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Association details:
Evidence:
Evidence Level:
Sensitive: C4 – Case Studies
New
Title:

SHP2 Inhibition Sensitizes Diverse Oncogene-Addicted Solid Tumors to Re-treatment with Targeted Therapy

Published date:
08/04/2023
Excerpt:
A patient with GOPC–ROS1 fusion–positive pancreatic adenocarcinoma was previously treated with gemcitabine + abraxane + nivolumab followed by repotrectinib (progressed after ∼10 months...After 6 weeks of monotherapy, imaging demonstrated progressive disease in two target lesion liver metastases (+26% overall), together with an increase in the GOPC–ROS1 and CTNNB1 S45F in ctDNA...The patient continued PF-07284892, and lorlatinib was added at 100 mg qd. After 2 weeks of combination (study week 8), both mutations in ctDNA decreased by 95% compared with baseline before starting any study treatment...After 6 weeks of combination (study week 12), target liver lesions decreased by −35% compared with precombination imaging consistent with PR, confirmed after 12 weeks of combination...
DOI:
https://doi.org/10.1158/2159-8290.CD-23-0361