701
TYRA-300
MEK inhibitor
62
MEK inhibitor
trametinib
PD-0325901
63
HER2 inhibitor, HER2 dimerization inhibitor
trastuzumab + pertuzumab
64
PARP inhibitor, AKT inhibitor
olaparib + capivasertib
65
Androgen receptor inhibitor, mTOR inhibitor, DNA PK inhibitor
enzalutamide capsule + CC-115
66
PD-L1 inhibitor, PARP inhibitor
avelumab + talazoparib
67
HER2 inhibitor
trastuzumab-pkrb
trastuzumab
68
PD1 inhibitor, IDO1 inhibitor
nivolumab + BMS-986205
pembrolizumab + INCB024360
69
HDAC inhibitor
vorinostat
70
DNA PK inhibitor
NU7441
M3814
71
CYP11A1 inhibitor
ODM-208
72
CDC7 kinase inhibitor
LY3143921
73
VEGFR inhibitor, PARP inhibitor
olaparib + cediranib
74
VEGF-A inhibitor, PI3Kγ inhibitor, Bcl2 inhibitor, Tubulin inhibitor
bevacizumab + albumin-bound paclitaxel + IPI-549
75
CDK4 inhibitor, CDK6 inhibitor
palbociclib
abemaciclib
76
VEGFR-2 inhibitor
ramucirumab
77
VEGFR inhibitor, mTOR inhibitor
temsirolimus + axitinib
78
HIF-2α antagonist
MK-3795
79
Microtubule inhibitor, CLDN6-targeted antibody-drug conjugate
TORL-1-23
IMAB027-vcMMAE
80
HDAC inhibitor, Multi-tyrosine kinase inhibitor
pazopanib + CG-781
81
PD1 inhibitor, EphB4 inhibitor
pembrolizumab + sEphB4-HSA
82
PD-L1 inhibitor, c-MET inhibitor
durvalumab + savolitinib
83
PD1 inhibitor, ICOS agonist
pembrolizumab + GSK3359609
84
PI3K inhibitor
AN2025
MEN1611
85
PI3Kβ inhibitor, PD1 inhibitor
pembrolizumab + GSK2636771
86
PI3Kβ inhibitor
GSK2636771
87
IL-6R antagonist, PD-L1 inhibitor
atezolizumab + tocilizumab
88
mTORC1 inhibitor, mTORC2 inhibitor
CB-228
89
Tubulin inhibitor
vinblastine
90
BRAF inhibitor, BRAF V600E inhibitor
vemurafenib
91
ALK inhibitor, Multi-tyrosine kinase inhibitor
crizotinib + pazopanib
92
PRMT5 inhibitor
AMG 193
EP
FOLFOX
GC
ddMVAC
GemPOx
VAC
93
Chemotherapy
TIP
VeIP
VIP
BEP
GemOx
VC
CaT
TI-CE
94
GnRH stimulant
GnRH stimulant
95
Immunotherapy
Immunotherapy
96
FGFR2 inhibitor
FGFR2 inhibitor
97
Tyrosine kinase inhibitor
Tyrosine kinase inhibitor
PD173074
98
Immunotherapy, Tyrosine kinase inhibitor
Immunotherapy + Tyrosine kinase inhibitor
99
VEGF inhibitor
VEGF inhibitor
100
VEGFR inhibitor, Immunotherapy
Immunotherapy + VEGFR inhibitor
101
ATM kinase inhibitor
ATM kinase inhibitor
102
Glutamate inhibitor
Glutamate inhibitor
103
Src kinase inhibitor, PARP inhibitor
PARP inhibitor + Src kinase inhibitor
104
mTORC1 inhibitor
mTORC1 inhibitor
105
VEGFR inhibitor, PDGFR inhibitor, c-KIT inhibitor
sunitinib
106
FGFR2 inhibitor, FGFR inhibitor, FGFR1 inhibitor, FGFR3 inhibitor, FGFR4 inhibitor
erdafitinib
erdafitinib + Debio 1347
docetaxel
107
Microtubule stabilizer, Tubulin polymerization promoter
carboplatin + docetaxel
docetaxel
108
FGFR inhibitor, VEGFR inhibitor, RET inhibitor, c-KIT inhibitor, PDGFR α antagonist
lenvatinib
109
Nectin-4-targeted antibody-drug conjugate, Microtubule inhibitor
enfortumab vedotin-ejfv
110
pan-RAF inhibitor, Multi-tyrosine kinase inhibitor
sorafenib
111
FGFR inhibitor, VEGFR inhibitor, RET inhibitor, PD1 inhibitor, c-KIT inhibitor, PDGFR α antagonist
pembrolizumab + lenvatinib
112
Tubulin polymerization promoter, PARP inhibitor
PARP inhibitor + carboplatin
113
Nectin-4-targeted antibody-drug conjugate, PD1 inhibitor, Microtubule inhibitor
pembrolizumab + enfortumab vedotin-ejfv
114
TROP-2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
sacituzumab govitecan-hziy
115
Topoisomerase II inhibitor, Tubulin polymerization promoter, DNA inhibitor
carboplatin + etoposide oral
116
Bifunctional alkylating agent, Tubulin polymerization promoter, Bcl2 inhibitor
paclitaxel + ifosfamide
117
VEGFR-1 inhibitor, VEGFR-2 inhibitor, VEGFR-3 inhibitor
tivozanib
goserelin acetate + flutamide
bicalutamide + goserelin acetate
bicalutamide + triptorelin
118
Androgen receptor inhibitor, GnRH agonist
triptorelin + flutamide
leuprolide acetate + bicalutamide
leuprolide acetate + flutamide
bicalutamide + histrelin acetate
histrelin acetate + flutamide
119
Tubulin polymerization promoter, DNA synthesis inhibitor, Bcl2 inhibitor
cisplatin + paclitaxel
gemcitabine + paclitaxel
120
GnRH antagonist, CYP17A1 inhibitor
abiraterone acetate + degarelix
121
DNA synthesis inhibitor, Thymidylate synthase inhibitor
cisplatin + 5-fluorouracil
5-fluorouracil + mitomycin
122
Bifunctional alkylating agent, Topoisomerase II inhibitor, DNA synthesis inhibitor
cisplatin + doxorubicin hydrochloride + ifosfamide + etoposide IV
gemcitabine + ifosfamide + pegylated liposomal doxorubicin
123
Topoisomerase II inhibitor, Tubulin polymerization promoter
carboplatin + etoposide IV
124
CD122 agonist, IL-2 stimulant
aldesleukin
125
TLR7 agonist, TLR8 agonist
imiquimod
126
Tubulin polymerization promoter, DNA synthesis inhibitor, DNA cross linking agent, Bcl2 inhibitor
gemcitabine + paclitaxel + oxaliplatin
127
FGFR inhibitor, VEGFR inhibitor, RET inhibitor, mTOR inhibitor, c-KIT inhibitor, PDGFR α antagonist
everolimus + lenvatinib
128
HER2 inhibitor, HER4 inhibitor, EGFR inhibitor
afatinib
129
PD-L1 inhibitor, Androgen receptor inhibitor
atezolizumab + enzalutamide capsule
130
PD-L1 inhibitor, CTLA4 inhibitor
durvalumab + tremelimumab
131
HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
fam-trastuzumab deruxtecan-nxki
SHR-A1811
132
Nectin-4-targeted peptide-drug conjugate, Microtubule inhibitor
BT8009
133
PSMA-targeted antibody-drug conjugate, Tubulin inhibitor
JNJ-8177
134
Cell death stimulant, GM-CSF agonist
CG0070
135
PD-L1 inhibitor, Multi-tyrosine kinase inhibitor
atezolizumab + cabozantinib tablet
136
FGFR2 inhibitor, FGFR inhibitor, FGFR1 inhibitor, FGFR3 inhibitor, PD1 inhibitor, FGFR4 inhibitor
erdafitinib + JNJ-63723283
137
HER2-targeted antibody-drug conjugate, Microtubule inhibitor
disitamab vedotin
ado-trastuzumab emtansine
138
PIK3CA inhibitor, PARP inhibitor, PI3Kδ inhibitor
rucaparib + copanlisib
139
Androgen receptor degrader, Androgen receptor inhibitor
ONCT-534
140
PD1 inhibitor, Androgen receptor inhibitor
pembrolizumab + enzalutamide capsule
141
PARP2 inhibitor, PARP1 inhibitor, CYP17A1 inhibitor
abiraterone / niraparib
142
PD1 inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor
toripalimab-tpzi + disitamab vedotin
tislelizumab + disitamab vedotin
143
IGF-2 inhibitor, Androgen receptor inhibitor, IGF1 inhibitor
enzalutamide capsule + BI-836845
144
PD-L1 inhibitor, PD1 inhibitor
durvalumab + MEDI0680
145
VEGFR inhibitor, PDGFR inhibitor, c-KIT inhibitor, FLT3 inhibitor
ABT-869
146
PD-L1 inhibitor, VEGF-A inhibitor, PI3Kγ inhibitor
bevacizumab + atezolizumab + IPI-549
147
TIM-1-targeted antibody-drug conjugate, Microtubule inhibitor
CDX-014
148
PD-L1 inhibitor, mTOR inhibitor, mTORC2 inhibitor
durvalumab + AZD2014
149
CYP17A1 inhibitor, Androgen receptor inhibitor, Androgen receptor antagonist
enzalutamide capsule + abiraterone acetate + apalutamide
150
PD-L1 inhibitor, CD47 inhibitor
atezolizumab + GS-4721
151
CD137 agonist, HER2 inhibitor
PRS-343
152
PD1 inhibitor, GDF15 inhibitor
nivolumab + CTL-002
153
STAT3 inhibitor, PD1 inhibitor
pembrolizumab + BBI608
154
Bifunctional alkylating agent, Topoisomerase II inhibitor, DNA inhibitor, DNA synthesis inhibitor
cisplatin + ifosfamide + etoposide oral
155
THF dehydrogenase inhibitor, Thymidylate synthase inhibitor
pemetrexed
156
STEAP1-targeted antibody-drug conjugate, Microtubule inhibitor
RG7450
157
PD-L1 inhibitor, VEGF-A inhibitor
bevacizumab + atezolizumab
158
Alkylating agent
cyclophosphamide
STAR-001
159
Topoisomerase II inhibitor, DNA synthesis inhibitor
etoposide IV + bleomycin
160
Ionizing radiation emitter, Androgen receptor inhibitor, PSMA inhibitor
enzalutamide capsule + lutetium Lu 177 vipivotide tetraxetan
161
PD1 inhibitor, HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
nivolumab + fam-trastuzumab deruxtecan-nxki
162
PD-L1 inhibitor, PI3K inhibitor, AKT inhibitor
atezolizumab + RG7440
163
B7-H3-targeted antibody-drug conjugate, Topoisomerase I inhibitor
DS-7300
164
Ionizing radiation emitter, PD1 inhibitor, PSMA inhibitor
pembrolizumab + lutetium Lu 177 vipivotide tetraxetan
165
VEGFR-2 inhibitor, c-MET inhibitor
GSK1363089
166
GnRH antagonist, CYP17A1 inhibitor, Androgen receptor antagonist
abiraterone acetate + degarelix + bicalutamide implant
167
AXL inhibitor, Multi-tyrosine kinase inhibitor, GAS6 inhibitor
cabozantinib tablet + AVB-500
168
Topoisomerase II inhibitor, Microtubule stabilizer, Tubulin polymerization promoter, Bcl2 inhibitor
paclitaxel + docetaxel + etoposide IV
169
VEGFR inhibitor, PDGFR inhibitor, Multi-tyrosine kinase inhibitor, c-KIT inhibitor
sunitinib + pazopanib
170
Glutathione peroxidase 4 inhibitor, Ferroptosis inducer
ML210
171
RAC1 inhibitor
NSC23766
172
C4.4a-targeted antibody-drug conjugate, Microtubule inhibitor
BAY1129980
173
MAT2A inhibitor
IDE397
174
EZH1 inhibitor, EZH2 inhibitor
CPI-0209
175
Ferroptosis inducer
erastin
RSL3
176
Bcr-abl tyrosine kinase inhibitor
INNO-406
MK-2206
177
AKT inhibitor
capivasertib
GSK690693
178
p53 reactivator
APR-246
APR-548
179
WEE1 inhibitor
AZD1775
180
FGFR inhibitor, VEGFR inhibitor, PDGFR inhibitor, pan-TRK inhibitor
TKI258
181
FGFR inhibitor, Bcr-abl tyrosine kinase inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib + infigratinib
182
DDX5 degrader
FL118
183
DNA methylation inhibitor
TdCyd
184
DNA synthesis inhibitor, Cytidine deaminase inhibitor, DNA methylation inhibitor
gemcitabine + EPI01
185
EZH2 inhibitor
GSK2816126
186
MEK2 inhibitor, MEK1 inhibitor
U0126
187
pan-RAF inhibitor, Hyaluronic acid synthase inhibitor, Multi-tyrosine kinase inhibitor
sorafenib + 4-methylumbelliferone
188
Androgen receptor antagonist, TMPRSS2 inhibitor
GT0918
189
WDR5 inhibitor
OICR-9429
190
AKT2 inhibitor, AKT1 inhibitor
BAY 1125976
191
Androgen receptor inhibitor, AKT inhibitor
enzalutamide capsule + capivasertib
192
ZG16B inhibitor
PBP1510
193
PIK3CA inhibitor, Androgen receptor inhibitor, PI3Kδ inhibitor
copanlisib + darolutamide
194
FGFR inhibitor, Androgen receptor inhibitor
enzalutamide capsule + Debio 1347
195
PRC2 inhibitor
MRTX2219
196
TGM2 inhibitor
MD102
197
BRD3 inhibitor, BRD4 inhibitor, BRD2 inhibitor
OTX015
198
B7-H3-targeted antibody-drug conjugate, DNA replication inhibitor
MGC018
199
ATR inhibitor
M6620
200
ROR1 inhibitor
UC-961
201
BTK inhibitor
ibrutinib
202
UCHL1 inhibitor, Androgen receptor inhibitor
enzalutamide capsule + 6RK73
203
MAPK inhibitor, p38 inhibitor
SB202190
204
CDK7 inhibitor
SY‑079
YPN-005
205
Integrin beta-6 -targeted antibody-drug conjugate, Microtubule inhibitor
SGN-B6A
206
Androgen receptor inhibitor, Microtubule inhibitor, PSMA-targeted antibody-drug conjugate
enzalutamide capsule + PSMA ADC
207
FGFR3-targeted antibody-drug conjugate, Microtubule inhibitor
LY3076226
208
SLC44A4-targeted antibody-drug conjugate, Microtubule inhibitor
ASG 5ME
209
DOT1L inhibitor
EPZ004777
EPZ-5676
210
KRAS G12C inhibitor
sotorasib
211
Bcr-abl tyrosine kinase inhibitor, mTOR inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib + AZD8055
212
PD-L1 inhibitor, NK cell stimulant
avelumab + CYNK-101
213
Adenosine A2A receptor antagonist
AZD4635
214
MEK1 inhibitor
cobimetinib
215
Adenosine A2A receptor antagonist, Androgen receptor antagonist
apalutamide + AZD4635
216
FGFR4 inhibitor
BLU 9931
217
EGFR inhibitor, IFN stimulant, TROP-2 inhibitor
ABN202
218
FGFR3-targeted antibody-drug conjugate, Topoisomerase I inhibitor
AMB302
219
KRAS G12C inhibitor, mTORC1 inhibitor
adagrasib + nanoparticle albumin-bound rapamycin
sotorasib + nanoparticle albumin-bound rapamycin
220
Androgen receptor inhibitor, ERK inhibitor, AKT inhibitor
darolutamide + ONC201
221
NF-κB inhibitor, SYK inhibitor
BAY-61-3606
222
CD3 agonist, STEAP1 inhibitor
AMG 509
223
Ionizing radiation emitter, CD37 inhibitor
177Lu-satetraxetan-lilotomab
224
HER2 inhibitor, EGFR inhibitor
lapatinib
225
PSMA-targeted CAR-T immunotherapy
AUTO7
226
Chk1 inhibitor, Chk2 inhibitor
ACR-368
227
CYP17A1 inhibitor, Androgen receptor inhibitor
enzalutamide capsule + abiraterone acetate
228
CD3 agonist, PSMA inhibitor
JNJ-63898081
229
HER3 inhibitor, α radiation emission
Ac-225 ErbB3 targeted radiotherapy
230
CA6-targeted antibody-drug conjugate, Microtubule inhibitor
SAR566658
231
DNA replication inhibitor, PSMA-targeted antibody-drug conjugate
MEDI3726
ADCT-212
232
Microtubule stabilizer, Tubulin polymerization promoter, Microtubule inhibitor
docetaxel + cabazitaxel
233
GnRH stimulant, CYP17A1 inhibitor, Androgen receptor antagonist
abiraterone acetate + bicalutamide implant + leuprorelin depot
234
CEACAM5-targeted antibody-drug conjugate, Topoisomerase I inhibitor
IMMU-130
235
CYP17A1 inhibitor, PI3K inhibitor, AKT inhibitor
abiraterone acetate + RG7440
236
MCL1 inhibitor
PRT1419
237
AXL-targeted antibody-drug conjugate, Microtubule inhibitor
BA3011
238
Aurora kinase A inhibitor
MLN8237
239
CDH6-targeted antibody-drug conjugate, Topoisomerase I inhibitor
CUSP06
240
pan-RAF inhibitor, VEGFR inhibitor, PDGFR inhibitor, Multi-tyrosine kinase inhibitor, c-KIT inhibitor
sorafenib + sunitinib
241
GPC-1-targeted antibody-drug conjugate
anti-GPC-1 ADC
242
Ionizing radiation emitter
radium Ra-223 dichloride
243
AR-V7 degrader
HSK38008
244
Androgen receptor inhibitor, AR-V7 degrader
enzalutamide capsule + HSK38008
245
PIK3C3 inhibitor, FGFR inhibitor
MPT0L145
No biomarker
PD-L1 expression
PD-L1 overexpression
TMB-H + PD-L1 expression
DDR + PD-L1 expression
PD-L1 underexpression
PD-L1 expression + T-cell gene signature
PD-L1 elevation
PD-L1 negative
FGFR3 mutation
FGFR3 fusion
FGFR3 R248C
FGFR3 Y373C
FGFR3 G370C
FGFR3 S249C
FGFR3 expression
FGFR3 rearrangement
FGFR3 Y375C
FGFR3 overexpression
FGFR3 G380R
FGFR3 A393E
FGFR3 L496V
FGFR3 S247C
FGFR3 K508M
FGFR3 V443M
FGFR3 V443L
MET amplification
MET mutation
MET fusion
MET expression
MSI-H/dMMR
PTEN deletion
PTEN mutation
PTEN negative
MSI-L/dMMR
PTEN expression
PTEN N323fs*21
PTEN overexpression
PTEN underexpression
AR wild-type
AR splice variant 7 negative
AR mutation
AR T878A
AR elevation
AR H875Y
AR T878S + AR H875Y
AR T878A + AR H875Y
AR T878S
AR overexpression
AR positive
AR F876L
AR splice variant 7
AR splice variant 7 expression
AR F877L
AR amplification
AR T877A
AR L329W
AR W741L
AR expression
AR H100Q
AR W741C
AR L702H
AR D891H
AR F877L + AR T878A
AR splice variant 9
TMB-H
FGFR mutation
BRCA2 mutation
BRCA2 deletion
BRCA2 positive
BRCA2 biallelic inactivation
FGFR fusion
FGFR overexpression
TMB-H + DDR
BRCA2 L557*
FGFR expression
BRCA2 A902fs*2
BRCA2 underexpression
BRCA2 amplification
BRCA2 exon 11 deletion
HER-2 positive
BRCA1 mutation
BRCA1 positive
HER-2 mutation
HER-2 overexpression
HER-2 expression
BRCA1 underexpression
BRCA1 deletion
BRCA1 N1018fs*8
HER-2 amplification
BRCA1 biallelic inactivation
BRCA1 expression
FANCL mutation
ERCC2 E606Q
ERCC2 D609E
ERCC2 D609G
ERCC2 G665A
ERCC2 mutation
ERCC2 N238S
ERCC2 E606G
ERCC2 P463L
ERCC2 V242F
ERCC2 Y24C
MTOR mutation
MTOR E2014K
MTOR E2419K
MTOR Q2223K
MTOR overexpression
FOLH1 expression
PBRM1 mutation
ATM positive
ATM mutation
ATM deletion
PBRM1 deletion
HRAS mutation
HRAS G13R
HRAS G12C
HRAS Q61R
HRAS H27_28fs*
HRAS G12S
FOLH1 overexpression
FOLH1 positive
PBRM1 overexpression
PBRM1 negative
HRAS Q61
PBRM1 underexpression
ATM biallelic inactivation
ATM underexpression
KDR rs2071559
FGFR2 fusion
FGFR2 mutation
KDR C482R
KDR expression
FGFR2 A391E
FGFR2 underexpression
KDR overexpression
RNASET2 overexpression
CD8 expression
FLT1 rs9554320
FGFR3-TACC3 fusion
TSC1 deletion
FGFR1 overexpression
TSC1 mutation
FGFR1 mutation
ERBB3 G284R
ERBB3 V104M
ERBB3 R103G
ERBB3 mutation
FGFR1 expression
FGFR3-TACC3 F17T8
FGFR1 amplification
CD8 overexpression
TSC1 deletion
FLT1 expression
TSC1 1907_1908del
ERBB3 expression
FLT1 overexpression
FGFR3-TACC3 fusion + FGFR3 V555M
HRD
AXL-L
ARID1A mutation
HLA-G positive
ROBO3 mutation
PD-1 expression
MSH2 deletion
MSH2 mutation
BAP1 mutation
BAP1 negative
BAP1 I696T
PD-1 overexpression
BAP1 deletion
AXL expression
AXL overexpression
PD-1 elevation
MTAP deletion
VHL mutation
SPOP mutation
ALK rearrangement
RB1 mutation
HDAC2 expression
FANCA deletion
BRCA2 mutation + ATM mutation
CTLA4 underexpression
CDK12 mutation
FH mutation
PALB2 mutation
TSC2 mutation
FANCA mutation
TFE3 translocation
MLH1 mutation
CYP17A1 expression
EGFR amplification
VCP-TFE3 fusion
TMB-H + PD-L1 negative
MSH6 mutation
PIK3CA mutation
PD-L1 expression + TMB-H
MSH2 mutation + MSH6 mutation
MSH2 negative + MSH6 negative
CYP17A1 V366M
PALB2 deletion
HMOX1-L
MSH6 deletion
HGF-L
HGF expression
EGFR L858R
TSC2 H1620R + TSC2 Y1650C
PIK3CA M1043I
MLH1 deletion
CTLA4 promoter hypomethylation
BRCA2 deletion + ATM mutation
CXCL10 expression
HMOX1 expression
WRN mutation
FH deletion
WRN expression
CXCL10 overexpression
HDAC2 mutation
CDK12 deletion
RB1 expression
VHL promoter methylation
ERBB3 mutation + TMB-H
HGF elevation
CXCL10 elevation
RB deletion
PIK3CA mutation + MSI-L/dMMR
PIK3CA amplification
MTAP mutation
FH negative
RB1 deletion
VHL deletion
KHDRBS1 overexpression
GNG4 overexpression
LRP1B mutation
CXCR3 overexpression
STEAP1 expression
BRCA1 mutation + ATM mutation
CPM elevation
Apolipoprotein B elevation
ITGAX underexpression
APH1A overexpression
NOTCH3 underexpression
PECAM1 underexpression
VTCN1 overexpression
TUBB1 rs151352
CYP2C8 rs1341164
TP53 mutation
SAAL1 overexpression
YBX1 rs10493112
DRD
EFNB2 expression
CD163 overexpression
CD68 overexpression
B2M overexpression
TNFRSF9 positive + CD4 positive
KDM6A mutation
CD3G overexpression
NCAM1 overexpression
TNFRSF9 positive + CD8 positive
CD4 underexpression
LAG3 positive + CD4 positive
CEACAM1 overexpression
PD-L1 expression + CD14 positive
PD-L2 overexpression
ATR mutation
BLM mutation
PMS1 expression
MLL2 mutation
FANCE expression
POLR2L expression
CD19 overexpression
PAX5 overexpression
PD-L1 overexpression + APOBEC3B overexpression
ELTD1 expression
NT5E underexpression
TNFRSF9 elevation
TMB-H + MLL2 mutation
TMB-H + KDM6A mutation
TMB-H + TERT promoter mutation
TMB-H + PIK3CA mutation
ISLR overexpression
FGFR2-CASP7 fusion
AXL elevation + GAS6 elevation
RAD50 mutation
FANCG mutation
FGFR2-BICC1 fusion
FANCI mutation
NECTIN4 expression
FANCM mutation
TGFB1 underexpression
TUBB3 overexpression
FGF10 amplification
PTTG1 overexpression
KDM5D overexpression
KIFC1 expression
PARP1 underexpression + PBRM1 mutation
CDKN2A mutation
FGF mutation
LAMP3 expression
CXCL10 overexpression + LAMP3 overexpression
EPHB2 expression
LDH elevation
PSMA1 overexpression
FGFR mutation + PD-L1 expression
CLDN6 expression
CD276 overexpression
CA9 expression
TP53 mutation + MDM2 mutation
SLC35A2 overexpression
CD31 expression
GBP5 expression
IFNG expression
CXCL9 expression
ITIH5 overexpression
PYCR1 underexpression
IGF1 overexpression
SRRM4 overexpression
TMEM72 underexpression
NPHS1 underexpression
NANOGNB mutation
TNFRSF18-H
SYNE1 mutation
IL18BP expression
CCDC69 overexpression
TLR3 overexpression
VEGFA expression
CSF1 expression
SNAI2 deletion
TIMP1 expression
WDR72 overexpression + PBRM1 mutation
WDR72 overexpression
BRCA2 mutation + SPOP mutation
TERT promoter mutation
BRAF mutation
ANGPT2 expression
TMB-H + PD-L1 expression + MSI-L/dMMR
IL18 expression
PBRM1 mutation + SETD2 mutation
MSI-H + MSH2 expression + MSH6 expression
ARID2 H1495fs*8
SMARCB1 deletion
RB1 mutation + PD-L1 expression
IL6-L
CXCL8-L
TLR4-L
SPP1-L
NRF1-BRAF fusion
GNAQ mutation
IKZF2-L
HAVCR2 expression
MSH4 L359I
KDM5C mutation
KMT2C mutation
ERVE-4 expression
PDGFRA expression
RNF43 mutation
AFP elevation
MSI-H/dMMR + TMB-H
miR-138 underexpression + miR-497 overexpression
RB1 mutation + TP53 mutation
EWSR1-POU5F1 fusion
PMS2 mutation + MLH1 mutation
MSH2 mutation + MSH6 mutation + BRCA1 mutation
NF2 mutation
BIRC5 expression
FGFR3-BAIAP2L1 fusion
AKT1 mutation + AR mutation
SETD2 mutation + TP53 mutation
PMS2 mutation
SND1-BRAF fusion
CHEK2 mutation
TMB-H + RB1 mutation + PD-L1 underexpression
TET1 mutation
FANCF mutation
FLCN mutation
KIM1 expression
BRIP1 mutation
CXCL13 expression
ATRX mutation
PCSK9 underexpression
SPOP mutation + CHD1 deletion
CXCL13 mutation + ARID1A mutation
TFEB translocation
HIF1A expression
CYB5A rs1790834
IFNA1 expression
BRCA1 mutation + TP53 mutation
BRCA2 mutation + TP53 mutation
BARD1 mutation
IL6ST elevation
RAD54L mutation
RAD51D mutation
IL6R L
RAD51C mutation
KRAS amplification
RAD51B mutation
CHEK1 mutation
CD93 underexpression
CREBBP mutation
ERCC1 underexpression
CALCR overexpression
CXCL13 elevation
CXCL8 elevation
KIM1 elevation
IL6 elevation
VEGFA elevation
KDM5D amplification
KDM6A amplification
CD276 expression
TP53 expression
PSMA1 expression
TP53 deletion
CDKN2A deletion
TP53 R175H
SETD2 mutation
SETD2 deletion
KRAS mutation
TERT overexpression
RAD51C expression
NT5E overexpression
NECTIN4 underexpression
CYP2C8 rs1058932
KRAS G12C
BRAF V595E
VEGFA overexpression
APOBEC mutagenesis
TSG gene expression signature
High MHC-II signature
Low MLR
DDR
Chr t(22)
AR-V7 expression
SBS5 signature
BONSAI high signature
Immune response prediction signature
T-cell-inflamed GEP signature
AR-V7 negative
IFNG 4-genes signature
IFNG gene signature
IFNG gene signature overexpression
12-CK gene signature
AR-V7 mutation
AP positive signature
Low NLR
MYC amplification
HLA-A*03
ETS rearrangment
ERG overexpression
ETV1 overexpression
SLC44A4 expression
RAC1 deletion
miR-155 underexpression
GAS5 underexpression
ALCAM elevation
CEACAM5 expression
SPINK1 overexpression
CA6 expression
HMGA2 overexpression
CD27 overexpression
IL7 elevation
GSDMB expression
STK11 expression
CDKN2B mutation
ESRP1-RAF1 fusion
SLC45A3-BRAF fusion
IRF8 expression
BTK overexpression
FLT3 overexpression
IL2R overexpression
ARG1 overexpression
ATM mutation + CDK12 mutation
CFLAR expression
SMARCA4 mutation
NOTCH1 mutation + MSI-L/dMMR
ELF3 mutation + MSI-L/dMMR
COL6A1 overexpression
SPI1 overexpression
EPAS1 G323E
ELF3 mutation + TMB-L + MSI-L/dMMR
AR-V7 positive
XPA expression
ZEB1 expression
SNAI1 expression
ADAMTS1 expression
KLK4 expression
KLK2 expression
FGF3 mutation
CCNE1 amplification
CTBP1 deletion
ACRBP amplification
GNAS amplification
LRP10 deletion
TMB-H + CDKN2B mutation
TMB-L + RB1 mutation
KRT20 overexpression
H19 overexpression
FGF4 mutation
FGF19 mutation
SULT1A3 amplification
NOTCH1 mutation + TMB-L + MSI-L/dMMR
BRCA2 mutation + CHEK2 mutation
BRCA2 mutation + CDK12 mutation
AKT1 mutation
KDM4B overexpression
NRAS G12D
TMPRSS2-ERG fusion
UGT1A9 expression
KIT mutation
ADCYAP1 deletion
NOTCH1 deletion
EPAS1 S304M
BRCA1 mutation + BRCA2 mutation
IL20RB overexpression
EPAS1 overexpression
CD44 positive
EZH2 amplification
DNMT3A amplification
PREX2 amplification
PIK3CB amplification
SLC3A2 expression
GPX4 expression
CD44 expression
SLC7A11 expression
ACSM3 overexpression
BRCA2 deletion + RB1 deletion
ACSM1 overexpression
SALL4 positive + POU5F1 positive + KIT positive + PLAA positive
BBOX1 underexpression
HER-2 mutation + TMB-H
YTHDC1 underexpression
TERC overexpression
DKC1 overexpression
LYPD3 expression
ZRANB1 overexpression
TUBA1C overexpression
Chr del(9)(p21.3)
TNFSF13B elevation
IL13RA2 overexpression
FGF4 amplification + HRAS Q61R + TP53 672+2T>G
FSCN1 elevation
AXL overexpression + PD-L1 expression
NUSAP1 overexpression
High NLR
DDX39B overexpression
FGF3 amplification + HRAS Q61R + TP53 672+2T>G
CYP11B1 rs4736349
FGF19 amplification + HRAS Q61R + TP53 672+2T>G
PD-1-L + PD-L1 elevation
CXCL11 elevation
NEIL3 deletion
PTGR1 elevation + HRD
HYAL4 V1
FGFR2 underexpression + FGFR3 overexpression
BAX underexpression
TET2 deletion + DNMT3A mutation
FGFR2 underexpression + FGFR3 mutation
miR-572 overexpression
PAI1 elevation
ITGB6 expression
WDR5 overexpression
CXCR4 overexpression
TDO2 overexpression
CXCL12 elevation
ZG16B positive
GPC1 overexpression
PLK1 overexpression
SNHG1 deletion
CDH6 expression
TGM2 overexpression
AR-V7 overexpression
CCL4 elevation
OXCT1 expression
ROR1 expression
WNT5A overexpression + FZD2 overexpression
PRCC-TFE3 fusion
RAD52 underexpression
HSD3B1 1245A>C
MTA2 overexpression
LAG3 expression
PGF overexpression
VEGFC underexpression
PDGFA underexpression
TSPYL1 P62S
PHLPP1 deletion
FLT4 overexpression
ZFHX3 deletion
VEGFD overexpression
SPARC amplification
PD-L1 expression + REV3L overexpression
VEGFB overexpression
PD-L1 expression + MTOR overexpression
MCAM overexpression
KAT6A-NRG1 fusion
PTEN deletion + KRAS G12C
CD70 expression
HDAC5 deletion
HAS3 expression
ACTA2 underexpression
FOXA mutation
AR expression + CYP17A1 expression
AKR1C3 expression
CHD1 deletion
PPP2R2A mutation
SRF overexpression
DAPK1 underexpression
PLAC8 overexpression
SOX2 expression
MYCN amplification
MAST4 mutation
FGFR4 amplification
TROP2 positive
MTAP mutation + CDKN2A mutation
Chr del(10)
HLA-DQB1*03:01