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BIOMARKER:
FLT3 D835
i
Other names:
FLT3, Fms Related Tyrosine Kinase 3, Receptor-Type Tyrosine-Protein Kinase FLT3, Stem Cell Tyrosine Kinase 1, Fms-Like Tyrosine Kinase 3, CD135, FLK-2, STK1, Growth Factor Receptor Tyrosine Kinase Type III, Fetal Liver Kinase 2
Associations
(8)
News
Trials
C2 | Sensitive
C3 | Sensitive
D | Sensitive
C2 | Resistant
C3 | Resistant
D | Resistant
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Include preclinical:
Drug categories
Tyrosine Kinase Inhibitors
Serine-Threonine Kinase Inhibitors
Heat Shock Protein Inhibitors
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Acute Myelogenous Leukemia
Chronic Myeloid Leukemia
gilteritinib
C2
FLT3 D835
|
Acute Myelogenous Leukemia
|
gilteritinib
ARO-002
C2
FLT3 D835
|
Acute Myelogenous Leukemia
|
ARO-002
midostaurin
C2
FLT3 D835
|
Acute Myelogenous Leukemia
|
midostaurin
quizartinib
C3
FLT3 D835
|
Acute Myelogenous Leukemia
|
quizartinib
sorafenib
C3
FLT3 D835
|
Acute Myelogenous Leukemia
|
sorafenib
sunitinib
C3
FLT3 D835
|
Chronic Myeloid Leukemia
|
sunitinib
LAM 003
D
FLT3 D835
|
Acute Myelogenous Leukemia
|
LAM 003
MLN518
D
FLT3 D835
|
Acute Myelogenous Leukemia
|
MLN518
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