^
Association details:
Biomarker:GNAQ Q209L
Cancer:Uveal Melanoma
Drug:U0126 (MEK1 inhibitor, MEK2 inhibitor)
Direction:Sensitive
Evidence:
Evidence Level:
Sensitive: D – Preclinical
New
Source:
Title:

Frequent somatic mutations of GNAQ in uveal melanoma and blue nevi

Excerpt:
Conversely, siRNA-mediated knock-down of GNAQ in the uveal melanoma cell line, OMM1.3, which harbors the GNAQ-Q209L mutation, resulted in a decrease of phospho-ERK levels (Figure 3a)....Knockdown of GNAQ in OMM1.3 cells results in MAP-kinase inhibition, reduced growth and apoptosis...After 72 hours, GNAQ knockdown results in marked reduction of cell numbers, similar to the effect of MEK inhibitor U0126.
DOI:
10.1038/nature07586