^
CANCER:

Breast Cancer





Show legend
Group by Gene:
Include preclinical:

HER2 inhibitor
trastuzumab
margetuximab
tucatinib
LZM-005
Zercepac (trastuzumab biosimilar)
trastuzumab + LZM-005
trastuzumab-dttb
trastuzumab-dkst
trastuzumab-anns
trastuzumab + tucatinib
trastuzumab-qyyp
trastuzumab-pkrb
TX05 (trastuzumab biosimilar)
Hervelous (trastuzumab biosimilar)
0
HER2 inhibitor
ZW25
KN026
DF1001
EG12014 (trastuzumab biosimilar)
trastuzumab / hyaluronidase-oysk
HERtiCAD (trastuzumab biosimilar)
ZN-A-1041
DZD1516
inetetamab
MP0274
Hercease (trastuzumab biosimilar)
VRN101099
AB-201
trastuzumab
trastuzumab-IFN-β mutein
CDK4 inhibitor + CDK6 inhibitor
ribociclib
abemaciclib
palbociclib
trilaciclib
XZP 3287
dalpiciclib
1
CDK4 inhibitor, CDK6 inhibitor
G1T38
palbociclib + ribociclib
TQB3616
FCN-437
BPI-16350
palbociclib + abemaciclib
PRT3645
CS3002
PARP inhibitor
olaparib
talazoparib
niraparib
2
PARP inhibitor
ABT-888
pamiparib
fluzoparib
IMP4297
NOV 1401
rucaparib
alpelisib
GDC-0032
CYH33
3
PIK3CA inhibitor
GDC-0077
alpelisib + GDC-0032
HS-10352
LX-086
RLY-2608
tamoxifen
4
Estrogen receptor antagonist
tamoxifen
tamoxifen
bevacizumab
Aybintio (bevacizumab biosimilar)
Krabeva (bevacizumab biosimilar)
5
VEGF-A inhibitor
bevacizumab-maly
bevacizumab-adcd
bevacizumab-bvzr
bevacizumab-awwb
Selective estrogen receptor degrader
fulvestrant
elacestrant
SAR439859
AZD9833
G1T48
6
Selective estrogen receptor degrader
GDC-0927
D-0502
ZN-c5
SCR-6852
LY3484356
LX-039
AZD9496
SCR6106
Aromatase inhibitor
exemestane
7
Aromatase inhibitor
anastrozole
letrozole
Aromatase inhibitor
pegylated liposomal doxorubicin
doxorubicin hydrochloride
non-pegylated liposomal doxorubicin
8
Topoisomerase II inhibitor
epirubicin
pegylated liposomal doxorubicin
doxorubicin hydrochloride
etoposide IV
PD1 inhibitor
pembrolizumab
nivolumab
9
PD1 inhibitor
toripalimab-tpzi
tislelizumab
cemiplimab-rwlc
nivolumab + toripalimab-tpzi
dostarlimab-gxly
atezolizumab
10
PD-L1 inhibitor
durvalumab
avelumab
capecitabine
11
Thymidylate synthase inhibitor
gimeracil / oteracil / tegafur
tegafur / uracil
5-fluorouracil
gemcitabine
12
DNA synthesis inhibitor
cisplatin
nedaplatin
13
mTOR inhibitor
everolimus
AZD8055
14
Tubulin polymerization promoter
carboplatin
15
Tubulin polymerization inhibitor
vinorelbine tartrate
vincristine
trastuzumab + pertuzumab
pertuzumab + trastuzumab-pkrb
16
HER2 inhibitor, HER2 dimerization inhibitor
pertuzumab + trastuzumab-dttb
pertuzumab + Zercepac (trastuzumab biosimilar)
pertuzumab + inetetamab
pertuzumab / trastuzumab / hyaluronidase-zzxf
toremifene
17
Selective estrogen receptor modulator
lasofoxifene
afimoxifene
18
Bcl2 inhibitor, Tubulin inhibitor
albumin-bound paclitaxel
paclitaxel oral
capivasertib
19
AKT inhibitor
TAS-117
MK-2206
GSK690693
FGFR inhibitor
futibatinib
infigratinib
20
FGFR inhibitor
ABSK091
Debio 1347
ARQ 087
E7090
ixabepilone
21
Microtubule inhibitor
E7389-LF
cabazitaxel
22
RNA polymerase 1 inhibitor
CX-5461
trastuzumab + abemaciclib
trastuzumab + palbociclib
23
HER2 inhibitor, CDK4 inhibitor, CDK6 inhibitor
palbociclib + tucatinib
palbociclib + ZW25
tucatinib + PRT3645
abemaciclib + tucatinib
24
Bone resorption factor inhibitor, Osteoclast inhibitor
zoledronic acid
25
GnRH agonist
leuprolide acetate for depot suspension
triptorelin
26
Mitosis inhibitor
vinorelbine
27
Progesterone receptor agonist
megestrol
28
Tubulin polymerization promoter, Bcl2 inhibitor
paclitaxel
carboplatin + paclitaxel
29
PI3K inhibitor, AKT inhibitor
RG7440
anlotinib
pazopanib
ponatinib
30
Multi-tyrosine kinase inhibitor
TT-00420
vandetanib
cabozantinib capsule
midostaurin
31
PD-L1 inhibitor, PARP inhibitor
avelumab + talazoparib
olaparib + durvalumab
tamoxifen + fulvestrant
32
Estrogen receptor antagonist, Selective estrogen receptor degrader
GDC-9545
OP-1250
pembrolizumab + niraparib
33
PD1 inhibitor, PARP inhibitor
tislelizumab + pamiparib
pembrolizumab + olaparib
PI3K inhibitor
AN2025
34
PI3K inhibitor
GDC-0941
MEN1611
SB02024
35
PARG inhibitor
IDE161
CT7001
36
CDK7 inhibitor
SY-5609
Q901
YPN-005
37
TrkB receptor inhibitor, TrkC kinase inhibitor, TrkA receptor inhibitor
larotrectinib
38
mTORC1 inhibitor, mTORC2 inhibitor
CB-228
39
VEGFR-2 inhibitor, PARP inhibitor
rivoceranib + fluzoparib
40
Androgen receptor inhibitor
enzalutamide capsule
darolutamide
41
HER2 dimerization inhibitor
QL1209 (pertuzumab biosimilar)
pertuzumab
42
Selective estrogen receptor α inhibitor
H3B-6545
43
Bcl2 inhibitor
venetoclax
44
Ubiquitin pathway modulator, Estrogen receptor alpha degrader
ARV-471
45
RANK ligand inhibitor
denosumab
46
Immunostimulant, G-CSF stimulant
SV-BR-1-GM
47
VEGFR-2 inhibitor
rivoceranib
fulvestrant + anastrozole
48
Aromatase inhibitor, Selective estrogen receptor degrader
fulvestrant + letrozole
letrozole + SAR439859
49
HER2 inhibitor, mTOR inhibitor
trastuzumab + everolimus
sirolimus + inetetamab
50
HER2 inhibitor, HER4 inhibitor, pan-EGFR inhibitor
poziotinib
51
CXCR4 antagonist
POL 6326
52
FGFR inhibitor, VEGFR inhibitor, PDGFR inhibitor, pan-TRK inhibitor
TKI258
53
HER2-targeted antibody-drug conjugate, DNA replication inhibitor
trastuzumab duocarmazine
54
Aurora kinase A inhibitor
MLN8237
55
PI3Kγ inhibitor
IPI-549
CZC24832
56
IGF-1R inhibitor
AMG 479
ASP7487
57
Alkylating agent, DNA synthesis inhibitor
cisplatin + cyclophosphamide
cyclophosphamide + thiotepa
58
eIF4A1 inhibitor, CDK4 inhibitor, CDK6 inhibitor
abemaciclib + eFT226
palbociclib + CR-1-31-B
59
PIK3CA inhibitor, HER2 inhibitor, HER2 dimerization inhibitor
trastuzumab + pertuzumab + alpelisib
60
TTK inhibitor
CFI-402257
VRN08
61
Tubulin inhibitor, Thymidylate synthase inhibitor
capecitabine + DJ 927
62
Alkylating agent
D19466
cyclophosphamide
63
HER2 inhibitor, HER3 inhibitor
MCLA-128
trastuzumab + MCLA-128
crizotinib
64
ALK inhibitor
alectinib
ceritinib
cetuximab
gefitinib
65
EGFR inhibitor
Hemay022
WZ4002
erlotinib
CL-387785
CDK2 inhibitor
66
CDK2 inhibitor
PF-07104091
BLU-222
67
PD1 inhibitor, CTLA4 inhibitor
nivolumab + ipilimumab
68
IL-6R antagonist
tocilizumab
69
ATR inhibitor, PARP inhibitor
olaparib + AZD6738
ABT-888 + M6620
70
PD1 inhibitor, Multi-tyrosine kinase inhibitor
camrelizumab + SHR 1020
71
HER2-targeted antibody-drug conjugate, Tubulin inhibitor
A166
72
VEGF-A inhibitor, PD1 inhibitor
nivolumab + bevacizumab
73
Microtubule inhibitor, Notch3-targeted antibody-drug conjugate
PF-06650808
74
PD-L1 inhibitor, PARP inhibitor, AKT inhibitor
olaparib + durvalumab + capivasertib
75
Proteasome inhibitor
ixazomib
bortezomib
76
PARP inhibitor, AKT inhibitor
olaparib + capivasertib
77
DNA synthesis inhibitor, Bcl2 inhibitor, Tubulin inhibitor
cisplatin + albumin-bound paclitaxel
78
VEGF-A inhibitor, HER2 inhibitor
bevacizumab + trastuzumab
79
Tubulin polymerization promoter, Bcl2 inhibitor, Tubulin inhibitor
carboplatin + albumin-bound paclitaxel
80
RET inhibitor
pralsetinib
selpercatinib
romidepsin
panobinostat
81
HDAC inhibitor
SB939
vorinostat
MGCD0103
trastuzumab + lapatinib
82
HER2 inhibitor, EGFR inhibitor
lapatinib
trastuzumab + S-222611
mobocertinib
83
HER2 inhibitor, PD1 inhibitor
pembrolizumab + trastuzumab
camrelizumab + inetetamab
84
Progesterone receptor antagonist
onapristone XR
RAIN-32
85
MDM2 inhibitor
KRT-232 + APG-115
CGM097
86
Tubulin polymerization promoter, DNA synthesis inhibitor
carboplatin + gemcitabine
87
MEK inhibitor
trametinib
selumetinib
88
Microtubule inhibitor, LY6E-targeted antibody-drug conjugate
DLYE5953A
89
ATR inhibitor
BAY 1895344
M6620
90
PIK3CA inhibitor, PARP inhibitor
olaparib + alpelisib
91
PLK4 inhibitor
CFI-400945
92
AXL inhibitor, HER2 inhibitor
trastuzumab + TP-0903
cyclophosphamide + non-pegylated liposomal doxorubicin
93
Topoisomerase II inhibitor, Alkylating agent
doxorubicin hydrochloride + cyclophosphamide
cyclophosphamide + epirubicin
94
VEGFR inhibitor, PD-L1 inhibitor, PARP inhibitor
olaparib + durvalumab + cediranib
95
Tubulin polymerization promoter, Alkylating agent, Bcl2 inhibitor
carboplatin + paclitaxel + cyclophosphamide
96
pan-AKT inhibitor
LAE002
97
PD-L1 inhibitor, CTLA4 inhibitor
KN046
98
CEBPB antagonist
ST101
99
Androgen receptor agonist
CR 1477
100
Wnt signalling pathway inhibitor
OMP-18R5
101
HDAC inhibitor, HDAC1 inhibitor, HDAC2 inhibitor, HDAC3 inhibitor
entinostat
102
WEE1 inhibitor
AZD1775
ZN-c3
103
Selective estrogen receptor degrader, AKT inhibitor
capivasertib + AZD9833
104
Topoisomerase I inhibitor
DAN-222
105
PD1 inhibitor, MEK inhibitor
pembrolizumab + binimetinib
106
HDAC6 inhibitor
ACY-1215
107
VEGFR-2 inhibitor, HER2 inhibitor
trastuzumab + rivoceranib
108
Tubulin polymerization inhibitor, Thymidylate synthase inhibitor
capecitabine + vinorelbine tartrate
109
Topoisomerase II inhibitor, DNA inhibitor
etoposide oral
110
KAT6 inhibitor
PF-07248144
ISM5043
111
Apoptosis stimulant
pelareorep
112
Estrogen receptor antagonist, mTOR inhibitor
everolimus + tamoxifen
113
PARP7 inhibitor
RBN-2397
114
THF dehydrogenase inhibitor, Dihydrofolic acid reductase inhibitor
methotrexate
115
Androgen receptor inhibitor, Selective estrogen receptor degrader
enzalutamide capsule + fulvestrant
116
Estrogen receptor antagonist, mTORC1 inhibitor, mTORC2 inhibitor
tamoxifen + CB-228
117
ERN1 inhibitor
ORIN1001
118
Androgen receptor antagonist, TMPRSS2 inhibitor
GT0918
119
MEK inhibitor, BRAF inhibitor
trametinib + dabrafenib
120
CDK4 inhibitor, CDK6 inhibitor, Multi-tyrosine kinase inhibitor
dalpiciclib + SHR 1020
121
PD-L1 inhibitor, VEGF-A inhibitor
BNT327
bevacizumab + atezolizumab
122
Notch inhibitor
RG4733
CB-103
123
DNA methylation inhibitor
azacitidine
TdCyd
124
VEGF-A inhibitor, mTOR inhibitor
bevacizumab + temsirolimus
125
PD1 inhibitor, CDK inhibitor
pembrolizumab + MK-7965
126
Alkylating agent, Thymidylate synthase inhibitor
capecitabine + D19466
127
APC activator
eftilagimod alpha
128
BRAF inhibitor, BRAF V600E inhibitor
vemurafenib
129
Selective androgen receptor modulator
EP0062
130
BET inhibitor, PARP inhibitor
talazoparib + ZEN-3694
131
Thymidine phosphorylase inhibitor
trifluridine / tipiracil
132
AKT inhibitor, p70S6K inhibitor
LY2780301
CCT128930
133
Tubulin inhibitor
DJ 927
134
CCR5 receptor antagonist, Viral entry inhibitor
leronlimab
135
CDK4 inhibitor
PF-07220060
136
FASN inhibitor
TVB-2640
137
PIK3CA inhibitor, HER2 inhibitor, HER3 inhibitor
trastuzumab + alpelisib + LJM-716
138
PVRIG inhibitor, PD1 inhibitor
nivolumab + COM701
139
PIK3CA inhibitor, Selective estrogen receptor degrader
alpelisib + LY3484356
140
mTOR inhibitor, Selective estrogen receptor degrader
everolimus + LY3484356
141
PIK3CA inhibitor, HER2 inhibitor
trastuzumab + alpelisib
142
DNA replication inhibitor, AXL-targeted antibody-drug conjugate
ADCT-601
143
Selective estrogen receptor covalent antagonist
HRS8807
144
Microtubule inhibitor, CD166-targeted antibody-drug conjugate
CX-2009
145
Topoisomerase II inhibitor, HER2-targeted antibody-drug conjugate
MM-302
146
IAP inhibitor
APG-1387
IGM-9427
FEC
TAC
Nab-PHP + PldCHP
EC-TH
CaT
THP
TC
TCHP
ECP-THP
CMF
TEC
CAF
TCbHP
VEX
147
Chemotherapy
PH-FECH
PCbTP
VIP
AC-THP
EC-P
TH
GC
EC
AC
GT
ACT
GemCarbo
FAC
AC-TH
TCH
148
FAK inhibitor
FAK inhibitor
VS-4718
149
HER2-targeted CAR-T immunotherapy
HER2-targeted CAR-T immunotherapy
150
Immunotherapy
Immunotherapy
151
MUC1 inhibitor
MUC1 inhibitor
152
HDAC inhibitor, AKT1 inhibitor
HDAC inhibitor + AKT1 inhibitor
153
HDAC inhibitor, AKT2 inhibitor
HDAC inhibitor + AKT2 inhibitor
154
CDK19 inhibitor
CDK19 inhibitor
155
CDK8 inhibitor
CDK8 inhibitor
156
EGFR-targeted antibody-drug conjugate
EGFR-targeted antibody-drug conjugate
157
Tyrosine kinase inhibitor
Tyrosine kinase inhibitor
PD173074
158
Immunotherapy, PARP inhibitor
Immunotherapy + PARP inhibitor
159
B7-H3-targeted antibody-drug conjugate
B7-H3-targeted antibody-drug conjugate
160
PI3K inhibitor, mTOR inhibitor, AKT inhibitor
mTOR inhibitor + PI3K inhibitor + AKT inhibitor
DFN-529
161
Aurora kinase inhibitor, WEE1 inhibitor
WEE1 inhibitor + Aurora kinase inhibitor
162
PD-L1 inhibitor, MYC inhibitor
PD-L1 inhibitor + MYC inhibitor
163
HER2 inhibitor, Erythropoiesis stimulating agent
HER2 inhibitor + Erythropoiesis stimulating agent
164
Aromatase inhibitor, HER2 inhibitor
HER2 inhibitor + Aromatase inhibitor
165
mTORC1 inhibitor
mTORC1 inhibitor
166
EZH2 inhibitor, PARP inhibitor
PARP inhibitor + EZH2 inhibitor
167
CDK4 inhibitor, EGFR inhibitor, CDK6 inhibitor
EGFR inhibitor + CDK4 inhibitor + CDK6 inhibitor
erlotinib + palbociclib
CDK4 inhibitor + CDK6 inhibitor + Aromatase inhibitor
168
Aromatase inhibitor, CDK4 inhibitor, CDK6 inhibitor
Aromatase inhibitor + palbociclib
letrozole + dalpiciclib
CDK4 inhibitor + CDK6 inhibitor + fulvestrant
169
CDK4 inhibitor, CDK6 inhibitor, Selective estrogen receptor degrader
palbociclib + SAR439859
abemaciclib + AZD9833
abemaciclib + LY3484356
170
PI3K inhibitor, Selective estrogen receptor degrader
PI3K inhibitor + fulvestrant
MEN1611 + elacestrant
171
Immunotherapy, Selective estrogen receptor degrader
Immunotherapy + fulvestrant
172
β-catenin inhibitor, CBP inhibitor, Microtubule inhibitor
eribulin mesylate
173
β-catenin inhibitor, CBP inhibitor, Microtubule inhibitor, Chemotherapy
HP + eribulin mesylate
174
Aromatase inhibitor, Thymidylate synthase inhibitor
Aromatase inhibitor + capecitabine
175
Aromatase inhibitor, HER2 inhibitor, EGFR inhibitor
Aromatase inhibitor + trastuzumab + lapatinib
176
Tyrosine kinase inhibitor, Thymidylate synthase inhibitor
Tyrosine kinase inhibitor + capecitabine
177
Aromatase inhibitor, HDAC inhibitor
HDAC inhibitor + exemestane
178
Aromatase inhibitor, mTOR inhibitor
exemestane + mTOR inhibitor
everolimus + exemestane
ado-trastuzumab emtansine
disitamab vedotin
DP303c
JNJ-0683
MRG002
TAA013
ZW49
179
HER2-targeted antibody-drug conjugate, Microtubule inhibitor
XMT-1522
IKS014
PF-06804103
MEDI4276
ALT-P7
BAT8001
BB-1701
MF-TTZ-MMAE
carboplatin + docetaxel
180
Microtubule stabilizer, Tubulin polymerization promoter
docetaxel
docetaxel
fam-trastuzumab deruxtecan-nxki
SHR-A1811
181
HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
BL-M07D1
BNT323
PRO1102
DAN-311
neratinib
pyrotinib
trastuzumab + neratinib
182
HER2 inhibitor, HER4 inhibitor, EGFR inhibitor
afatinib
trastuzumab + pyrotinib
pyrotinib + inetetamab
ASLAN001
lapatinib + neratinib
sacituzumab govitecan-hziy
MK-2870
183
TROP-2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
DS-1062a
ESG401
BL-M02D1
BAT8008
184
Microtubule stabilizer, Tubulin polymerization promoter, Thymidylate synthase inhibitor
docetaxel + capecitabine
185
Topoisomerase II inhibitor, Microtubule stabilizer, Tubulin polymerization promoter
docetaxel + doxorubicin hydrochloride
docetaxel + epirubicin
186
Topoisomerase II inhibitor, Microtubule stabilizer, Tubulin polymerization promoter, Alkylating agent
docetaxel + doxorubicin hydrochloride + cyclophosphamide
187
HER2-targeted antibody-drug conjugate, Microtubule inhibitor, HER2 dimerization inhibitor
pertuzumab + ado-trastuzumab emtansine
188
HER3-targeted antibody-drug conjugate, Topoisomerase I inhibitor
U3-1402
DB-1310
189
CDK4 inhibitor, PI3K inhibitor, mTOR inhibitor, mTORC1 inhibitor, CDK6 inhibitor, mTORC2 inhibitor
palbociclib + PF-05212384
190
HER2 inhibitor, PI3K inhibitor, mTOR inhibitor, mTORC1 inhibitor, mTORC2 inhibitor
PF-05212384 + trastuzumab-pkrb
191
Microtubule stabilizer, Tubulin polymerization promoter, DNA synthesis inhibitor
gemcitabine + docetaxel
192
Androgen receptor modulator, Selective androgen receptor modulator
enobosarm
193
FGFR inhibitor, CDK4 inhibitor, CDK6 inhibitor
palbociclib + BAY 1163877
palbociclib + ABSK091
194
FGFR inhibitor, VEGFR inhibitor, RET inhibitor, c-KIT inhibitor, PDGFR α antagonist
lenvatinib
195
VEGFR inhibitor, PDGFR inhibitor, c-KIT inhibitor
sunitinib
palbociclib + GDC-0032
palbociclib + GDC-0077
palbociclib + alpelisib
196
PIK3CA inhibitor, CDK4 inhibitor, CDK6 inhibitor
alpelisib + ribociclib
alpelisib + abemaciclib
abemaciclib + RLY-2608
palbociclib + RLY-2608
197
Topoisomerase II inhibitor, Tubulin polymerization promoter, Alkylating agent, Bcl2 inhibitor
paclitaxel + cyclophosphamide + epirubicin
198
TNKS inhibitor, PARP inhibitor
JPI-547
199
PD-L1 inhibitor, Multi-tyrosine kinase inhibitor
anlotinib + APL-502
200
TrkB receptor inhibitor, TrkC kinase inhibitor, ROS1 inhibitor, TrkA receptor inhibitor, ALK inhibitor, JAK2 inhibitor, TNK2 inhibitor
entrectinib
pyrotinib + dalpiciclib
201
HER2 inhibitor, HER4 inhibitor, CDK4 inhibitor, EGFR inhibitor, CDK6 inhibitor
trastuzumab + palbociclib + pyrotinib
palbociclib + neratinib
202
FGFR inhibitor, VEGFR inhibitor, PDGFR α-β inhibitor, Tyrosine kinase inhibitor
E 3810
203
PI3K inhibitor, mTOR inhibitor, mTORC1 inhibitor, mTORC2 inhibitor
PF-05212384
204
B7-H4-targeted antibody-drug conjugate, Tubulin inhibitor
XMT-1660
205
P-glycoprotein inhibitor, Bcl2 inhibitor, Tubulin inhibitor
oral paclitaxel / encequidar
206
AKT3 inhibitor, AKT1 inhibitor, AKT inhibitor, p70S6K inhibitor
DIACC3010
207
Topoisomerase II inhibitor, Alkylating agent, Bcl2 inhibitor, Tubulin inhibitor
albumin-bound paclitaxel + cyclophosphamide + epirubicin
208
PI3K inhibitor, mTOR inhibitor, mTORC1 inhibitor, PARP inhibitor, mTORC2 inhibitor
talazoparib + PF-05212384
209
Selective estrogen receptor modulator, Estrogen receptor antagonist
Z-endoxifen hydrochloride
210
FGFR2 inhibitor, FGFR inhibitor, FGFR1 inhibitor, FGFR3 inhibitor, CDK4 inhibitor, FGFR4 inhibitor, CDK6 inhibitor
palbociclib + erdafitinib
211
Topoisomerase II inhibitor, Tubulin polymerization inhibitor
epirubicin + vinorelbine tartrate
212
HER2 inhibitor, HER4 inhibitor, HER2-targeted antibody-drug conjugate, EGFR inhibitor, Microtubule inhibitor
neratinib + ado-trastuzumab emtansine
ado-trastuzumab emtansine + pyrotinib
213
PD-L1 inhibitor, PI3K inhibitor, AKT inhibitor
atezolizumab + RG7440
214
RNA polymerase inhibitor, Alkylating agent, Apoptosis stimulant
lurbinectedin
215
Estrogen receptor antagonist, HER2 inhibitor, Selective estrogen receptor degrader
HER2 inhibitor + OP-1250
216
Aromatase inhibitor, HER2 inhibitor, HER4 inhibitor, EGFR inhibitor
pyrotinib + letrozole
217
PD1 inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor
pembrolizumab + ado-trastuzumab emtansine
disitamab vedotin + zimberelimab
218
DNA synthesis inhibitor, PARP inhibitor
temozolomide + ABT-888
219
PD1 inhibitor, HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
nivolumab + fam-trastuzumab deruxtecan-nxki
220
TSP1 stimulant, CD36 stimulant
VT1021
221
Ubiquitin pathway modulator, CDK4 inhibitor, CDK6 inhibitor, Estrogen receptor alpha degrader
palbociclib + ARV-471
222
Estrogen receptor antagonist, CDK4 inhibitor, CDK6 inhibitor, Selective estrogen receptor degrader
palbociclib + OP-1250
223
PARP inhibitor, Topoisomerase I inhibitor
niraparib + DAN-222
224
β-catenin inhibitor, DNA synthesis inhibitor, CBP inhibitor, Microtubule inhibitor
gemcitabine + eribulin mesylate
225
Microtubule stabilizer, Tubulin polymerization promoter, Alkylating agent
docetaxel + cyclophosphamide
226
DDR enhancer, PARP inhibitor, Topoisomerase I inhibitor
rucaparib + PLX038
227
PD-L1 inhibitor, HER2 inhibitor, HER2 dimerization inhibitor
trastuzumab + atezolizumab + pertuzumab
228
Protein synthesis inhibitor, HER2 inhibitor
MT-5111
229
Topoisomerase II inhibitor, HER2 inhibitor, HER2-targeted antibody-drug conjugate
trastuzumab + MM-302
230
PD-L1 inhibitor, Immunostimulant
atezolizumab + RG6180
231
Lyase inhibitor, Androgen receptor antagonist
TAK 700
paclitaxel + epirubicin
232
Topoisomerase II inhibitor, Tubulin polymerization promoter, Bcl2 inhibitor
carboplatin + paclitaxel + doxorubicin hydrochloride
carboplatin + paclitaxel + non-pegylated liposomal doxorubicin
paclitaxel + doxorubicin hydrochloride
233
CDK4 inhibitor, PI3K inhibitor, CDK6 inhibitor
ribociclib + AN2025
234
HER2 inhibitor, JAK1 inhibitor, JAK2 inhibitor
trastuzumab + ruxolitinib
235
HER2 inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor
ado-trastuzumab emtansine + tucatinib
tucatinib + disitamab vedotin
236
Chk1 inhibitor, Chk2 inhibitor
ACR-368
AZD-7762
237
HDAC inhibitor, MAPK inhibitor, HDAC10 inhibitor, HDAC1 inhibitor, PI3K inhibitor, HDAC2 inhibitor, AKT inhibitor, HDAC3 inhibitor
chidamide
238
VEGF-A inhibitor, Mitochondrial OXHPHOS inhibitor, mTOR inhibitor
bevacizumab + ME-344
239
β-catenin inhibitor, Tubulin polymerization promoter, CBP inhibitor, Microtubule inhibitor
carboplatin + eribulin mesylate
palbociclib + everolimus
240
CDK4 inhibitor, mTOR inhibitor, CDK6 inhibitor
everolimus + ribociclib
everolimus + abemaciclib
241
AKT3 inhibitor, HER2 inhibitor, AKT1 inhibitor, AKT inhibitor, p70S6K inhibitor
trastuzumab + DIACC3010
242
HER2 inhibitor, CTLA4 inhibitor
trastuzumab + tremelimumab
243
JAK1 inhibitor, JAK2 inhibitor
ruxolitinib
244
DNA replication inhibitor, Thymidylate synthase inhibitor
capecitabine + bendamustine
245
PD-L1 inhibitor, HER2 inhibitor, CTLA4 inhibitor
KN046 + KN026
246
PIK3CA inhibitor, Estrogen receptor antagonist
tamoxifen + GDC-0032
PF-06873600
247
CDK2 inhibitor, CDK4 inhibitor, CDK6 inhibitor
palbociclib + BLU-222
RGT-419B
ribociclib + BLU-222
248
Androgen receptor antagonist, Selective estrogen receptor degrader, TMPRSS2 inhibitor
fulvestrant + GT0918
249
BRAF inhibitor, MEK1 inhibitor, BRAF V600E inhibitor
vemurafenib + cobimetinib
250
Topoisomerase II inhibitor, Alkylating agent, G-CSF stimulant, Bcl2 inhibitor, Tubulin inhibitor
albumin-bound paclitaxel + cyclophosphamide + epirubicin + pegfilgrastim
251
Estrogen receptor antagonist, GnRH agonist
tamoxifen + goserelin acetate
252
MDMX inhibitor, MDM2 inhibitor
ALRN-6924
253
HER2 inhibitor, PD1 inhibitor, HER2 dimerization inhibitor
pembrolizumab + pertuzumab + trastuzumab-qyyp
254
CDK4 inhibitor, Selective estrogen receptor α inhibitor, CDK6 inhibitor
palbociclib + H3B-6545
255
HER2 inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor, HER2 dimerization inhibitor
trastuzumab + pertuzumab + ado-trastuzumab emtansine
256
HER2-targeted antibody-drug conjugate, Microtubule inhibitor, Topoisomerase I inhibitor
ado-trastuzumab emtansine + fam-trastuzumab deruxtecan-nxki
257
PD-L1 inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor
atezolizumab + ado-trastuzumab emtansine
258
HER2 inhibitor, PD1 inhibitor, LAG-3 inhibitor
margetuximab + MGD013
259
PD1 inhibitor, GM-CSF agonist, CTLA4 inhibitor
nivolumab + ipilimumab + talimogene laherparepvec
260
PD-L1 inhibitor, PD1 inhibitor
pembrolizumab + durvalumab
261
GPNMB-targeted antibody-drug conjugate, Microtubule inhibitor
CDX-011
262
PD-L1 inhibitor, HER2 inhibitor
trastuzumab + atezolizumab
trastuzumab + durvalumab
263
CD137 agonist, HER2 inhibitor
PRS-343
264
TLR9 agonist, PD1 inhibitor
pembrolizumab + SD-101
265
β-catenin inhibitor, CBP inhibitor, PD1 inhibitor, Microtubule inhibitor
pembrolizumab + eribulin mesylate
266
PI3K inhibitor, JAK2 inhibitor
GDC-0941 + AZ 960
267
IGF-2 inhibitor, CDK4 inhibitor, IGF1 inhibitor, CDK6 inhibitor
abemaciclib + BI-836845
268
HER2 inhibitor, PI3K inhibitor
trastuzumab + MEN1611
trastuzumab + SAR245408
269
THF dehydrogenase inhibitor, Alkylating agent, Dihydrofolic acid reductase inhibitor, Thymidylate synthase inhibitor
capecitabine + cyclophosphamide + methotrexate
270
HER2 inhibitor, HER2-targeted antibody-drug conjugate, EGFR inhibitor, Microtubule inhibitor
lapatinib + ado-trastuzumab emtansine
271
IGF-2 inhibitor, mTOR inhibitor, IGF1 inhibitor
everolimus + BI-836845
272
β-catenin inhibitor, CBP inhibitor, Microtubule inhibitor, Thymidylate synthase inhibitor
capecitabine + eribulin mesylate
273
Tubulin polymerization promoter, Apoptosis stimulant, Bcl2 inhibitor
paclitaxel + pelareorep
274
DNA synthesis inhibitor, DNA cross linking agent, Apoptosis inhibitor, Microtubule inhibitor
INT230-6
275
Bcr-abl tyrosine kinase inhibitor, CDK4 inhibitor, Src kinase inhibitor, CDK6 inhibitor
palbociclib + bosutinib
276
HER2 inhibitor, CD20 inhibitor
trastuzumab + TQB2303 (rituximab biosimilar)
277
PD-L1 inhibitor, HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
durvalumab + fam-trastuzumab deruxtecan-nxki
278
Aromatase inhibitor, mTOR inhibitor, GnRH agonist
everolimus + letrozole + leuprolide acetate
279
PD-L1 inhibitor, GM-CSF agonist
atezolizumab + talimogene laherparepvec
280
CDK4 inhibitor, PD1 inhibitor, CDK6 inhibitor
pembrolizumab + palbociclib
pembrolizumab + abemaciclib
281
PIK3CA inhibitor, HER2 inhibitor, PI3Kδ inhibitor
trastuzumab + copanlisib
282
Microtubule stabilizer, Tubulin polymerization promoter, Sortilin inhibitor
TH 1902
283
CDK4 inhibitor, HER2-targeted antibody-drug conjugate, CDK6 inhibitor, Microtubule inhibitor
palbociclib + ado-trastuzumab emtansine
284
VEGF-A inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor
bevacizumab + disitamab vedotin
285
HER2-targeted antibody-drug conjugate, TROP-2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
fam-trastuzumab deruxtecan-nxki + sacituzumab govitecan-hziy
286
PIK3CA inhibitor, CDK4 inhibitor, CDK6 inhibitor, PI3Kδ inhibitor
abemaciclib + copanlisib
287
CDK4 inhibitor, PI3K inhibitor, CDK6 inhibitor, AKT inhibitor
palbociclib + RG7440
288
PIK3CA inhibitor, Estrogen receptor antagonist, Selective estrogen receptor degrader
GDC-9545 + GDC-0077
289
HER2 inhibitor, CDK4 inhibitor, CDK6 inhibitor, HER2 dimerization inhibitor
trastuzumab + palbociclib + pertuzumab
290
SIK3 inhibitor, PI3K inhibitor, PI3Kγ inhibitor, PI3Kδ inhibitor
RP6530
291
EGFR inhibitor, MUC1 inhibitor
gatipotuzumab + tomuzotuximab
292
PD-L1 inhibitor, CDK4 inhibitor, CDK6 inhibitor
atezolizumab + abemaciclib
293
PTK7-targeted antibody-drug conjugate, TROP-2-targeted antibody-drug conjugate
BCG033
294
HER2 inhibitor, CDK4 inhibitor, EGFR inhibitor, CDK6 inhibitor
palbociclib + lapatinib
295
CDK4 inhibitor, CDK6 inhibitor, PARP inhibitor
talazoparib + abemaciclib
olaparib + palbociclib
296
p53 reactivator
APR-246
297
PIK3CA inhibitor, HER2 inhibitor, HER4 inhibitor, EGFR inhibitor
alpelisib + pyrotinib
298
HER2 inhibitor, α radiation emission
BAY2701439
299
PI3K inhibitor, mTOR inhibitor
GDC-0980
RTB101
300
PD1 inhibitor, PI3Kδ inhibitor
camrelizumab + linperlisib
301
HER2-targeted antibody-drug conjugate, NMT inhibitor
MYX2449
302
Microtubule inhibitor, EGFR-targeted antibody-drug conjugate
LR004-VC-MMAE
HTI-1511
303
MUC1-targeted antibody-drug conjugate, Microtubule inhibitor
3D1-MMAE
304
MERTK-targeted antibody-drug conjugate, Microtubule inhibitor
RGX-019-MMAE
305
Microtubule inhibitor, LIV-1-targeted antibody-drug conjugate
BRY812
SGN-LIV1A
306
Melanotransferrin modulator, HER2-targeted antibody-drug conjugate
BT2111
307
Nectin-4-targeted antibody-drug conjugate, Microtubule inhibitor
9MW2821
308
Microtubule inhibitor, TROP-2-targeted antibody-drug conjugate
LCB84
BAT8003
309
IGF-1R-targeted antibody-drug conjugate, Microtubule inhibitor
W0101
310
HER2-targeted antibody-drug conjugate, HER3-targeted antibody-drug conjugate, GSPT1 degrader
ORM-5029
311
Prolactin receptor-targeted antibody-drug conjugate, DNA cross linking agent
ABBV-176
312
LAMP1-targeted antibody-drug conjugate, Microtubule inhibitor
SAR428926
313
Globo H-targeted antibody-drug conjugate, Microtubule inhibitor
OBI-999
314
DNA replication inhibitor, ROR1-targeted antibody-drug conjugate
NBE-002
315
5T4-targeted antibody-drug conjugate, Microtubule inhibitor
ASN004
316
PARP inhibitor, WEE1 inhibitor
olaparib + AZD1775
niraparib + AZD1775
317
B7-H3-targeted antibody-drug conjugate, DNA replication inhibitor
ITC-6102RO
MGC018
STX-478
318
PI3Kα H1047R mutation inhibitor
OKI-219
LOXO-783
319
MNK1 degrader, MNK2 degrader
VNLG-152R
320
HER2 inhibitor, HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
fam-trastuzumab deruxtecan-nxki + tucatinib
321
CDK4 inhibitor, CDK6 inhibitor, CDK9 inhibitor
palbociclib + AZD4573
322
ATM kinase inhibitor
AZD1390
323
SIRPA inhibitor, STAT3 inhibitor, HER2-targeted antibody-drug conjugate, TNF inhibitor, Topoisomerase I inhibitor
fam-trastuzumab deruxtecan-nxki + INB03
324
XPO1 inhibitor, Nuclear export inhibitor
KPT-8602
325
PLK1 inhibitor
PCM-075
326
CDK6 degrader, CDK4 degrader
BTX-9341
327
CDK19 inhibitor, CDK8 inhibitor
RVU120
328
PLK1 inhibitor, PIK3CA inhibitor
alpelisib + PCM-075
329
PI3Kα H1047R mutation inhibitor, CDK4 inhibitor, CDK6 inhibitor
palbociclib + STX-478
330
PI3Kα H1047R mutation inhibitor, Selective estrogen receptor degrader
AZD9833 + OKI-219
elacestrant + OKI-219
331
HER2 inhibitor, PI3Kα H1047R mutation inhibitor
tucatinib + OKI-219
332
IDO inhibitor
NLG8189
333
Angiopoietin 1 inhibitor, TIE-2 antagonist, Angiopoietin 2 inhibitor
AMG 386
334
BET inhibitor
JQ-1
ZEN-3694
335
Ribonucleotide reductase inhibitor
NSC-324360
336
NEDD8 activating enzyme inhibitor
MLN4924
337
HER2-targeted antibody-drug conjugate, DNA replication inhibitor, PARP inhibitor
olaparib + niraparib + trastuzumab duocarmazine
338
Microtubule inhibitor, CD228-targeted antibody-drug conjugate
SGN-CD228A
339
pan-CLK inhibitor, DYRK inhib
SM08502
340
Androgen receptor antagonist
apalutamide
HC-1119
341
CBP inhibitor, EP300 inhibitor
FT-6876
342
CDK4 inhibitor, CDK6 inhibitor, PDK1 inhibitor
palbociclib + VRx-510
ribociclib + VRx-510
343
CDK4 inhibitor, CDK6 inhibitor, MDM2 inhibitor
palbociclib + CGM097
344
Bcr-abl tyrosine kinase inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib
345
Bcr-abl tyrosine kinase inhibitor, HER2 inhibitor, EGFR inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib + lapatinib
346
HER2 inhibitor, HER4 inhibitor, HER2-targeted antibody-drug conjugate, EGFR inhibitor, Topoisomerase I inhibitor
neratinib + fam-trastuzumab deruxtecan-nxki
347
DRD1 partial agonist
levo-tetrahydropalmatine
348
Ferroptosis inducer
erastin
349
NRF2 inhibitor
brusatol
trastuzumab + GS-4721
350
HER2 inhibitor, CD47 inhibitor
IMM2902
D3L-001
351
Microtubule inhibitor, Bcl2 inhibitor, Bcl-xL inhibitor, Bcl-w inhibitor, EGFR-targeted antibody-drug conjugate
ABT 263 + ABT-414
352
DNA replication inhibitor, Bcl2 inhibitor, Bcl-xL inhibitor, Bcl-w inhibitor, EGFR-targeted antibody-drug conjugate
ABT 263 + ABBV-321
353
Aurora kinase inhibitor
ENMD-2076
354
HER2 inhibitor, EGFR inhibitor, Multi-tyrosine kinase inhibitor
AEE788
355
PI3Kβ inhibitor
AZD8186
356
mTOR inhibitor, EGFR inhibitor
gefitinib + everolimus
357
VEGFR inhibitor, PDGFR inhibitor, ALK inhibitor, c-KIT inhibitor
crizotinib + sunitinib
358
mTOR inhibitor, mTORC1 inhibitor
RapaLink-1
359
γ-secretase inhibitor
nirogacestat
360
mTOR inhibitor, mTORC2 inhibitor
PP242
361
pan-AKT inhibitor, CDK4 inhibitor, CDK6 inhibitor
palbociclib + ARQ 751
362
JNK inhibitor
JNK-IN-8
363
LIF inhibitor
EC359
364
TrxR inhibitor, AKT inhibitor
MK-2206 + D9
365
HER2 inhibitor, HER4 inhibitor, mTOR inhibitor, EGFR inhibitor
everolimus + neratinib
366
HER2 inhibitor, HER4 inhibitor, MEK inhibitor, EGFR inhibitor
trametinib + neratinib
367
pan-RAF inhibitor, Apoptosis inducer, PP2A activator, Multi-tyrosine kinase inhibitor
sorafenib + nanoliposomal ceramide
368
MERTK-targeted antibody-drug conjugate
RGX-019
369
SF3B1 inhibitor, RNA splicing modulator
SSA
370
ER-α 36 modulator
SNG-162
371
eIF4A1 inhibitor
eFT226
372
BET inhibitor, CDK4 inhibitor, CDK6 inhibitor
palbociclib + ZEN-3694
abemaciclib + ZEN-3694
373
CDK4 inhibitor, CDK6 inhibitor, Bcl2 inhibitor
palbociclib + APG-2575
374
p53 stimulant
COTI-2
375
PP2A inhibitor
LB-100
376
PD-L1 inhibitor, CD73 inhibitor
durvalumab + MEDI9447
377
ERK2 inhibitor, PI3K inhibitor, ERK inhibitor, ERK1 inhibitor, GnRH agonist
triptorelin + AEZS 136 + AEZS-134
378
PI3K inhibitor, ERK inhibitor, GnRH agonist
triptorelin + AEZS-129
379
GnRH agonist, AKT inhibitor
triptorelin + D21266
380
NQO1 inhibitor
ARQ 761
381
THF dehydrogenase inhibitor, Thymidylate synthase inhibitor
pemetrexed
382
Haspin inhibitor
CHR-6494
383
β-catenin inhibitor, Tubulin polymerization promoter, CBP inhibitor, Microtubule inhibitor, Bcl2 inhibitor
paclitaxel + eribulin mesylate
384
Chk1 inhibitor, WEE1 inhibitor
AZD1775 + SRA737
385
PIK3CA inhibitor, CDK4 inhibitor, mTOR inhibitor, CDK6 inhibitor, Selective estrogen receptor degrader
everolimus + alpelisib + abemaciclib + LY3484356
386
HER2 inhibitor, HER4 inhibitor, EGFR inhibitor, PARP inhibitor
neratinib + niraparib
olaparib + neratinib
387
PARP1 inhibitor
AZD5305
388
T-cell stimulant, HER2 inhibitor, CD3 agonist, CD28 agonist
SAR443216
389
ADAM9-targeted antibody-drug conjugate, Microtubule inhibitor
IMGC936
390
EGFR inhibitor, CD16A agonist
AFM24
391
Annexin A1 inhibitor
MDX-124
392
PARP2 inhibitor, PARP1 inhibitor
TQB3823
393
pan-RAF inhibitor, Multi-tyrosine kinase inhibitor
sorafenib
394
AMPK activator
metformin
395
HER3 inhibitor
MM-121
396
β-catenin inhibitor, CBP inhibitor, Wnt signalling pathway inhibitor
PRI724
397
XPO1 inhibitor
selinexor
398
TGF-β RI kinase inhibitor, TGF-β R2 kinase inhibitor
LY2109761
399
DNA synthesis inhibitor, DNA cross linking agent
oxaliplatin
400
ERK2 inhibitor
VTX-11e
401
CDK2 inhibitor, CDK9 inhibitor
CYC065
402
CDK2 inhibitor, CDK9 inhibitor, PARP inhibitor
olaparib + CYC065
403
MCL1 inhibitor, Bcl-xL inhibitor
S63845 + A-1331852
404
PI3K inhibitor, Bcl-xL inhibitor, AKT inhibitor
RG7440 + A-1331852
405
Topoisomerase II inhibitor, Selective estrogen receptor modulator, Selective estrogen receptor α inhibitor, PKCβ inhibitor
doxorubicin hydrochloride + Z-endoxifen
406
ICAM-1-targeted CAR-T immunotherapy
AIC100
407
MUC1-targeted CAR-T immunotherapy
P-MUC1C-ALLO1
408
B7-H4-targeted antibody-drug conjugate, Microtubule inhibitor
SGN-B7H4V
409
Retinoid X receptor agonist, HER2 inhibitor, HER4 inhibitor, EGFR inhibitor
neratinib + IRX4204
410
Retinoid X receptor agonist, HER2 inhibitor
tucatinib + IRX4204
trastuzumab + IRX4204
411
Retinoid X receptor agonist
IRX4204
412
CDK19 inhibitor, CDK4 inhibitor, CDK6 inhibitor, CDK8 inhibitor
palbociclib + Senexin B
palbociclib + SNX-631
413
CDK4 inhibitor, CDK6 inhibitor, Serine protease inhibitor, TMPRSS2 inhibitor
palbociclib + nafamostat
414
Serine protease inhibitor, TMPRSS2 inhibitor
nafamostat
415
Bcr-abl tyrosine kinase inhibitor, HER2-targeted antibody-drug conjugate, Src kinase inhibitor, c-KIT inhibitor, Microtubule inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib + ado-trastuzumab emtansine
416
PI3K inhibitor, PARP inhibitor, FAK inhibitor, AKT inhibitor
talazoparib + LY294002
417
β-catenin inhibitor, Microtubule stabilizer, Tubulin polymerization promoter, Alkylating agent, CBP inhibitor, Microtubule inhibitor
docetaxel + cyclophosphamide + eribulin mesylate
418
CDK4 inhibitor, Sonic hedgehog inhibitor, Stem cell inhibitor, Apoptosis stimulant, CDK6 inhibitor
palbociclib + GZ17-6.02
419
HDAC inhibitor, XPO1 inhibitor, MAPK inhibitor, HDAC10 inhibitor, HDAC1 inhibitor, PI3K inhibitor, HDAC2 inhibitor, AKT inhibitor, HDAC3 inhibitor
selinexor + chidamide
420
Topoisomerase II inhibitor, DNMT inhibitor
doxorubicin hydrochloride + decitabine
421
MCL1 inhibitor, BET inhibitor
JQ-1 + S63845
422
ERK2 inhibitor, ERK1 inhibitor
BVD-523
423
RSK inhibitor
PMD-026
424
Immunostimulant, Free radical stimulant, Oxidative stress enhancer
SM-88
425
PARP1 inhibitor, HER2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
fam-trastuzumab deruxtecan-nxki + AZD5305
426
HER2-targeted antibody-drug conjugate, Microtubule inhibitor, PARP inhibitor
ado-trastuzumab emtansine + talazoparib
427
HER2 inhibitor, PARP inhibitor
trastuzumab + talazoparib
428
Tubulin polymerization promoter, DNA synthesis inhibitor, Bcl2 inhibitor
cisplatin + paclitaxel
429
HER2 inhibitor, WEE1 inhibitor
trastuzumab + ZN-c3
430
Selective estrogen receptor degrader, WEE1 inhibitor
ZN-c3 + ZN-c5
431
CDK4 inhibitor, CDK6 inhibitor, WEE1 inhibitor
palbociclib + ZN-c3
432
YES1 inhibitor, Src kinase inhibitor
NXP900
433
HER2-targeted antibody-drug conjugate, STING agonist
XMT-2056
434
CYP51A1 inhibitor
itraconazole
435
TGM2 inhibitor
MD102
436
STAT3 inhibitor
BP1003
437
PKC inhibitor
AEB071
438
Bcr-abl tyrosine kinase inhibitor, HER2 inhibitor, HER4 inhibitor, EGFR inhibitor, Src kinase inhibitor, c-KIT inhibitor, PDGFR β antagonist, EphA2 receptor antagonist
dasatinib + neratinib
439
mTOR inhibitor, HER2-targeted antibody-drug conjugate, Microtubule inhibitor
everolimus + ado-trastuzumab emtansine
MK-8776
LY 2603618
440
Chk1 inhibitor
CHIR-124
PD-407824
PF-00477736
441
LATS kinase inhibitor
VT02956
442
MCL1 inhibitor
S63845
443
DOT1L inhibitor
EPZ-5676
444
MYC inhibitor
MYCi975
445
CDK9 degrader
THAL-SNS-032
446
Androgen receptor inhibitor, ALK inhibitor
enzalutamide capsule + ceritinib
447
USP8 inhibitor
DC-U4106
448
Reactive oxygen species stimulant, Apoptosis stimulant, HSP70 stimulant
STA-4783
449
Steroid receptor inhibitor, Estrogen receptor modulator
SR16157
450
Src kinase inhibitor, FAK inhibitor
AZD0530
451
PD-L1 inhibitor, DNA synthesis inhibitor, DNA cross linking agent
PD-L1 inhibitor + oxaliplatin
452
HER2 degrader
CH7C4
453
USP1 inhibitor, PARP inhibitor
olaparib + RG6614
454
HER2-targeted antibody-drug conjugate, Microtubule inhibitor, CD47 inhibitor
disitamab vedotin + ABBV-IMAB-TJC4
455
PD-L1 inhibitor, NK cell stimulant
avelumab + CYNK-101
456
KU70/KU80 inhibitor, PARP1 inhibitor, MRN complex inhibitor
VIO-01
457
Androgen receptor inhibitor, CDK7 inhibitor
enzalutamide capsule + KRLS-017
458
ATR inhibitor, TROP-2-targeted antibody-drug conjugate, Topoisomerase I inhibitor
sacituzumab govitecan-hziy + BAY 1895344
459
CDK19 inhibitor, mTOR inhibitor, CDK8 inhibitor
everolimus + SNX-631
460
PIK3CA inhibitor, pan-NOS inhibitor
alpelisib + L-NMMA
461
PD-L1 inhibitor, HER2 inhibitor, PD1 inhibitor
trastuzumab + BMS-202
462
ATR inhibitor, HER2-targeted antibody-drug conjugate, PARP inhibitor, Topoisomerase I inhibitor
olaparib + fam-trastuzumab deruxtecan-nxki + BAY 1895344
acalabrutinib
463
BTK inhibitor
zanubrutinib
ibrutinib
464
KU70/KU80 inhibitor, PARP1 inhibitor, MRN complex inhibitor, PARP inhibitor
olaparib + VIO-01
465
CXCR2 antagonist
SB225002
466
Selective estrogen receptor activator, Cell death stimulant, Unfolded protein response activator
TEQ103
467
β-tubulin inhibitor, α-tubulin inhibitor
VERU-111
468
PRMT5 inhibitor
GSK3326595
469
B7-H4-targeted antibody-drug conjugate, Topoisomerase I inhibitor
AZD8205
470
HER2 inhibitor, CD47 inhibitor, HER2 dimerization inhibitor
pertuzumab + D3L-001
471
MUC1-targeted antibody-drug conjugate, HER3-targeted antibody-drug conjugate, Topoisomerase I inhibitor
DM002
472
γδ TCR modulator, EGFR inhibitor
ACE2016
473
ATR inhibitor, HER3-targeted antibody-drug conjugate, Topoisomerase I inhibitor
U3-1402 + BAY 1895344
474
DDX3 inhibitor, PARP inhibitor
PARP inhibitor + RK-33
No biomarker
HER-2 positive
HER-2 negative
HER-2 amplification
HER-2 underexpression
HER-2 overexpression
HER-2 mutation
HER-2 expression
HER-2 L755S
HER-2 S310F
HER-2 778insGSP
HER-2 exon 19 deletion
HER-2 exon 20 insertion
HER-2 L755P
HER-2 V777L
HER-2 mutation + HER-2 T798I
HER-2 A1170P
HER-2 elevation
HER-2 I655V
HER-2 D769H
HER-2 D769Y
HER-2 R896C
HER-2 V842I
HER-2 L755_T759del
HER-2 amplification + HER-2 L755S
HER-2 amplification + HER-2 R157W
HER-2 T862A + HER-2 L755S
HER-2 K753E
HER-2 L768S
p95HER2 mutation
HER-2 C634R
HER-2 L869R
HER-2 T798I
HER-2 G309A
HER-2 G778_P780dup
HER-2 T798M
HER-2 K676R
HER-2 V773L
HER-2 755_759del
HER-2 Q680R
HER-2 P780ins
HER-2 R647K
HER-2 R678Q
HR positive
HR negative
ESR1 mutation + HR positive
ER positive + PGR positive
ESR1 wild-type + HR positive
ER positive + PGR negative
HR overexpression
HR positive + ER overexpression
HR positive + APOBEC signature
ER positive + TP53 mutation
ER positive
ESR1 mutation
ER positive + ESR1 mutation
ER rs2234693
ER mutation
ER negative
ER D538G
ER Y537S
ER E380Q
ER Y537N + ER positive
ER Y537S + ER positive
ESR1 rs1801132
ESR1 rs2228480
ER positive + ESR1 mutation + TP53 mutation
ESR1 rs2234693T>C
ER D538G + ER positive
ER F404L
ER E380Q + ER positive
ER L536Q
ESR1 rs9322354
ER Y537C
ER Y537N
ER overexpression
ER amplification
ER-L
ER E380Q + ER F404L
ER underexpression + ER Y537S
ER underexpression
ER T594T
ER D538G + ER F404L
PIK3CA mutation
PIK3CA E542K
PIK3CA Q75E
PIK3CA E545
PIK3CA N345K
PIK3CA N345K + PIK3CA N1044K
PIK3CA K111N
PIK3CA G106_108del
PIK3CA Q546
PIK3CA G1049R
PIK3CA H1047X
PIK3CA E545X
PIK3CA R38C
PIK3CA H1047
PIK3CA M1043I
PIK3CA H1047R
PIK3CA E545K
PIK3CA amplification
PIK3CA wild-type
PIK3CA E542Q
PIK3CA E453K
PIK3CA H1047L
PIK3CA mutation + HR negative
PIK3CA mutation + MSI-L/dMMR
PIK3CA I391M
PIK3CA C420R
PIK3CA exon 20 mutation + HR positive
PIK3CA exon 9 mutation + HR positive
PIK3CA exon 7 mutation + HR positive
PIK3CA mutation + HR positive
PIK3CA E542K + HR positive
HR positive + PIK3CA exon 10 mutation
HR-positive + PIK3CA wild-type
HR positive + PIK3CA H1047R + PIK3CA D350G + ER D538G
ESR1 mutation + PIK3CA mutation + HR positive
PIK3CA amplification + PIK3CA mutation + HR positive
HR positive + PIK3CA H1047R + ER D538G
HR positive + PIK3CA H1047R
BRCA2 mutation
BRCA2 overexpression
BRCA2 5396insC
BRCA2 N255fs + D252fs
PD-L1 expression
PD-L1 underexpression
PD-L1 overexpression
TMB-H + PD-L1 expression
PD-L1 negative
PD-L1 amplification
MSI-H/dMMR + PD-L1 expression
PD-L1 elevation
BRCA2 mutation + HR positive
HR negative + BRCA2 mutation
HR positive + BRCA2 mutation
BRCA2 mutation + ER positive + PGR positive
BRCA1 mutation + HR positive
HR negative + BRCA1 mutation
HR positive + BRCA1 mutation
HR positive + HER-2 negative
ER positive + PGR negative + HER-2 negative
HR positive + HER-2 positive
HER-2 amplification + ER positive + PGR negative
HR positive + HER-2 amplification
HR positive + HER-2 mutation
HR positive + HER-2 underexpression
HR negative + PD-L1 expression
PIK3CA mutation + HR positive + HER-2 negative
BRCA1 mutation
BRCA1 promoter methylation
BRCA1 E1446*
HR positive + PD-L1 expression
BRCA1 307 T> A (L63*)
ER negative + HER-2 positive + PGR positive + PIK3CA mutation
BRCA1 2080delA
BRCA1 R1443*
BRCA1 2080delA + CCNE1 overexpression
BRCA1 3363delGAAA
BRCA1 5396insC
BRCA1 deletion
BRCA1 L1780P
ERBB3 overexpression
ERBB3 expression
ERBB3 positive
ERBB3 G284R
ERBB3 mutation
ERBB3 E952Q
PTEN deletion
PTEN mutation
PTEN K237fs
PTEN-L
PTEN Hypermethylation
PTEN V85
PTEN underexpression
PTEN expression
PTEN rs701848
BRCA wild-type
PIK3CA mutation + ER positive
PIK3CA mutation + ER negative
BRCA1 mutation + BRCA2 mutation
ER positive + ESR1 mutation + PIK3CA mutation
PIK3CA mutation + ER mutation
PIK3CA mutation + ESR1 mutation
ER negative + PIK3CA H1047R
ER positive + PIK3CA H1047R
PIK3CA mutation + ESR1 wild-type
PIK3CA wild-type+ ESR1 wild-type
PIK3CA H1047R + PIK3CA D959N + ER E380Q
FCGR3A 158V
FCGR3A 158F
HRD
FGFR1 amplification
AKT1 mutation
EGFR expression
FGFR2 amplification
EGFR mutation
FGFR2 overexpression
FGFR2 Y375C
AKT1 E17K
FGFR2 fusion
AKT1 amplification
EGFR amplification
FGFR1 overexpression
FGFR1 expression
EGFR overexpression
AKT1 overexpression
FGFR2 mutation
FGFR1 mutation
EGFR positive
AR positive
HER-2 underexpression + ER underexpression
TMB-H
TMB-L
TP53 R209fs*
TP53 mutation
ABCB1 C3435T
TP53 wild-type
AR overexpression
ABCB1 C1236T
ER positive + HER-2 D769H + HER-2 V777L
ABCB1 G1236T + ABCB1 G2677T
TP53 D281E
ABCB1 G2677T
ER positive + HER-2 negative
TP53 expression
AR underexpression
AR negative
AR expression
TP53 R273H
ER negative + HER-2 negative
TP53 R175H
RAB5A expression
INPP4b deletion
MDM2 mutation
PD-1 overexpression
ATM mutation
HSD17B2 overexpression
FRS2 mutation
HIF1A overexpression
CDKN2A mutation
BACH1 overexpression
BRCA1 mutation + HER-2 negative
BRCA2 mutation + HER-2 negative
ACTA2 elevation
miR-21 overexpression
IGFBP7 overexpression
NES expression
AR positive + ER positive
MYBL2 overexpression
ADRB2 overexpression
PD-L1 overexpression + ER positive
BRCA mutation
CDKN2B mutation
PRKCA mutation
FGFR1 overexpression + HR positive
BRAF V600E
FGFR1 amplification + HR positive
PGR positive
PGR expression
CD8 positive
RB1 mutation + HR positive
PGR overexpression
RB1 mutation
KDR overexpression
BRAF G469E
CD8-H
RB1 expression
KDR V297I
KDR rs1870377
CD8 overexpression
RB1 deletion
RB1 overexpression
BRAF T1799A
CDKN2A deletion
MDM2 amplification
RB1 negative
CDKN2A overexpression
PGR negative
BRAF mutation
ACTA2 overexpression
NTRK1 fusion
MSI-H/dMMR
AKT1 E17K + HR positive
TOP2A amplification
EZH2 A490T
CDK12 amplification
TOP2A deletion
FGFR3 overexpression
NRG1 fusion
NF2 K159fs*16
NF2 mutation
CCR5 expression
AKT1 mutation + ER negative
AKT1 mutation + ER positive
CXCR4 positive
ER positive + ESR1 mutation + CCND1 amplification
ER positive + ESR1 mutation + FGFR1 amplification
RET fusion
BARD1 T351T
CCR5 positive
YAP1 underexpression
ER positive + FGFR1 amplification
ER L536H + ER D538G + CCND1 amplification
AKT1 mutation + HR positive
PARD3 expression
BARD1 mutation
CDK12 mutation
AXL-L
YAP1 overexpression
CXCR4 expression
NRG1 overexpression
HR positive + ERBB3 underexpression
AXL expression
HR positive + ERBB3 overexpression
FGFR3 mutation
RET overexpression
EZH2 rs2302427C>G
VEGFA overexpression
PARD3 overexpression
VEGFA rs833061
CXCR4 overexpression
EZH2 rs201135441C>T
NF2 negative
WSB2 expression
EGF overexpression
PD-L2 overexpression
CTLA4 overexpression
RAD51 underexpression
CHEK2 mutation
SLCO1B1 rs2306283
TA-MUC1 elevation + EGFR expression
IRS1-L
IGFBP5-L
ASXL1 mutation
HRD + BRCA wild-type
TMEM45B overexpression
RRM2 overexpression
BAG1 overexpression
GRB7 overexpression
PTEN deletion + BRCA1 mutation
CD38 expression
PSIP1 expression
ACSL4 overexpression
GPX4 overexpression
CCNE1 mutation
ANXA6 underexpression
COL4A5 mutation
COL22A1 mutation
LLGL2 underexpression + SLC7A5 underexpression
SLC7A5 underexpression
LLGL2 underexpression
PCDHA1 mutation
SDK2 mutation
L1CAM mutation
KPRP mutation
CXCL12-L
CFAP58 mutation
CACNA1S mutation
ARID1A mutation
TMB-H + HER-2 positive
MMP11 overexpression
PTEN deletion + ER positive
KRAS mutation
CCNA2 overexpression
FOXP3 overexpression
CD4 overexpression
FCRL1 overexpression
KDM1A expression
IRF8 overexpression + ER negative
KMT2B mutation
KIR3DL2 mutation
MUC16 mutation
TUBB3 deletion
RRM1 deletion
LRRC3B hypomethylation
High HDAC6 score + HR positive
IL6 elevation
TNFA elevation
IL18 elevation
CCNE2 overexpression + PIK3CA mutation + ER positive
TFF3 overexpression + ER positive
TFF1 overexpression + ER positive
MYC mutation + ER positive
BRCA2 mutation + ER positive
miR-142 overexpression
MCM10 overexpression
VHL mutation
RBPMS expression
UNC13D mutation
SLBP expression
miR-621 overexpression
ADAMTS3 mutation
WNT7A mutation
BPIFB2 mutation
MSI2 overexpression
FOXA1 expression + ER positive
CAV1 overexpression + CAV2 overexpression
KLF4 overexpression
PRMT5 overexpression
FSIP1 overexpression
MYC expression
BLM mutation
NOTCH3 expression
NOTCH3 expression + ER positive + PGR positive
CCND1 mutation + HR positive
CDKN1B mutation + HR positive
CDK4 mutation + HR positive
CCND2 mutation + HR positive
FRS2 amplification + MDM2 amplification
HR positive + TNFRSF11A overexpression
MAF1 overexpression
miR-221 underexpression
miR-125b-2 underexpression
RAD51 overexpression + HR positive
MUC1 elevation
WBP2 overexpression
CCNB2 expression
HR positive + AR positive
CCDC69 overexpression
IGHG1 overexpression
DNMT3A mutation
AKT2 expression
FGFR4 overexpression
SIRT3 expression
ATR mutation
MSH6 mutation
KIM1 overexpression
EMSY mutation
PARP10 mutation
PPM1D mutation
ATRX mutation
FGF3 amplification
FGF amplification
FANCA mutation
PALB2 mutation
ZNF689 underexpression
RAD21 mutation
CDX-2 expression
HER-2 amplification + EGFR-ZNF880 fusion + EGFR E114K
TGFBI promoter hypermethylation
PD-L1 expression + CD68 positive
MMP17 expression + EGFR expression + RB1 expression
BRCA1 mutation + HER-2 negative + ER positive + PGR positive
STK11 F354L
ETV6-NTRK3 fusion
EML4-ALK fusion
FOXD1 expression
PIK3CA H1047R + PIK3C2B amplification
CCNE1 overexpression + PIK3CA muattion + ER positive
HR positive + BRCA positive
POLE E790Q + ERBB2 amplification + TMB-H
PTEN mutation + STK11 mutation
AKT1 mutation + mTOR mutation
SEMA7A expression
ATM expression + ATM T2333fs* + EGFR negative
PIK3CA H1047R + HER-2 amplification
MTOR mutation + HR positive
BRCA1 mutation + RAD51B deletion
ALK fusion
HR positive + TMB-L
MSI-H/dMMR + TMB-H
PIK3R1 EY451delinsD
POLE mutation + PD-L1 negative + TMB-H
BAP1 R300Gfs*6 + PD-L1 expression
BAP1 deletion + TMB-L + PD-L1 expression
STRN-ALK fusion
SLC3A2-NRG1 fusion
ETV6-NTRK3 fusion + CRTC3-NTRK3 fusion
HR positive + BRAF V600E
CCDC6-RET fusion
ER positive + MLH1 1835del3 + MSI-H/dMMR + TMB-H
TK1 elevation
NOS2 underexpression
ER positive + FGFR3 amplification
LMNA-NTRK1 fusion
CD47 overexpression
MLL2 mutation
FGF4 amplification + ER positive
PTCH1 mutation
NEFH mutation
USH2A mutation
TYMS overexpression + HR positive
FGF3 amplification + ER positive
EGFR mutation + ER positive
FGF19 amplification + ER positive
TLE3 expression
HMGB1 positive
BIN3 expression
CTDSP1 expression
FTO expression
EPRS1 expression
GPNMB overexpression
GATA3 mutation
APOBEC3B deletion
RAD51D mutation
SORT1 expression
FANCL mutation
PPP2R2A mutation
RAD51B mutation
RAD51C mutation
RAD54L mutation
BRIP1 mutation
CHEK1 mutation
BCL2 positive
NTRK2 fusion
NTRK3 fusion
PTEN mutation + HR positive
SEMA7A overexpression
MUC1 expression
CCNE1 expression
MYC amplification
miR-125b-2 expression
ARID1A deletion
CCNE1 overexpression
HR positive + TMB-H
CCNE1 amplification
MYC overexpression
MYC mutation
RAD21 amplification
PIK3R1 mutation
CD47 positive
SORT1 positive
FGF3 mutation
HR positive + CCND1 amplification
MYC underexpression
HER-2 V777L + PIK3CA H1047R
PIK3CA mutation + HER-2 amplification
HMGB1 underexpression
miR-221 expression
HR positive + PTEN deletion
High ALC
Low NLR
DDR
TROP2 overexpression
Rbsig overexpression
AR-regulated gene expression pathway signature
DDR signature score
Low PLR
TOP1 deletion
14-gene IGG signature overexpression
GeparSixto immune signature
6-gene WNT pathway signature
76-gene signature
MAF1 expression
MHC-II expression
Choline elevation
CDYL2 overexpression
KLF8 overexpression
FOXA1 mutation
BRCA1 mutation + TP53 mutation
NF1 deletion
HR negative + EGFR amplification
CCDC170 overexpression
AFAP1-AS1 overexpression
PPP2R2B underexpression
PPP3CA expression
PIK3CA mutation + PTEN mutation
HPGD underexpression
ADAM9 overexpression
PTPN12 deletion
NOTCH2 mutation
FOXA1 overexpression
ANXA1 overexpression
CCL2 elevation
LIFR expression
CACNA1D E953D
HDAC5 deletion
IGF1R amplification
TENM4-NRG1 fusion
BOP1 overexpression
CCND1 overexpression
ABCC4 overexpression
CD276 overexpression
CDK2 overexpression
CEACAM6 positive + HER-2 positive
MIA underexpression
KRT5 underexpression
CDH3 underexpression
KRT17 underexpression
SFRP1 underexpression
CXXC5 overexpression
GPR160 overexpression
MLPH overexpression
CASP9 mutation
KRT14 underexpression
ABCC2 overexpression
miR-503-5p overexpression
ABCB4 overexpression
TET2 deletion + DNMT3A mutation
miR-34a expression
ABCG2 overexpression
TUSC7 overexpression
NSD3 overexpression
CCND1 amplification
SPP1 elevation
SPP1 mutation
miR-210 overexpression
TLS gene signature
CD36 overexpression
lncRNA DILA1 overexpression
RET fusion + TP53 mutation
miR-1246 overexpression
CHID1 overexpression
AGR3 expression
ICAM1 overexpression
EPCAM positive + CD44 positive + CD24 negative
VTCN1 underexpression
EPCAM positive + CD44 positive + CD24-L
IGF1 rs2016347
KRAS mutation + CDK9 overexpression + HR positive
ERBB4 H809G + ER positive
SMARCB1 mutation
ANXA1 expression
ZNF649-AS1 overexpression
High MLR
High NLR
LDH elevation
SH3BGRL overexpression
RBM38 overexpression
NF1 mutation
AKR1C3 overexpression
AKR1C2 overexpression
AKR1C1 overexpression
YES1 amplification
SEMA6D underexpression
SLC9A2 overexpression
EPCAM expression
ERBB4 expression
CDH1 deletion
CDH1 mutation
MDM4 mutation
FBXW7 underexpression
NPY1R underexpression
CCAT2 overexpression
DLGAP1-AS1 overexpression
DDX11-AS1 overexpression
USP18 overexpression
SPRED2 deletion
miR-101-5p overexpression
PIK3CA mutation + PTEN underexpression
MMP1 hypomethylation
MMP1 overexpression
HR positive + CCNE1 overexpression
TROP2 expression
HR positive + PLK1 overexpression
SOX9 expression
CD73 elevation
BIRC5 overexpression
CTSD positive + ER positive
High PLR
AGR2 overexpression
HGF amplification
ADRM1 overexpression
MET amplification
PTPN2 amplification
STAT6 deletion + HER-2 overexpression
HDC overexpression + HR positive
TNFRSF1A overexpression + HR positive
miR-155 expression
TGM2 overexpression
BCL6 overexpression
IL21R overexpression
LIG1 deletion
STAT3 expression
HR positive + TP53 mutation
PRO-C3 elevation
PC3X elevation
TP53 wild-type + ER positive
GJA1 expression
CD24 expression
NCOR2 overexpression
ERCC1 negative
ERCC1 overexpression
XRCC1 overexpression
CDKN2C mutation
ER positive + CDK6 overexpression
BCL11B mutation
FER overexpression
LZTS1 overexpression
MCL1 overexpression + HER-2 amplification
HR positive + BRCA2 mutation + PALB2 mutation
ALDH1A1 positive
CHD4 mutation
HR positive + BRCA1 mutation + PALB2 mutation
35-gene signature
MLH1 mutation
HER-2 amplification + AXL expression
SMO mutation
MUC4 expression
SPARC overexpression
THBS1 overexpression
SOX9 overexpression
KIF11 overexpression
RUNX3 underexpression
miR-638 overexpression
HLA-E mutation
MCL1 amplification
HNRNPD overexpression
H3F3C mutation
FGF23 mutation
SNHG16 mutation
MPZL3 overexpression
CDK4 overexpression
CYP2D6 deletion
GNAS mutation
BCL2L1 mutation
LAG3 mutation
CCND2 mutation
LINC00667 overexpression
SESN1 mutation
RFC3 overexpression + ER positive
MLH3 overexpression + HR positive
TROP2 positive
PCNA overexpression + HR positive
CETN2 overexpression + MLH3 overexpression + PCNA overexpression + HR positive
CETN2 overexpression + HR positive
TNFRSF1B overexpression
GSTP1 overexpression
IL6R overexpression
TCEAL9 overexpression
SAMHD1 expression
IL10 overexpression
DLD overexpression
LCN2 overexpression
SAA2 overexpression
SAA1 overexpression
KLK7 overexpression
IL19 overexpression
ACAT1 overexpression
NDUFA4L2 overexpression
PLK1 overexpression
MIR497HG deletion
ANIB1 overexpression
NOTCH4 expression
NOTCH1 expression + NOTCH4 expression
NOTCH1 expression
CCL20 overexpression
HR positive + MYC mutation
HR positive + MYC amplification
HR positive + RB1 mutation
APBB1 expression
NODAL overexpression
SALL4 overexpression
TRIM3 overexpression
BRCA wild-type + TP53 mutation
AGR2 elevation
SOX2 overexpression
KMT2D mutation
MELTF overexpression
ERBB3 expression + MUC1 expression
PTPRT overexpression
PTK7 expression + TROP2 expression
RAD50 deletion
TSC2 C1450G
BRCA2 mutation + RB1 deletion
BRCA1 mutation + RB1 deletion
TP53 R280K + BRCA wild-type
TNC overexpression
DCN overexpression
CPA3 overexpression
HNRNPAB overexpression
SLC39A6 overexpression
EGFR overexpression + KRAS 13D
MAPT overexpression
MERTK expression
GSTP1 rs1138272
TMEM225B rs10273424
NECTIN4 overexpression
IGF1R overexpression
GSPT1 deletion
miR-98-5p underexpression
PRLR underexpression
LAMP1 expression
GH1 overexpression
SLC39A6 expression
VTCN1 expression
ROR1 expression
TXNIP underexpression
TPBG overexpression
LAMTOR5 overexpression
MTOR A2034V
CDK6 overexpression
KRAS mutation + HR positive
RSF1 amplification
MYC amplification + HER-2 amplification
NCAPG overexpression
AURKA overexpression
GSK3B overexpression
APC mutation
CSMD1 overexpression
DUSP6 expression
EIF4EBP1 overexpression
ZNF268 overexpression
AKT3 expression
miR-186 overexpression
SMARCA4 mutation
PKD1 mutation
HR positive + BRIP1 amplification
MALAT1 overexpression
PIK3CA mutation + PTEN deletion
HER-2 amplification + PTEN deletion
MTOR M2327I
MTOR F2108L
HR positive + AURKA mutation
ER-CCDC170 fusion
RBBP8 E281
CUL7 overexpression
NOTCH1 mutation
PARP1 overexpression
DEDD overexpression
PSMD4 amplification
TIMP1 overexpression
SF3B1 K700E
SF3B1 K666Q
SF3B1 K666E
TIAM1 overexpression
CD276 expression
STAT6 underexpression
FGFR mutation
HAVCR2 deletion
ST14 expression
miR-155 overexpression
FERMT1 expression
MFI2 expression
PAK4 deletion
HR positive + AURKA amplification
PTK7 expression
CASP8 overexpression
CASP9 underexpression
GFRA1 overexpression
CREBBP deletion
CREBBP mutation
FOXC1 expression
HR positive + RAD51C amplification
PAX2 promoter methylation
SORL1 deletion
miR-381 underexpression
CCND1-H
MAP3K6 overexpression
GNRHR expression
NQO1 positive
ABCC5 expression
HASPIN expression
MAP3K1 mutation
IGF2 overexpression
SETDB1 overexpression