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Association details:
Evidence:
Evidence Level:
Resistant: C4 – Case Studies
Title:

Acquired Resistance Mutations to ALK Inhibitors Identified by Single Circulating Tumor Cell Sequencing in ALK-Rearranged Non-Small-Cell Lung Cancer

Published date:
08/22/2019
Excerpt:
We asked whether single circulating tumor cell (CTC) sequencing can inform on resistance mutations to ALK inhibitors and underlying tumor heterogeneity in ALK-rearranged NSCLC....Mutations were examined in CTCs from three patients (P41, P45, and P48) resistant to lorlatinib.At PD on lorlatinib, the patient underwent a tumor biopsy and was sampled for CTC analysis. ALKG1202R and ALKF1174L were detected with a VAF of 29% and 9% respectively in the tumor biopsy...CTC-10 harbored ALKG1202R/T1151M compound mutation with a VAF of 98% and 100% respectively...
DOI:
10.1158/1078-0432.CCR-19-1176