Group by Gene: Include preclinical: Tyrosine Kinase Inhibitors Serine-Threonine Kinase Inhibitors EGFR CD Protein Inhibitors Immune Checkpoint Inhibitors Immunotherapy Epigenetics | EGFR inhibitor erlotinib | PD1 inhibitor pembrolizumab | nivolumab | mTOR inhibitor everolimus | EZH2 inhibitor tazemetostat | pan-RAF inhibitor, Multi-tyrosine kinase inhibitor sorafenib | HER2 inhibitor, EGFR inhibitor lapatinib | VEGFR inhibitor, PDGFR inhibitor, c-KIT inhibitor sunitinib | Bcr-abl tyrosine kinase inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist dasatinib | PDGFR inhibitor, Bcr-abl tyrosine kinase inhibitor, c-KIT inhibitor imatinib | HER2 inhibitor, HER4 inhibitor, EGFR inhibitor afatinib | PDGFR inhibitor PDGFR inhibitor | PDGFR inhibitor, HDAC inhibitor PDGFR inhibitor + HDAC inhibitor |
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No biomarker | |||||||||||||
EGFR expression | |||||||||||||
SMARCB1 negative | |||||||||||||
PIK3CA amplification | |||||||||||||
PIK3CA M1043I | |||||||||||||
SMARCB1 deletion | |||||||||||||
TMB-H | |||||||||||||
MSI-H/dMMR | |||||||||||||
AXL underexpression | |||||||||||||
PTEN deletion | |||||||||||||
STK33 underexpression | |||||||||||||
PBRM1 mutation |