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CANCER:

Gastric Cancer





Show legend
Group by Gene:
Include preclinical:

PD1 inhibitor
nivolumab
pembrolizumab
sintilimab
tislelizumab
0
PD1 inhibitor
camrelizumab
toripalimab-tpzi
dostarlimab-gxly
zimberelimab
pucotenlimab
PDR001
HER2 inhibitor
trastuzumab
trastuzumab-anns
trastuzumab-qyyp
trastuzumab-dkst
Zercepac (trastuzumab biosimilar)
trastuzumab-pkrb
1
HER2 inhibitor
ZW25
trastuzumab-dttb
Her-VAXX
AST-301
KN026
trastuzumab + tucatinib
tucatinib
trastuzumab-IFN-β mutein
5-fluorouracil
2
Thymidylate synthase inhibitor
capecitabine
raltitrexed
PD-L1 inhibitor
durvalumab
3
PD-L1 inhibitor
envafolimab
atezolizumab
sugemalimab
avelumab
4
DNA synthesis inhibitor, Thymidylate synthase inhibitor
cisplatin + capecitabine
cisplatin + 5-fluorouracil
5
VEGFR-2 inhibitor
ramucirumab
rivoceranib
6
CTLA4 inhibitor
tremelimumab
zolbetuximab
7
CLDN18.2 inhibitor
ZL-1211
TST001
AB011
8
DNA synthesis inhibitor, DNA cross linking agent, Thymidylate synthase inhibitor
5-fluorouracil + oxaliplatin
capecitabine + oxaliplatin
9
Thymidine phosphorylase inhibitor
trifluridine / tipiracil
10
Topoisomerase I inhibitor
irinotecan
11
Tubulin polymerization promoter, Bcl2 inhibitor
paclitaxel
carboplatin + paclitaxel
12
DNA synthesis inhibitor, DNA cross linking agent
oxaliplatin
13
DNA synthesis inhibitor, Topoisomerase I inhibitor
cisplatin + irinotecan
14
Thymidylate synthase inhibitor, Topoisomerase I inhibitor
5-fluorouracil + irinotecan
15
FGFR2b inhibitor
AMG 552
16
HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
fam-trastuzumab deruxtecan-nxki
SHR-A1811
FGFR inhibitor
infigratinib
futibatinib
17
FGFR inhibitor
ABSK091
ARQ 087
KIN-3248
Debio 1347
nivolumab + ramucirumab
camrelizumab + rivoceranib
18
VEGFR-2 inhibitor, PD1 inhibitor
tislelizumab + rivoceranib
pembrolizumab + ramucirumab
toripalimab-tpzi + rivoceranib
19
VEGF-A inhibitor
bevacizumab
20
PD1 inhibitor, CTLA4 inhibitor
nivolumab + ipilimumab
cadonilimab
savolitinib
tepotinib
ARQ 197
RG3638
21
c-MET inhibitor
S95027
savolitinib + capmatinib
AMG 102
SGX523
JNJ-38877605
pembrolizumab + trastuzumab
pembrolizumab + margetuximab
nivolumab + trastuzumab
22
HER2 inhibitor, PD1 inhibitor
margetuximab + retifanlimab-dlwr
tislelizumab + ZW25
trastuzumab + camrelizumab
trastuzumab + tislelizumab
23
PI3Kβ inhibitor
AZD8186
GSK2636771
24
DKK1 protein inhibitor
DKN-01
25
Gastrin-17 inhibitor
PAS
26
TrkB receptor inhibitor, TrkC kinase inhibitor, TrkA receptor inhibitor
larotrectinib
27
VEGFR-2 inhibitor, HER2 inhibitor
trastuzumab + ramucirumab
trastuzumab + ramucirumab + tucatinib
EGFR inhibitor
cetuximab
28
EGFR inhibitor
GC-1118A
WZ4002
CL-387785
CLDN18.2-targeted CAR-T immunotherapy
29
CLDN18.2-targeted CAR-T immunotherapy
IBI-345
CT041
30
DNA synthesis inhibitor
cisplatin
31
VEGFR inhibitor, FGFR1 inhibitor, PD1 inhibitor
toripalimab-tpzi + surufatinib
32
Microtubule inhibitor
cabazitaxel
33
ALK inhibitor
crizotinib
34
STAB1 inhibitor
bexmarilimab
pazopanib
35
Multi-tyrosine kinase inhibitor
regorafenib
ponatinib
nintedanib
36
PIK3CA inhibitor
CYH33
alpelisib
PARP inhibitor
37
PARP inhibitor
olaparib
ABT-888
38
DKK1 protein inhibitor, PD1 inhibitor
tislelizumab + DKN-01
pembrolizumab + DKN-01
39
PD-L1 inhibitor, TGF-β R2 kinase inhibitor
SHR-1701
40
PD1 inhibitor, LAG-3 inhibitor
sintilimab + IBI110
41
CLDN18.2 inhibitor, CD137 agonist
TJ-CD4B
42
mTOR inhibitor, mTORC2 inhibitor
AZD2014
43
AKT inhibitor
capivasertib
44
CD19-targeted CAR-T immunotherapy
AT101
45
HER2-targeted antibody-drug conjugate, Tubulin inhibitor
A166
46
BRAF inhibitor, BRAF V600E inhibitor
vemurafenib
47
HER2 inhibitor, HER3 inhibitor
MCLA-128
48
PD-L1 inhibitor, CD137 agonist
PM1003
49
PD-L1 inhibitor, Multi-tyrosine kinase inhibitor
durvalumab + cabozantinib tablet
anlotinib + APL-502
50
VEGFR-2 inhibitor, HER2 inhibitor, CD47 inhibitor
trastuzumab + ramucirumab + ALX148
51
NK cell stimulant
CYNK-101
52
HER2 inhibitor, CD47 inhibitor
D3L-001
53
PD-L1 inhibitor, HER2 inhibitor
trastuzumab + avelumab
54
Aromatase inhibitor
letrozole
55
HER2 inhibitor, HER2 dimerization inhibitor
trastuzumab + pertuzumab
56
MEK inhibitor, BRAF inhibitor
trametinib + dabrafenib
57
RET inhibitor
selpercatinib
58
ATR inhibitor
M6620
SC0245
59
PD1 inhibitor, CTLA4 inhibitor, CD47 inhibitor
cadonilimab + AK117
60
HER2 inhibitor, γδ TCR modulator
Undisclosed allogeneic Vγ9Vδ2 HER2-TAC T
61
PD-L1 inhibitor, PARP inhibitor
olaparib + durvalumab
62
Tubulin polymerization promoter
carboplatin
63
PD1 inhibitor, Multi-tyrosine kinase inhibitor
nivolumab + regorafenib
ECF
TPF
DOF
TCF
FP
CaT
64
Chemotherapy
FOLFIRI
CAPOX
DP
FLOT
IP
FOLFOX
TEX
65
Immunotherapy
Immunotherapy
66
CLDN18.2-targeted antibody-drug conjugate
CLDN18.2-targeted antibody-drug conjugate
ATG-022
67
EZH2 inhibitor
EZH2 inhibitor
68
c-MET-targeted CAR-T immunotherapy
c-MET-targeted CAR-T immunotherapy
69
FGFR21 inhibitor
FGFR21 inhibitor
70
PD-L1-targeted CAR-T immunotherapy
PD-L1-targeted CAR-T immunotherapy
disitamab vedotin
ado-trastuzumab emtansine
JNJ-0683
71
HER2-targeted antibody-drug conjugate, Microtubule inhibitor
ZW49
PF-06804103
MRG002
XMT-1522
72
PD-L1 inhibitor, CTLA4 inhibitor
durvalumab + tremelimumab
73
Microtubule stabilizer, Tubulin polymerization promoter, Topoisomerase I inhibitor
docetaxel + irinotecan
74
Tubulin polymerization promoter, Bcl2 inhibitor, Thymidylate synthase inhibitor
paclitaxel + capecitabine
paclitaxel + 5-fluorouracil
75
Microtubule stabilizer, Tubulin polymerization promoter, DNA synthesis inhibitor, Thymidylate synthase inhibitor
cisplatin + docetaxel + 5-fluorouracil
76
Tubulin polymerization promoter, DNA synthesis inhibitor, Bcl2 inhibitor
cisplatin + paclitaxel
77
Microtubule stabilizer, Tubulin polymerization promoter, Thymidylate synthase inhibitor
carboplatin + docetaxel + 5-fluorouracil
78
Microtubule stabilizer, Tubulin polymerization promoter, DNA synthesis inhibitor
cisplatin + docetaxel
79
Microtubule stabilizer, Tubulin polymerization promoter
docetaxel
AZD0901
80
CLDN18.2-targeted antibody-drug conjugate, Microtubule inhibitor
EO-3021
BMS-986476
pyrotinib
81
HER2 inhibitor, HER4 inhibitor, EGFR inhibitor
ASLAN001
afatinib
neratinib
82
TrkB receptor inhibitor, TrkC kinase inhibitor, ROS1 inhibitor, TrkA receptor inhibitor, ALK inhibitor, JAK2 inhibitor, TNK2 inhibitor
entrectinib
83
CEACAM5-targeted antibody-drug conjugate, Microtubule inhibitor
SAR408701
84
Tubulin polymerization promoter, HSP70 inhibitor, Bcl2 inhibitor
paclitaxel + minnelide
85
PDGFR inhibitor, Bcr-abl tyrosine kinase inhibitor, c-KIT inhibitor
imatinib
86
VEGFR inhibitor, PDGFR inhibitor, c-KIT inhibitor
sunitinib
87
HER2 inhibitor, EGFR inhibitor
lapatinib
88
FGFR2 inhibitor, FGFR inhibitor, FGFR1 inhibitor, FGFR3 inhibitor, FGFR4 inhibitor
erdafitinib
89
c-MET inhibitor, CSF-1R inhibitor, Src kinase inhibitor
TPX-0022
90
PD-L1 inhibitor, VEGF-A inhibitor, TGF-β R2 kinase inhibitor
bevacizumab + SHR-1701
91
VEGF-A inhibitor, Folate receptor 1-targeted antibody-drug conjugate, Microtubule inhibitor
bevacizumab + mirvetuximab soravtansine-gynx
92
TGFβ inhibitor, PD-L1 inhibitor
M7824
93
HER2 inhibitor, HER4 inhibitor, PD1 inhibitor, EGFR inhibitor
camrelizumab + pyrotinib
94
PD-L1 inhibitor, HER2 inhibitor, CTLA4 inhibitor
KN046 + KN026
95
CLDN18.2-targeted antibody-drug conjugate, DNA replication inhibitor
SOT102
96
CLDN18.2 inhibitor, CD3 agonist
ASP2138
AZD5863
97
Tubulin polymerization promoter, DNA synthesis inhibitor, Bcl2 inhibitor, Thymidylate synthase inhibitor
cisplatin + paclitaxel + capecitabine
98
FGFR inhibitor, VEGFR inhibitor, RET inhibitor, PD1 inhibitor, c-KIT inhibitor, PDGFR α antagonist
pembrolizumab + lenvatinib
99
ADAM9-targeted antibody-drug conjugate, Microtubule inhibitor
IMGC936
100
HER2 inhibitor, HER4 inhibitor, CDK4 inhibitor, EGFR inhibitor, CDK6 inhibitor
pyrotinib + dalpiciclib
101
CD137 agonist, HER2 inhibitor
PRS-343
102
VEGFR-2 inhibitor, Caprin-1 inhibitor
ramucirumab + TRK-950
103
ATR inhibitor, PD-L1 inhibitor
durvalumab + AZD6738
104
HER2 inhibitor, ALK inhibitor
trastuzumab + crizotinib
105
CLDN18.2 inhibitor, PD-L1 inhibitor
Q-1802
106
SLC44A4-targeted antibody-drug conjugate, Microtubule inhibitor
ASG 5ME
107
Protein synthesis inhibitor, HER2 inhibitor
MT-5111
108
TIGIT inhibitor, PD1 inhibitor
pembrolizumab + MK-7684
zimberelimab + AB154
109
PD1 inhibitor, PORCN inhibitor, Wnt signalling pathway inhibitor
pembrolizumab + CGX1321
110
c-MET-targeted antibody-drug conjugate, DNA replication inhibitor
BYON3521
111
PD1 inhibitor, HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
nivolumab + fam-trastuzumab deruxtecan-nxki
112
VEGFR inhibitor, PD1 inhibitor
sintilimab + fruquintinib
vorinostat
113
HDAC inhibitor
MGCD0103
SB939
114
HDAC inhibitor, HDAC1 inhibitor, HDAC2 inhibitor, HDAC3 inhibitor
entinostat
115
MYC inhibitor
WB100
116
KRAS G12C inhibitor
APG-1842
117
CDK9 inhibitor
KB-0742
118
HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor, WEE1 inhibitor
fam-trastuzumab deruxtecan-nxki + AZD1775
119
ALPP-targeted antibody-drug conjugate, ALPPL2-targeted antibody-drug conjugate, Microtubule inhibitor
SGN-ALPV
120
HER2-targeted antibody-drug conjugate, STING agonist
XMT-2056
121
TGM2 inhibitor
MD102
122
AKT3 inhibitor, AKT1 inhibitor, AKT inhibitor, p70S6K inhibitor
DIACC3010
123
Bcr-abl tyrosine kinase inhibitor, HER2 inhibitor, HER4 inhibitor, EGFR inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib + neratinib
124
Cyclin modulator
ON 013105
125
FGFR2b inhibitor, FGF7 inhibitor
GB2102
126
CLDN18.2 inhibitor, CD137 agonist, PD1 inhibitor
nivolumab + TJ-CD4B
127
CDK2 inhibitor
INX-315
128
HER2 inhibitor, CD47 inhibitor, HER2 dimerization inhibitor
pertuzumab + D3L-001
129
MUC1-targeted antibody-drug conjugate, HER3-targeted antibody-drug conjugate
DM002
130
HER2 inhibitor, EGFR inhibitor, Multi-tyrosine kinase inhibitor
AEE788
131
PI3K inhibitor
MEN1611
132
FGFR inhibitor, c-MET inhibitor
WXSH0011
133
BET inhibitor, BRD4 inhibitor
SRA515
134
Bcr-abl tyrosine kinase inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib
135
STAT3 inhibitor
BBI608
136
c-MET-targeted antibody-drug conjugate, 5T4-targeted antibody-drug conjugate
DM004
137
PLK1 inhibitor
NBL-001
138
PLK1 inhibitor, BRD4 inhibitor
BI2536
139
HER2 inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor
ado-trastuzumab emtansine + AST-301
140
TROP-2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
sacituzumab govitecan-hziy
141
Microtubule inhibitor, TROP-2-targeted antibody-drug conjugate
LCB84
142
Bcl2 inhibitor, Bcl-xL inhibitor
APG-1252
143
Macrophage modulator
HF-CAR-PMs
144
PI3K inhibitor, mTOR inhibitor
RTB101
145
MCL1 inhibitor, Bcl2 inhibitor, Bcl-xL inhibitor
AT 101
146
MAT2A inhibitor
IDE397
147
HER2 inhibitor, EGFR inhibitor, Bcl2 inhibitor, Bcl-xL inhibitor
lapatinib + APG-1252
148
HER2 inhibitor, NK cell stimulant
trastuzumab + CYNK-101
149
p53 reactivator
PC14586
150
HER2-targeted antibody-drug conjugate, Microtubule inhibitor, HER2 dimerization inhibitor
pertuzumab + ado-trastuzumab emtansine
151
CDK4 inhibitor, CDK6 inhibitor
abemaciclib
152
Topoisomerase II inhibitor, HER2 inhibitor, HER2-targeted antibody-drug conjugate
trastuzumab + MM-302
153
c-MET inhibitor, HER2 inhibitor
trastuzumab + savolitinib
154
5T4-targeted antibody-drug conjugate, Microtubule inhibitor
ASN004
155
c-MET-targeted antibody-drug conjugate, Topoisomerase I inhibitor
HRA00129-C004
156
ICAM-1-targeted CAR-T immunotherapy
AIC100
157
DNMT inhibitor
decitabine
158
AKT3 inhibitor, HER2 inhibitor, AKT1 inhibitor, AKT inhibitor, p70S6K inhibitor
trastuzumab + DIACC3010
No biomarker
HER-2 negative
HER-2 positive
HER-2 expression
HER-2 overexpression
HER-2 amplification
HER-2 positive + HER-2 amplification
HER-2 underexpression
HER-2 mutation
HER-2 expression + HER-2 amplification
HER-2 mutation + HER-2 positive
HER-2 S310Y
HER-2 L755S
HER-2 V777L
HER-2 T862A
HER-2 1899‐1G>A
HER-2 expression + HER-2 D769H
HER-2 expression + HER-2 L869R
PD-L1 expression
PD-L1 overexpression
PD-L1 amplification
PD-L1 underexpression
MSI-H/dMMR
CLDN18.2 expression
CLDN18.2 positive
CLDN18.2 overexpression
CLDN18 fusion
CLDN18.2 underexpression
MET amplification
FGFR2 fusion
MET mutation
FGFR2 amplification
FGFR2b overexpression
MET overexpression
FGFR2b expression
FGFR2 mutation
MET exon 14 mutation
FGFR2b positive
FGFR2 overexpression
MET expression
MET positive
FGFR2 N549K
HER-2 negative + PD-L1 expression
HER-2 positive + PD-L1 expression
HER-2 amplification + PD-L1 expression
PD-L1 expression + HER-2 overexpression
CLDN18.2 positive + HER-2 negative
CLDN18.2 expression + HER-2 negative
DKK1 overexpression
EGFR overexpression
HER-2 expression + TMB-H
TMB-H + HER-2 positive
EGFR mutation
EGFR amplification
HER-2 elevation + TMB-H
HER-2 elevation + TMB-L
VEGFA elevation
NRP1 elevation
KDM6A mutation
FGFR2b overexpression + HER-2 negative
VSNL1 underexpression + CD44 underexpression
PIK3CA mutation
CEACAM5 positive
CEACAM5 expression
PIK3CA E545K
CEACAM5 overexpression
PIK3CA amplification
VEGFA overexpression
KDM6A underexpression
PIK3CA E542K
NTRK3 fusion
TMB-H
BRAF V600E
ERBB3 V104L + HER-2 negative
TP53 mutation
IL6 elevation
ATM underexpression
ATM mutation
EGFR amplification + ERBB2 amplification
IL6 expression
PD-1 expression
EGFR expression + HER-2 expression
FGFR3 mutation
TP53 wild-type
PD-1 overexpression
ERBB3 V104L
FGFR3 amplification
TP53 Y220C
ATM expression
TMB-L
ATM overexpression
TP53 R175H
TNFA-L
CLDN18-ARHGAP fusion
FGFR1 amplification
MSI-H/dMMR + POLE mutation
POLD1 mutation
POLE mutation
CCKBR expression
ERBB4 mutation + HER-2 positive
HLA-A*02
PIK3R1 M326I
NF1 mutation + HER-2 positive
IFNG-L
ITGAM overexpression + LAG3 overexpression
ITGAM overexpression + CTLA4 overexpression
PMS2 mutation
CPEB1 underexpression
ACTA2 underexpression
MLH1 mutation
CAPRIN-1 expression
PIK3CB mutation
RSPO3 fusion
IL2 expression
PMS2 mutation + MLH1 mutation
MSH2 mutation
MFSD2A overexpression
SLC44A4 expression
INHBA overexpression
PDGFRA mutation
KIT exon 11 mutation
VEGFC elevation
CFB overexpression
MSH6 mutation
RICTOR amplification
ER positive
MSI-H/dMMR + MLH1 negative + PMS2 negative
HER-2 amplification + MET amplification
PTEN deletion
ADAM9 expression
POLD2 mutation
PMS1 mutation
MSH3 mutation
MLH3 mutation
TYMS expression
LAG3 expression
RET fusion
TNFRSF4 expression
TGFB1 elevation
HRD
FOLR1 overexpression
NTRK1 fusion
ATRX mutation
ATR mutation
NTRK2 fusion
ARID1A mutation
ICAM1 elevation
CXCL8 elevation
TET1 mutation
WIF1 unmethylation
RASSF1 methylation
FGFR3-TACC3 fusion
CTAG1A expression
SMARCA4 mutation
NQO1 overexpression
PIK3CA mutation + HER-2 positive
PIK3R1 mutation + HER-2 positive
PIK3C3 mutation + HER-2 positive
GAST expression
MET expression + HER-2 expression
PTEN mutation
ACTA2 overexpression
PDGFRA D842Y
PDGFRA D846Y
PDGFRA DI842_843IM
PDGFRA Y849K
FGFR1 overexpression
PDGFRA D842V
FGFR1 mutation
ICAM1 overexpression
KIT exon 9 mutation
ARID1A deletion
PDGFRA exon 12 mutation
PDGFRA HDSN845_848P
PDGFRA N659K
PDGFRA N848K
PDGFRA RD841_842KI
MET overexpression + HER-2 overexpression
IFNG 6-gene signature
18-gene expanded immune signature
S100A10 overexpression
FGFR overexpression
MUS81 overexpression
STAT3 expression
NFKB1 expression
HER-2 overexpression + CCNE1 amplification
CCNA2 expression
ALPP expression
Chr del(13)(q12.12)
PTEN mutation + MSI-H/dMMR
MSI-H/dMMR + TMB-L
CRKL amplification
SNHG5 overexpression
HER-2 overexpression + PTEN deletion
CEACAM6 overexpression
CCNE1 amplification
FGFR4 amplification
SKAP1 overexpression
FGFR4 mutation
CDKN2B deletion
CD47 positive + HER-2 positive
CDKN2A deletion
MDM4 amplification
MDM2 amplification
VEGFB overexpression
Chr amplification(11)(q13)
TGM2 overexpression
BCL2 overexpression + MCL1 overexpression
BCAR4 overexpression
TUBB3 overexpression
MAP3K1 rs889312
MTAP deletion
TPBG expression + MET expression
GPR176 overexpression
TACC2-FGFR2 fusion
KRAS mutation + HER-2 positive
MAP3K10 R304C
MAP3K10 H211R
MAP3K10 A30E
ERBB3 expression + MUC1 expression
TROP2 expression
LDH elevation
ALPG expression
CDKN2A promoter methylation
HER-2 positive + GATA6 amplification
HER-2 positive + APC mutation
HER-2 positive + MYC amplification
KRAS mutation
MTA2 expression
TPBG underexpression + HER-2 overexpression
TGFBR2 P525L
TGFBR2 P129Afs*3
TGFBR2 E269*
RHOA L57V
KRAS G12R
CMTM4 expression + PD-L1 expression
RHOA D45N
RHOA L69P
CMTM6 expression + PD-L1 expression
APC V2194fs + EGFR amplification + EGFR-SEPTIN14 fusion
LINC00963 overexpression
miR-200-b underexpression
miR-199b overexpression + miR-152 overexpression
PREX2 M627V
PREX2 W519G
PREX2 R1567Q
MSI-H/dMMR + TMB-H
IGF2R overexpression
miR-152 overexpression
HER-2 positive + CAV1 overexpression
miR‐223 overexpression
DNMT3A overexpression
ATG5 overexpression
miR-199b overexpression
BCL2L1 overexpression
miR-103a underexpression
miR-200b underexpression + miR-103a underexpression
SOX17 methylation
CDH1 deletion
HOTAIR overexpression
MET overexpression + MUC5B overexpression
CD73 overexpression
MYC overexpression
CDH1 mutation
AREG overexpression
KRAS G12C
MYC amplification
miR‑106-a expression
NLRP6 overexpression
ARPP19 overexpression
CD44 expression
ERBB2 G778A + CCNE1 amplification
HER-2 underexpression + CCNE1 amplification
HER-2 amplification + CCNE1 expression