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BIOMARKER:
PIK3R1 mutation
i
Other names:
PIK3R1, Phosphoinositide-3-Kinase Regulatory Subunit 1, Phosphatidylinositol 3-Kinase 85 KDa Regulatory Subunit Alpha, Phosphoinositide-3-Kinase, Regulatory Subunit 1 (Alpha), Phosphatidylinositol 3-Kinase Regulatory Subunit Alpha, Phosphoinositide-3-Kinase Regulatory Subunit Alpha, PtdIns-3-Kinase Regulatory Subunit Alpha, PI3K Regulatory Subunit Alpha, PI3-Kinase Subunit P85-Alpha, GRB1, Phosphatidylinositol 3-Kinase, Regulatory Subunit, Polypeptide 1 (P85 Alpha), Phosphatidylinositol 3-Kinase
Associations
(3)
News
Trials
C3 | Sensitive
D | Sensitive
C3 | Resistant
D | Resistant
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Include preclinical:
Drug categories
Tyrosine Kinase Inhibitors
FGF
Serine-Threonine Kinase Inhibitors
PI3 Kinase Inhibitors
Other
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Endometrial Cancer
Hormone Receptor Positive Breast Cancer
Breast Cancer
LY3023414
C3
PIK3R1 mutation
|
Endometrial Cancer
|
LY3023414
lenvatinib
C3
PIK3R1 mutation
|
Hormone Receptor Positive Breast Cancer
|
lenvatinib
alpelisib + L-NMMA
D
PIK3R1 mutation
|
Breast Cancer
|
alpelisib + L-NMMA
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