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Association details:
Evidence:
Evidence Level:
Resistant: D – Preclinical
New
Title:

The ALK inhibitor ceritinib overcomes crizotinib resistance in non-small cell lung cancer

Excerpt:
However, we observed that ceritinib did not overcome two crizotinib-resistant ALK mutations, G1202R and F1174C, and one of these mutations were identified in 5 out of 11 biopsies from patients with acquired resistance to ceritinib….In the wild-type and I1171T resistant models, ceritinib demonstrated impressive anti-tumor activity, while it was less active in the C1156Y resistant model and was inactive against the G1202R resistant model.
DOI:
10.1158/2159-8290.CD-13-0846